AR082501A1 - Usos terapeuticos de 1-[2-(2,4-dimetil-fenilsulfanil)fenil]piperazina - Google Patents
Usos terapeuticos de 1-[2-(2,4-dimetil-fenilsulfanil)fenil]piperazinaInfo
- Publication number
- AR082501A1 AR082501A1 ARP110103029A ARP110103029A AR082501A1 AR 082501 A1 AR082501 A1 AR 082501A1 AR P110103029 A ARP110103029 A AR P110103029A AR P110103029 A ARP110103029 A AR P110103029A AR 082501 A1 AR082501 A1 AR 082501A1
- Authority
- AR
- Argentina
- Prior art keywords
- piperazine
- dimethyl
- phenyl
- therapeutic uses
- phenylsulphanil
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
Abstract
Usos terapéuticos de 1-[2-(2,4-dimetil-fenilsulfanil)fenil)]piperazina y sus sales farmacéuticamente aceptables. Uso del mismo en la preparación de un medicamento para el tratamiento a largo plazo de una enfermedad del SNC no asociada a un aumento de peso y también cuando el paciente padece una enfermedad adicional a la del SNC en la cual debería evitarse el aumento de peso tal como diabetes tipo II y cardiopatías coronarias.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DKPA201000739 | 2010-08-23 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR082501A1 true AR082501A1 (es) | 2012-12-12 |
Family
ID=44532506
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP110103029A AR082501A1 (es) | 2010-08-23 | 2011-08-19 | Usos terapeuticos de 1-[2-(2,4-dimetil-fenilsulfanil)fenil]piperazina |
Country Status (30)
Country | Link |
---|---|
US (4) | US20130184291A1 (es) |
EP (1) | EP2608789B1 (es) |
JP (1) | JP5902169B2 (es) |
KR (1) | KR101816953B1 (es) |
CN (1) | CN103068389A (es) |
AP (1) | AP3583A (es) |
AR (1) | AR082501A1 (es) |
AU (1) | AU2011295465B8 (es) |
BR (2) | BR112013002194A2 (es) |
CA (1) | CA2807062C (es) |
CL (1) | CL2013000492A1 (es) |
CO (1) | CO6680652A2 (es) |
CY (1) | CY1118886T1 (es) |
DK (1) | DK2608789T3 (es) |
ES (1) | ES2625142T3 (es) |
HR (1) | HRP20170608T1 (es) |
HU (1) | HUE034155T2 (es) |
IL (1) | IL224371A (es) |
LT (1) | LT2608789T (es) |
ME (1) | ME02674B (es) |
MX (1) | MX349724B (es) |
PL (1) | PL2608789T3 (es) |
PT (1) | PT2608789T (es) |
RS (1) | RS55851B1 (es) |
RU (1) | RU2564666C2 (es) |
SG (1) | SG187649A1 (es) |
SI (1) | SI2608789T1 (es) |
TW (1) | TW201212918A (es) |
WO (1) | WO2012025123A1 (es) |
ZA (1) | ZA201301385B (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US9822086B2 (en) | 2014-01-31 | 2017-11-21 | Egis Gyogyszergyar Zrt. | Process for the preparation of vortioxetine salts |
CN104119299B (zh) * | 2014-08-13 | 2016-08-17 | 北京蓝贝望生物医药科技股份有限公司 | 沃赛汀或沃替西汀的氢溴酸盐 |
CN104119298B (zh) * | 2014-08-13 | 2016-08-24 | 北京蓝贝望生物医药科技股份有限公司 | 氢溴酸沃赛汀或氢溴酸沃替西汀 |
CN104610195B (zh) * | 2015-01-30 | 2017-06-27 | 上虞京新药业有限公司 | 沃替西汀的天冬氨酸盐或其水合物及其制备方法和用途 |
US9820984B1 (en) | 2016-07-01 | 2017-11-21 | H. Lundbeck A/S | Dosing regimens for fast onset of antidepressant effect |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8430581D0 (en) * | 1984-12-04 | 1985-01-09 | Ferrosan As | Treatment |
ATE138374T1 (de) * | 1991-11-18 | 1996-06-15 | Lilly Industries Ltd | Benzo(b)thiophen-2-carboxamide zur behandlung von krankheiten des zentralnervensystems |
US20080103179A1 (en) * | 2006-10-27 | 2008-05-01 | Tam Peter Y | Combination Therapy |
