RU92016595A - SUBSTITUTED THIAZOLYL AND SUBSTITUTED PYRIDINYL DERIVATIVES, PHARMACEUTICAL COMPOSITION AND METHOD FOR PRODUCING THEM - Google Patents

SUBSTITUTED THIAZOLYL AND SUBSTITUTED PYRIDINYL DERIVATIVES, PHARMACEUTICAL COMPOSITION AND METHOD FOR PRODUCING THEM

Info

Publication number
RU92016595A
RU92016595A RU92016595/04A RU92016595A RU92016595A RU 92016595 A RU92016595 A RU 92016595A RU 92016595/04 A RU92016595/04 A RU 92016595/04A RU 92016595 A RU92016595 A RU 92016595A RU 92016595 A RU92016595 A RU 92016595A
Authority
RU
Russia
Prior art keywords
substituted
producing
pharmaceutical composition
thiazolyl
pyridinyl derivatives
Prior art date
Application number
RU92016595/04A
Other languages
Russian (ru)
Other versions
RU2067978C1 (en
Inventor
Эдуард Жанссен Франс
Мариа Соммен Франсуа
Станислас Марселла Диел Гастон
Original Assignee
Жансен Фармасетика Н.В.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Жансен Фармасетика Н.В. filed Critical Жансен Фармасетика Н.В.
Priority claimed from PCT/EP1991/001292 external-priority patent/WO1992001697A1/en
Application granted granted Critical
Publication of RU2067978C1 publication Critical patent/RU2067978C1/en
Publication of RU92016595A publication Critical patent/RU92016595A/en

Links

Claims (1)

Замещенные тиазолиловые и замещенные пиридиниловые производные и их фармацевтически приемлемые кислые аддитивные соли и стереохимические изомеры.Substituted thiazolyl and substituted pyridinyl derivatives and their pharmaceutically acceptable acid addition salts and stereochemical isomers.
RU9192016595A 1990-07-19 1991-07-09 Substituted thiazolyl and substituted pyridinyl derivatives or their pharmaceutically acceptable acid additive salts, method for their production and composition possessing antiallergic activity RU2067978C1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US55432590A 1990-07-19 1990-07-19
US554325 1990-07-19
PCT/EP1991/001292 WO1992001697A1 (en) 1990-07-19 1991-07-09 Novel substituted thiazolyl and substituted pyridinyl derivatives

Publications (2)

Publication Number Publication Date
RU2067978C1 RU2067978C1 (en) 1996-10-20
RU92016595A true RU92016595A (en) 1996-11-27

Family

ID=24212925

Family Applications (1)

Application Number Title Priority Date Filing Date
RU9192016595A RU2067978C1 (en) 1990-07-19 1991-07-09 Substituted thiazolyl and substituted pyridinyl derivatives or their pharmaceutically acceptable acid additive salts, method for their production and composition possessing antiallergic activity

Country Status (27)

Country Link
EP (1) EP0539420B1 (en)
JP (1) JP3085707B2 (en)
KR (1) KR100206723B1 (en)
CN (1) CN1037770C (en)
AT (1) ATE188477T1 (en)
AU (1) AU646280B2 (en)
CA (1) CA2086546A1 (en)
CZ (1) CZ279903B6 (en)
DE (1) DE69131895T2 (en)
DK (1) DK0539420T3 (en)
ES (1) ES2142802T3 (en)
FI (1) FI102753B1 (en)
GR (1) GR3032999T3 (en)
HU (1) HU221298B1 (en)
IE (1) IE912533A1 (en)
IL (1) IL98865A (en)
MX (1) MX9100307A (en)
NO (1) NO304791B1 (en)
NZ (1) NZ238863A (en)
PH (1) PH31063A (en)
PL (1) PL170580B1 (en)
PT (1) PT98366B (en)
RU (1) RU2067978C1 (en)
SK (1) SK280690B6 (en)
TW (1) TW209217B (en)
WO (1) WO1992001697A1 (en)
ZA (1) ZA915654B (en)

