RU92016595A - SUBSTITUTED THIAZOLYL AND SUBSTITUTED PYRIDINYL DERIVATIVES, PHARMACEUTICAL COMPOSITION AND METHOD FOR PRODUCING THEM - Google Patents
SUBSTITUTED THIAZOLYL AND SUBSTITUTED PYRIDINYL DERIVATIVES, PHARMACEUTICAL COMPOSITION AND METHOD FOR PRODUCING THEMInfo
- Publication number
- RU92016595A RU92016595A RU92016595/04A RU92016595A RU92016595A RU 92016595 A RU92016595 A RU 92016595A RU 92016595/04 A RU92016595/04 A RU 92016595/04A RU 92016595 A RU92016595 A RU 92016595A RU 92016595 A RU92016595 A RU 92016595A
- Authority
- RU
- Russia
- Prior art keywords
- substituted
- producing
- pharmaceutical composition
- thiazolyl
- pyridinyl derivatives
- Prior art date
Links
- -1 PYRIDINYL Chemical class 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 239000002253 acid Substances 0.000 claims 1
- 125000004076 pyridyl group Chemical group 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
- 239000011780 sodium chloride Substances 0.000 claims 1
- 125000000335 thiazolyl group Chemical group 0.000 claims 1
Claims (1)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US55432590A | 1990-07-19 | 1990-07-19 | |
US554325 | 1990-07-19 | ||
PCT/EP1991/001292 WO1992001697A1 (en) | 1990-07-19 | 1991-07-09 | Novel substituted thiazolyl and substituted pyridinyl derivatives |
Publications (2)
Publication Number | Publication Date |
---|---|
RU2067978C1 RU2067978C1 (en) | 1996-10-20 |
RU92016595A true RU92016595A (en) | 1996-11-27 |
Family
ID=24212925
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU9192016595A RU2067978C1 (en) | 1990-07-19 | 1991-07-09 | Substituted thiazolyl and substituted pyridinyl derivatives or their pharmaceutically acceptable acid additive salts, method for their production and composition possessing antiallergic activity |
Country Status (27)
Country | Link |
---|---|
EP (1) | EP0539420B1 (en) |
JP (1) | JP3085707B2 (en) |
KR (1) | KR100206723B1 (en) |
CN (1) | CN1037770C (en) |
AT (1) | ATE188477T1 (en) |
AU (1) | AU646280B2 (en) |
CA (1) | CA2086546A1 (en) |
CZ (1) | CZ279903B6 (en) |
DE (1) | DE69131895T2 (en) |
DK (1) | DK0539420T3 (en) |
ES (1) | ES2142802T3 (en) |
FI (1) | FI102753B (en) |
GR (1) | GR3032999T3 (en) |
HU (1) | HU221298B1 (en) |
IE (1) | IE912533A1 (en) |
IL (1) | IL98865A (en) |
MX (1) | MX9100307A (en) |
NO (1) | NO304791B1 (en) |
NZ (1) | NZ238863A (en) |
PH (1) | PH31063A (en) |
PL (1) | PL170580B1 (en) |
PT (1) | PT98366B (en) |
RU (1) | RU2067978C1 (en) |
SK (1) | SK280690B6 (en) |
TW (1) | TW209217B (en) |
WO (1) | WO1992001697A1 (en) |
ZA (1) | ZA915654B (en) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2048109B1 (en) * | 1992-07-20 | 1994-12-16 | Espanola Prod Quimicos | PROCEDURE FOR THE PREPARATION OF NEW PIPERIDIC DERIVATIVES OF BENCIMIDAZOLE. |
US6211199B1 (en) | 1995-11-17 | 2001-04-03 | Aventis Pharmaceuticals Inc. | Substituted 4-(1H-benzimidazol-2-yl-amino)piperidines useful for the treatment of allergic diseases |
US6194406B1 (en) | 1995-12-20 | 2001-02-27 | Aventis Pharmaceuticals Inc. | Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic disease |
