SE419440B - SET TO MAKE SOMATOSTATIN ANALOGS - Google Patents

SET TO MAKE SOMATOSTATIN ANALOGS

Info

Publication number
SE419440B
SE419440B SE7608300A SE7608300A SE419440B SE 419440 B SE419440 B SE 419440B SE 7608300 A SE7608300 A SE 7608300A SE 7608300 A SE7608300 A SE 7608300A SE 419440 B SE419440 B SE 419440B
Authority
SE
Sweden
Prior art keywords
somatostatin analogs
make
make somatostatin
analogs
somatostatin
Prior art date
Application number
SE7608300A
Other languages
Swedish (sv)
Other versions
SE7608300L (en
Inventor
D F Veber
F W Holly
R G Strachan
W J Paleveda
R F Nutt
R F Hirschmann
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of SE7608300L publication Critical patent/SE7608300L/en
Publication of SE419440B publication Critical patent/SE419440B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/655—Somatostatins
    • C07K14/6555—Somatostatins at least 1 amino acid in D-form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
    • C07K5/1013—Tetrapeptides with the first amino acid being neutral and aliphatic the side chain containing O or S as heteroatoms, e.g. Cys, Ser
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SE7608300A 1975-08-08 1976-07-21 SET TO MAKE SOMATOSTATIN ANALOGS SE419440B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US60306775A 1975-08-08 1975-08-08
US68000576A 1976-04-23 1976-04-23

Publications (2)

Publication Number Publication Date
SE7608300L SE7608300L (en) 1977-02-09
SE419440B true SE419440B (en) 1981-08-03

Family

ID=27084324

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7608300A SE419440B (en) 1975-08-08 1976-07-21 SET TO MAKE SOMATOSTATIN ANALOGS

Country Status (8)

Country Link
JP (1) JPS5219659A (en)
CH (1) CH626328A5 (en)
DE (1) DE2635558A1 (en)
DK (1) DK328876A (en)
FR (1) FR2320109A1 (en)
GB (1) GB1502573A (en)
NL (1) NL7607987A (en)
SE (1) SE419440B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4115554A (en) * 1977-08-29 1978-09-19 Merck & Co., Inc. Somatostatin analogs
LU78191A1 (en) * 1977-09-28 1979-05-25 Ciba Geigy Ag METHOD FOR PRODUCING NEW CYCLOPEPTIDES
US4139526A (en) * 1977-12-01 1979-02-13 Merck & Co., Inc. Somatostatin analogs
US4140767A (en) * 1977-12-01 1979-02-20 Merck & Co., Inc. Somatostatin analogs
JPS5819669B2 (en) * 1978-10-28 1983-04-19 白井松新薬株式会社 Novel bioactive peptide compounds and their production methods
US4316890A (en) * 1979-03-16 1982-02-23 Ciba-Geigy Corporation Peptides and processes for the manufacture thereof
US4244947A (en) * 1979-08-13 1981-01-13 Ayerst Mckenna And Harrison Inc. Carba decapeptide derivatives of [TYR6 ]-somatostatin
HU198626B (en) * 1986-05-27 1989-11-28 Sandoz Ag Process for producing pharmaceutical compositions comprising somatostatin analogues as active ingredient
US5443815A (en) * 1991-11-27 1995-08-22 Diatech, Inc. Technetium-99m labeled peptides for imaging
AU664855B2 (en) * 1991-08-09 1995-12-07 Winfried Kolbeck Lanthionine bridged peptides
US5716596A (en) * 1992-06-23 1998-02-10 Diatide, Inc. Radioactively labeled somatostatin-derived peptides for imaging and therapeutic uses
US6017512A (en) * 1992-06-23 2000-01-25 Diatide, Inc. Radiolabeled peptides
US5620675A (en) 1992-06-23 1997-04-15 Diatech, Inc. Radioactive peptides
CN1378450A (en) * 1999-09-08 2002-11-06 斯隆-凯特林癌症研究院 Novel class of cytodifferentiating agents and histone deactylase inhibitors, and methods of use thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL6509712A (en) * 1964-07-27 1966-01-28
DE2460469A1 (en) * 1974-12-20 1976-07-01 Hoechst Ag Cyclic peptides inhibiting hormone release - prepd by cyclisation of linear undecapeptides contg a terminal omega- amino acid gp

Also Published As

Publication number Publication date
CH626328A5 (en) 1981-11-13
DK328876A (en) 1977-02-09
FR2320109B1 (en) 1979-05-25
JPS5219659A (en) 1977-02-15
GB1502573A (en) 1978-03-01
DE2635558A1 (en) 1977-02-17
FR2320109A1 (en) 1977-03-04
SE7608300L (en) 1977-02-09
NL7607987A (en) 1977-02-10

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