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ES2048109B1 (en) * 1992-07-20 1994-12-16 Espanola Prod Quimicos PROCEDURE FOR THE PREPARATION OF NEW PIPERIDIC DERIVATIVES OF BENCIMIDAZOLE.
US6211199B1 (en) 1995-11-17 2001-04-03 Aventis Pharmaceuticals Inc. Substituted 4-(1H-benzimidazol-2-yl-amino)piperidines useful for the treatment of allergic diseases
US6423704B2 (en) 1995-12-20 2002-07-23 Aventis Pharmaceuticals Inc. Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic diseases
US6194406B1 (en) 1995-12-20 2001-02-27 Aventis Pharmaceuticals Inc. Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic disease
US5922737A (en) * 1996-02-21 1999-07-13 Hoechst Marion Roussel, Inc. Substituted N-methyl-N-(4-(4-(1H-Benzimidazol-2-YL-amino) piperidin-1-YL)-2-(arlyl) butyl) benzamides useful for the treatment of allergic diseases
US5932571A (en) * 1996-02-21 1999-08-03 Hoechst Marion Roussel, Inc. Substituted N-methyl-N-(4-(4-(1H-benzimidazol-2-yl) {1,4}diazepan-1-yl)-2-(aryl) butyl) benzamides useful for the treatment of allergic diseases
US5998439A (en) 1996-02-21 1999-12-07 Hoescht Marion Roussel, Inc. Substituted N-methyl-N-(4-(piperidin-1-yl)-2-(aryl)butyl)benzamides useful for the treatment of allergic diseases
EP1196410B1 (en) 1999-06-28 2004-02-18 Janssen Pharmaceutica N.V. Respiratory syncytial virus replication inhibitors
TR200103804T2 (en) * 1999-06-28 2002-05-21 Janssen Pharmaceutica N.V. Substances that inhibit the replication of the respiratory syncytial virus
PT1196409E (en) * 1999-06-28 2004-06-30 Janssen Pharmaceutica Nv RESPIRATORY SYNCIC VIRUS REPLICATION INHIBITORS
EP1599468B1 (en) 2003-01-14 2007-10-03 Arena Pharmaceuticals, Inc. 1,2,3-trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia
AR045047A1 (en) 2003-07-11 2005-10-12 Arena Pharm Inc ARILO AND HETEROARILO DERIVATIVES TRISUSTITUIDOS AS MODULATORS OF METABOLISM AND PROFILAXIS AND TREATMENT OF DISORDERS RELATED TO THEMSELVES
WO2005113511A1 (en) * 2004-05-12 2005-12-01 Bristol-Myers Squibb Company Urea antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
DOP2006000010A (en) 2005-01-10 2006-07-31 Arena Pharm Inc PROCEDURE TO PREPARE AROMATIC ETERES
EA201390421A1 (en) 2010-09-22 2013-09-30 Арена Фармасьютикалз, Инк. GPR119 RECEPTOR MODULATORS AND TREATMENT OF RELATED DISORDERS
EP3040334A1 (en) * 2014-12-29 2016-07-06 Faes Farma, S.A. New benzimidazole derivatives as antihistamine agents
KR102595163B1 (en) 2015-01-06 2023-10-30 아레나 파마슈티칼스, 인크. Methods for Treating Conditions Associated with the S1P1 Receptor
WO2016209809A1 (en) 2015-06-22 2016-12-29 Arena Pharmaceuticals, Inc. Crystalline l-arginine salt of (r)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclo-penta[b]indol-3-yl)acetic acid(compound1) for use in sipi receptor-associated disorders

Family Cites Families (11)

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US4556660A (en) * 1982-07-12 1985-12-03 Janssen Pharmaceutica N.V. N-(Bicyclic heterocyclyl)-4-piperidinamines
US4634704A (en) * 1983-10-06 1987-01-06 Janssen Pharmaceutica, N.V. Anti-allergic five membered heterocyclic ring containing N-(bicyclic heterocycyl)-4-piperidinamines
US4695569A (en) * 1983-11-30 1987-09-22 Janssen Pharmaceutica N.V. Bicyclic heterocyclyl containing N-(bicyclic heterocyclyl)-4-piperidinamines
US4588722A (en) * 1984-01-09 1986-05-13 Janssen Pharmaceutica N.V. N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives
US4695575A (en) * 1984-11-13 1987-09-22 Janssen Pharmaceutica, N.V. 4-[(bicycle heterocyclyl)-methyl and -hetero]-piperidines
GB8515934D0 (en) * 1985-06-24 1985-07-24 Janssen Pharmaceutica Nv (4-piperidinomethyl and-hetero)purines
US4835161A (en) * 1986-02-03 1989-05-30 Janssen Pharmaceutica N.V. Anti-histaminic compositions containing n-heterocyclyl-4-piperidinamines
DE3701863A1 (en) * 1987-01-23 1988-08-04 Standard Elektrik Lorenz Ag Transmitter for coherent optical communications
US4897401A (en) * 1987-06-19 1990-01-30 Janssen Pharmaceutical N.V. N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives useful in treating allergic diseases
CA1317939C (en) * 1987-07-01 1993-05-18 Janssen Pharmaceutica Naamloze Vennootschap ¬(bicyclic heterocyclyl)methyl and -hetero| substituted hexahydro-1h-azepines and pyrrolidines
GB8900380D0 (en) * 1989-01-09 1989-03-08 Janssen Pharmaceutica Nv 2-aminopyrimidinone derivatives

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