US6423704B2 (en) | 1995-12-20 | 2002-07-23 | Aventis Pharmaceuticals Inc. | Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic diseases |
US5932571A (en) * | 1996-02-21 | 1999-08-03 | Hoechst Marion Roussel, Inc. | Substituted N-methyl-N-(4-(4-(1H-benzimidazol-2-yl) {1,4}diazepan-1-yl)-2-(aryl) butyl) benzamides useful for the treatment of allergic diseases |
US5998439A (en) | 1996-02-21 | 1999-12-07 | Hoescht Marion Roussel, Inc. | Substituted N-methyl-N-(4-(piperidin-1-yl)-2-(aryl)butyl)benzamides useful for the treatment of allergic diseases |
US5922737A (en) * | 1996-02-21 | 1999-07-13 | Hoechst Marion Roussel, Inc. | Substituted N-methyl-N-(4-(4-(1H-Benzimidazol-2-YL-amino) piperidin-1-YL)-2-(arlyl) butyl) benzamides useful for the treatment of allergic diseases |
UA74787C2 (en) | 1999-06-28 | 2006-02-15 | Janssen Pharmaceutica Nv | Respiratory syncytial virus replication inhibitors |
PL198021B1 (en) | 1999-06-28 | 2008-05-30 | Janssen Pharmaceutica Nv | Respiratory syncytial virus replication inhibitors |
CZ20014573A3 (en) * | 1999-06-28 | 2002-05-15 | Janssen Pharmaceutica N. V. | Respiratory syncytial virus replication inhibitors |
ATE374766T1 (en) | 2003-01-14 | 2007-10-15 | Arena Pharm Inc | 1,2,3-TRISUBSTITUTED ARYL AND HETEROARYL DERIVATIVES AS MODULATORS OF METABOLISM FOR THE PREVENTION AND TREATMENT OF METABOLISM-RELATED DISEASES SUCH AS DIABETES OR HYPERGLYCEMIA |
AR045047A1 (en) | 2003-07-11 | 2005-10-12 | Arena Pharm Inc | ARILO AND HETEROARILO DERIVATIVES TRISUSTITUIDOS AS MODULATORS OF METABOLISM AND PROFILAXIS AND TREATMENT OF DISORDERS RELATED TO THEMSELVES |
EP1751113B1 (en) * | 2004-05-12 | 2010-03-10 | Brystol-Myers Squibb Company | Urea antagonists of p2y1 receptor useful in the treatment of thrombotic conditions |
DOP2006000010A (en) | 2005-01-10 | 2006-07-31 | Arena Pharm Inc | PROCEDURE TO PREPARE AROMATIC ETERES |
BR112013008100A2 (en) | 2010-09-22 | 2016-08-09 | Arena Pharm Inc | "gpr19 receptor modulators and the treatment of disorders related thereto." |
EP3040334A1 (en) * | 2014-12-29 | 2016-07-06 | Faes Farma, S.A. | New benzimidazole derivatives as antihistamine agents |
US11007175B2 (en) | 2015-01-06 | 2021-05-18 | Arena Pharmaceuticals, Inc. | Methods of treating conditions related to the S1P1 receptor |
NZ738862A (en) | 2015-06-22 | 2023-12-22 | Arena Pharm Inc | Crystalline l-arginine salt of (r)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclo-penta[b]indol-3-yl)acetic acid(compound1) for use in sipi receptor-associated disorders |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4556660A (en) * | 1982-07-12 | 1985-12-03 | Janssen Pharmaceutica N.V. | N-(Bicyclic heterocyclyl)-4-piperidinamines |
US4634704A (en) * | 1983-10-06 | 1987-01-06 | Janssen Pharmaceutica, N.V. | Anti-allergic five membered heterocyclic ring containing N-(bicyclic heterocycyl)-4-piperidinamines |
US4695569A (en) * | 1983-11-30 | 1987-09-22 | Janssen Pharmaceutica N.V. | Bicyclic heterocyclyl containing N-(bicyclic heterocyclyl)-4-piperidinamines |