EP1322854A4 (en) | 2000-10-02 | 2004-08-04 | Rohr Inc | APPARATUS, METHOD AND SYSTEM FOR REDUCING THE NOISE OF A GAS TURBINE |
UA81749C2 (uk) | 2001-10-04 | 2008-02-11 | Х. Луннбек А/С | Фенілпіперазинові похідні як інгібітори зворотного захоплення серотоніну |
SI2044043T2 (sl) | 2006-06-16 | 2021-04-30 | H. Lundbeck A/S | 1-2(-2,4-dimetilfenilsulfanil)-fenil)piperazin hidrobromid kot spojina s kombinirano aktivnostjo ponovnega privzema serotonina, 5-ht3 in 5-ht1a za zdravljenje kognitivne motnje |
TW200848411A (en) | 2007-03-20 | 2008-12-16 | Lundbeck & Co As H | Novel therapeutic uses of 1-[2-(2, 4-dimethylphenylsulfanyl)phenyl]-piperazine |
TW200932233A (en) * | 2007-11-13 | 2009-08-01 | Lundbeck & Co As H | Therapeutic uses of compounds having combined SERT, 5-HT3 and 5-HT1a activity |
-
2011
- 2011-08-17 TW TW100129338A patent/TW201212918A/zh unknown
- 2011-08-19 AR ARP110103029A patent/AR082501A1/es not_active Application Discontinuation
- 2011-08-22 US US13/812,073 patent/US20130184291A1/en not_active Abandoned
- 2011-08-22 DK DK11749331.2T patent/DK2608789T3/en active
- 2011-08-22 MX MX2013001570A patent/MX349724B/es active IP Right Grant
- 2011-08-22 BR BR112013002194A patent/BR112013002194A2/pt not_active Application Discontinuation
- 2011-08-22 AP AP2013006768A patent/AP3583A/xx active
- 2011-08-22 CN CN2011800406861A patent/CN103068389A/zh active Pending
- 2011-08-22 PL PL11749331T patent/PL2608789T3/pl unknown
- 2011-08-22 ME MEP-2017-94A patent/ME02674B/me unknown
- 2011-08-22 PT PT117493312T patent/PT2608789T/pt unknown
- 2011-08-22 JP JP2013525143A patent/JP5902169B2/ja active Active
- 2011-08-22 CA CA2807062A patent/CA2807062C/en active Active
- 2011-08-22 HU HUE11749331A patent/HUE034155T2/en unknown
- 2011-08-22 KR KR1020137004481A patent/KR101816953B1/ko active IP Right Grant
- 2011-08-22 AU AU2011295465A patent/AU2011295465B8/en active Active
- 2011-08-22 LT LTEP11749331.2T patent/LT2608789T/lt unknown
- 2011-08-22 RU RU2013112890/15A patent/RU2564666C2/ru active
- 2011-08-22 EP EP11749331.2A patent/EP2608789B1/en active Active
- 2011-08-22 BR BR122020025600A patent/BR122020025600A2/pt not_active Application Discontinuation
- 2011-08-22 SI SI201131177A patent/SI2608789T1/sl unknown
- 2011-08-22 WO PCT/DK2011/050317 patent/WO2012025123A1/en active Application Filing
- 2011-08-22 ES ES11749331.2T patent/ES2625142T3/es active Active
- 2011-08-22 SG SG2013007380A patent/SG187649A1/en unknown
- 2011-08-22 RS RS20170404A patent/RS55851B1/sr unknown
-
2013
- 2013-01-23 IL IL224371A patent/IL224371A/en active IP Right Grant
- 2013-02-20 CL CL2013000492A patent/CL2013000492A1/es unknown
- 2013-02-21 CO CO13035030A patent/CO6680652A2/es unknown
- 2013-02-22 ZA ZA2013/01385A patent/ZA201301385B/en unknown
-
2017
- 2017-04-18 HR HRP20170608TT patent/HRP20170608T1/hr unknown
- 2017-05-10 CY CY20171100501T patent/CY1118886T1/el unknown
-
2018
- 2018-09-07 US US16/124,497 patent/US20190000836A1/en not_active Abandoned
-
2020
- 2020-05-18 US US16/877,108 patent/US20210085674A1/en not_active Abandoned
-
2022
- 2022-01-07 US US17/570,998 patent/US20220370439A1/en not_active Abandoned
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Legal Events
Date | Code | Title | Description |
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FC | Refusal |