RU94031479A - Новое применение производных аминокислот, способ лечения, фармацевтическая композиция - Google Patents

Новое применение производных аминокислот, способ лечения, фармацевтическая композиция

Info

Publication number
RU94031479A
RU94031479A RU94031479/14A RU94031479A RU94031479A RU 94031479 A RU94031479 A RU 94031479A RU 94031479/14 A RU94031479/14 A RU 94031479/14A RU 94031479 A RU94031479 A RU 94031479A RU 94031479 A RU94031479 A RU 94031479A
Authority
RU
Russia
Prior art keywords
amino acid
pharmaceutical composition
treatment method
acid derivatives
new application
Prior art date
Application number
RU94031479/14A
Other languages
English (en)
Inventor
Танака Еко
Jp]
Кагаяма Акира
Хата Такехиса
Original Assignee
Фудзисава Фармасьютикал Ко.
Фудзисава Фармасьютикал Ко., Лтд.
Лтд. (Jp)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Фудзисава Фармасьютикал Ко., Фудзисава Фармасьютикал Ко., Лтд., Лтд. (Jp) filed Critical Фудзисава Фармасьютикал Ко.
Publication of RU94031479A publication Critical patent/RU94031479A/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/55Protease inhibitors
    • A61K38/553Renin inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Ophthalmology & Optometry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Изобретение относится к применению соединений формулы, приведенной в описании, или их фармацевтически приемлемых солей для лечения глаукомы или снижения и/или регулирования внутриглазного давления.

Claims (1)

  1. Изобретение относится к применению соединений формулы, приведенной в описании, или их фармацевтически приемлемых солей для лечения глаукомы или снижения и/или регулирования внутриглазного давления.
RU94031479/14A 1991-12-20 1992-12-18 Новое применение производных аминокислот, способ лечения, фармацевтическая композиция RU94031479A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9127041.3 1991-12-20
GB919127041A GB9127041D0 (en) 1991-12-20 1991-12-20 New use

Publications (1)

Publication Number Publication Date
RU94031479A true RU94031479A (ru) 1996-10-20

Family

ID=10706572

Family Applications (1)

Application Number Title Priority Date Filing Date
RU94031479/14A RU94031479A (ru) 1991-12-20 1992-12-18 Новое применение производных аминокислот, способ лечения, фармацевтическая композиция

Country Status (11)

Country Link
EP (1) EP0617622A1 (ru)
JP (1) JPH07506807A (ru)
KR (1) KR940703665A (ru)
AU (1) AU661748B2 (ru)
CA (1) CA2126211A1 (ru)
GB (1) GB9127041D0 (ru)
HU (2) HUT68175A (ru)
MX (1) MX9207429A (ru)
RU (1) RU94031479A (ru)
WO (1) WO1993012796A1 (ru)
ZA (1) ZA929738B (ru)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1994025062A1 (en) * 1993-04-28 1994-11-10 Fujisawa Pharmaceutical Co., Ltd. Oral pharmaceutical compositions containing renin inhibitors
AU2001268490A1 (en) 2000-06-15 2001-12-24 Pharmacia Corporation Dihydrostilbene alkanoic acid derivatives useful as vitronectin antagonists
US6476046B1 (en) 2000-12-04 2002-11-05 Sepracor, Inc. Diazabicyclo[4.3.0]nonanes, and methods of use thereof
AR040126A1 (es) 2002-05-29 2005-03-16 Glaxo Group Ltd Compuesto de fenilsulfonilo, composicion farmaceutica que lo comprende y su uso para la elaboracion de un medicamento
CA2839703A1 (en) 2011-06-24 2012-12-27 Amgen Inc. Trpm8 antagonists and their use in treatments
MY157429A (en) 2011-06-24 2016-06-15 Amgen Inc Trpm8 antagonists and their use in treatments
US8952009B2 (en) 2012-08-06 2015-02-10 Amgen Inc. Chroman derivatives as TRPM8 inhibitors
CN116096714A (zh) 2020-06-10 2023-05-09 安力高医药股份有限公司 用于治疗冠状病毒、小核糖核酸病毒和诺罗病毒感染的抗病毒化合物
IL309732A (en) 2021-07-09 2024-02-01 Aligos Therapeutics Inc Antiviral compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4906613A (en) * 1985-11-05 1990-03-06 Schering Corporation Antiglaucoma compositions and methods
US4921855A (en) * 1987-06-22 1990-05-01 Fujisawa Pharmaceutical Co., Ltd. New Histidyl amino acid derivatives, and pharmaceutical composition comprising the same
US4927807A (en) * 1987-10-06 1990-05-22 Abbott Laboratories Glaucoma treatment
US5151513A (en) * 1988-04-29 1992-09-29 E. R. Squibb & Sons, Inc. N-heterocyclic alcohol derivatives
IL99389A0 (en) * 1990-09-17 1992-08-18 Fujisawa Pharmaceutical Co Amino acid derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same

Also Published As

Publication number Publication date
KR940703665A (ko) 1994-12-12
WO1993012796A1 (en) 1993-07-08
AU3171293A (en) 1993-07-28
AU661748B2 (en) 1995-08-03
HUT68175A (en) 1995-05-29
EP0617622A1 (en) 1994-10-05
HU211939A9 (en) 1996-01-29
MX9207429A (es) 1993-06-01
CA2126211A1 (en) 1993-07-08
GB9127041D0 (en) 1992-02-19
ZA929738B (en) 1993-06-17
JPH07506807A (ja) 1995-07-27
HU9401833D0 (en) 1994-09-28

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