US4588722A (en) * | 1984-01-09 | 1986-05-13 | Janssen Pharmaceutica N.V. | N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives |
US4695575A (en) * | 1984-11-13 | 1987-09-22 | Janssen Pharmaceutica, N.V. | 4-[(bicycle heterocyclyl)-methyl and -hetero]-piperidines |
GB8515934D0 (en) * | 1985-06-24 | 1985-07-24 | Janssen Pharmaceutica Nv | (4-piperidinomethyl and-hetero)purines |
US4835161A (en) * | 1986-02-03 | 1989-05-30 | Janssen Pharmaceutica N.V. | Anti-histaminic compositions containing n-heterocyclyl-4-piperidinamines |
DE3701863A1 (en) * | 1987-01-23 | 1988-08-04 | Standard Elektrik Lorenz Ag | Transmitter for coherent optical communications |
US4897401A (en) * | 1987-06-19 | 1990-01-30 | Janssen Pharmaceutical N.V. | N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives useful in treating allergic diseases |
CA1317939C (en) * | 1987-07-01 | 1993-05-18 | Janssen Pharmaceutica Naamloze Vennootschap | ¬(bicyclic heterocyclyl)methyl and -hetero| substituted hexahydro-1h-azepines and pyrrolidines |
GB8900380D0 (en) * | 1989-01-09 | 1989-03-08 | Janssen Pharmaceutica Nv | 2-aminopyrimidinone derivatives |
-
1991
- 1991-07-05 NZ NZ238863A patent/NZ238863A/en unknown
- 1991-07-09 RU RU9192016595A patent/RU2067978C1/en not_active IP Right Cessation
- 1991-07-09 HU HU9300096A patent/HU221298B1/en not_active IP Right Cessation
- 1991-07-09 DK DK91912667T patent/DK0539420T3/en active
- 1991-07-09 PL PL91297612A patent/PL170580B1/en not_active IP Right Cessation
- 1991-07-09 AT AT91912667T patent/ATE188477T1/en not_active IP Right Cessation
- 1991-07-09 JP JP03511645A patent/JP3085707B2/en not_active Expired - Fee Related
- 1991-07-09 AU AU82093/91A patent/AU646280B2/en not_active Ceased
- 1991-07-09 DE DE69131895T patent/DE69131895T2/en not_active Expired - Fee Related
- 1991-07-09 WO PCT/EP1991/001292 patent/WO1992001697A1/en active IP Right Grant
- 1991-07-09 ES ES91912667T patent/ES2142802T3/en not_active Expired - Lifetime
- 1991-07-09 CA CA002086546A patent/CA2086546A1/en not_active Abandoned
- 1991-07-09 KR KR1019930700122A patent/KR100206723B1/en not_active IP Right Cessation
- 1991-07-09 EP EP91912667A patent/EP0539420B1/en not_active Expired - Lifetime
- 1991-07-11 PH PH42771A patent/PH31063A/en unknown
- 1991-07-17 IL IL9886591A patent/IL98865A/en not_active IP Right Cessation
- 1991-07-18 IE IE253391A patent/IE912533A1/en not_active Application Discontinuation
- 1991-07-18 ZA ZA915654A patent/ZA915654B/en unknown
- 1991-07-18 SK SK2239-91A patent/SK280690B6/en unknown
- 1991-07-18 PT PT98366A patent/PT98366B/en not_active IP Right Cessation
- 1991-07-18 CZ CS912239A patent/CZ279903B6/en not_active IP Right Cessation
- 1991-07-19 CN CN91104906A patent/CN1037770C/en not_active Expired - Fee Related
- 1991-07-19 MX MX9100307A patent/MX9100307A/en not_active IP Right Cessation
- 1991-08-03 TW TW080106084A patent/TW209217B/zh active
-
1993
- 1993-01-15 NO NO924313A patent/NO304791B1/en unknown
- 1993-01-18 FI FI930199A patent/FI102753B/en active
-
2000
- 2000-03-21 GR GR20000400699T patent/GR3032999T3/en not_active IP Right Cessation
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