RU2564666C2 - Терапевтическое применение 1-[2-(2,4-диметилфенилсульфанил)фенил]пиперазина - Google Patents
Терапевтическое применение 1-[2-(2,4-диметилфенилсульфанил)фенил]пиперазина Download PDFInfo
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- RU2564666C2 RU2564666C2 RU2013112890/15A RU2013112890A RU2564666C2 RU 2564666 C2 RU2564666 C2 RU 2564666C2 RU 2013112890/15 A RU2013112890/15 A RU 2013112890/15A RU 2013112890 A RU2013112890 A RU 2013112890A RU 2564666 C2 RU2564666 C2 RU 2564666C2
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
Landscapes
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- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| Application Number | Priority Date | Filing Date | Title |
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| DKPA201000739 | 2010-08-23 | ||
| DKPA201000739 | 2010-08-23 | ||
| PCT/DK2011/050317 WO2012025123A1 (en) | 2010-08-23 | 2011-08-22 | Therapeutic uses of 1-[2-(2,4-dimethyl-phenylsulfanyl)phenyl]piperazine |
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| Publication Number | Publication Date |
|---|---|
| RU2013112890A RU2013112890A (ru) | 2014-09-27 |
| RU2564666C2 true RU2564666C2 (ru) | 2015-10-10 |
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| Application Number | Title | Priority Date | Filing Date |
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| RU2013112890/15A RU2564666C2 (ru) | 2010-08-23 | 2011-08-22 | Терапевтическое применение 1-[2-(2,4-диметилфенилсульфанил)фенил]пиперазина |
Country Status (32)
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2859008C2 (ru) * | 2020-04-03 | 2026-03-25 | Х. Лундбекк А/С | 1-[2-(2,4-диметилфенилсульфанил)фенил]пиперазин для предупреждения или лечения эмоциональной притупленности |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EA029060B1 (ru) | 2014-01-31 | 2018-02-28 | Эгиш Дьёдьсердьяр Зрт. | Способ получения солей вортиоксетина |
| CN104119299B (zh) * | 2014-08-13 | 2016-08-17 | 北京蓝贝望生物医药科技股份有限公司 | 沃赛汀或沃替西汀的氢溴酸盐 |
| CN104119298B (zh) * | 2014-08-13 | 2016-08-24 | 北京蓝贝望生物医药科技股份有限公司 | 氢溴酸沃赛汀或氢溴酸沃替西汀 |
| CN104610195B (zh) * | 2015-01-30 | 2017-06-27 | 上虞京新药业有限公司 | 沃替西汀的天冬氨酸盐或其水合物及其制备方法和用途 |
| BR112018003930A2 (pt) | 2016-07-01 | 2018-09-25 | H Lundbeck As | regimes de dosagem de vortioxetina para início rápido de efeito antidepressivo |
| EP3870292A4 (en) | 2018-10-26 | 2022-11-09 | The Research Foundation for The State University of New York | COMBINATION OF SEROTONIN-SPECIFIC RESUPPUT INHIBITOR AND SEROTONIN 1A RECEPTOR PARTIAL AGONIST TO REDUCE L-DOPA-INDUCED DYSKINESIA |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2008153632A2 (en) * | 2007-06-15 | 2008-12-18 | Vivus, Inc. | Compositions and methods for treating obesity and related disorders |
| WO2009062517A1 (en) * | 2007-11-13 | 2009-05-22 | H. Lundbeck A/S | Therapeutic uses of compounds having combined sert, 5-ht3 and 5-ht1a activity |
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| GB8430581D0 (en) * | 1984-12-04 | 1985-01-09 | Ferrosan As | Treatment |
| EP0543584B1 (en) * | 1991-11-18 | 1996-05-22 | Lilly Industries Limited | Benzo(b)thiophene-2-carboxamides for the treatment of disorders of the central nervous system |
| US7159383B2 (en) | 2000-10-02 | 2007-01-09 | Rohr, Inc. | Apparatus, method and system for gas turbine engine noise reduction |
| UA81749C2 (uk) | 2001-10-04 | 2008-02-11 | Х. Луннбек А/С | Фенілпіперазинові похідні як інгібітори зворотного захоплення серотоніну |
| KR101627901B1 (ko) * | 2006-06-16 | 2016-06-13 | 하. 룬트벡 아크티에 셀스카브 | 인지기능 장애의 치료를 위한, 세로토닌 재흡수, 5-ht3 및 5-ht1a 활성이 조합된 화합물로서의 1-[2-(2,4-디메틸페닐술파닐)-페닐]피페라진 |
| TW200848411A (en) | 2007-03-20 | 2008-12-16 | Lundbeck & Co As H | Novel therapeutic uses of 1-[2-(2, 4-dimethylphenylsulfanyl)phenyl]-piperazine |
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Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2008153632A2 (en) * | 2007-06-15 | 2008-12-18 | Vivus, Inc. | Compositions and methods for treating obesity and related disorders |
| WO2009062517A1 (en) * | 2007-11-13 | 2009-05-22 | H. Lundbeck A/S | Therapeutic uses of compounds having combined sert, 5-ht3 and 5-ht1a activity |
Non-Patent Citations (1)
| Title |
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| LAM D.D. et al., Distribution and neurochemical characterization of neurons within the nucleus of the solitary tract responsive to serotonin agonist-induced hypophagia, Behav Brain Res. 2009 Jan 3;196(1):139-43-реферат. doi: 10.1016/j.bbr.2008.07.039. Найдено из Интернета на сайте: http://www.ncbi.nlm.nih.gov/pubmed/18762217. CASSANO P. et al., Tolerability issues during long-term treatment with antidepressants, Ann Clin Psychiatry. 2004 Jan-Mar;16(1):15-25 -реферат. Найдено из Интернета на сайте: http://www.ncbi.nlm.nih.gov/pubmed/15147109 * |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2859008C2 (ru) * | 2020-04-03 | 2026-03-25 | Х. Лундбекк А/С | 1-[2-(2,4-диметилфенилсульфанил)фенил]пиперазин для предупреждения или лечения эмоциональной притупленности |
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