RO72980A - PROCESS FOR PREPARING DERIVATIVES OF 3-TRIAZINYL-TOMOTIL-PHYALOSPORINE - Google Patents

PROCESS FOR PREPARING DERIVATIVES OF 3-TRIAZINYL-TOMOTIL-PHYALOSPORINE

Info

Publication number
RO72980A
RO72980A RO7593489A RO9348975A RO72980A RO 72980 A RO72980 A RO 72980A RO 7593489 A RO7593489 A RO 7593489A RO 9348975 A RO9348975 A RO 9348975A RO 72980 A RO72980 A RO 72980A
Authority
RO
Romania
Prior art keywords
tomotil
phyalosporine
triazinyl
preparing derivatives
derivatives
Prior art date
Application number
RO7593489A
Other languages
French (fr)
Romanian (ro)
Inventor
William H W Lunn
Original Assignee
Eli Lilly And Co,Us
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly And Co,Us filed Critical Eli Lilly And Co,Us
Publication of RO72980A publication Critical patent/RO72980A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36Methylene radicals, substituted by sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
RO7593489A 1974-08-02 1975-07-25 PROCESS FOR PREPARING DERIVATIVES OF 3-TRIAZINYL-TOMOTIL-PHYALOSPORINE RO72980A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US49414874A 1974-08-02 1974-08-02
US58392475A 1975-06-10 1975-06-10

Publications (1)

Publication Number Publication Date
RO72980A true RO72980A (en) 1981-08-30

Family

ID=27051316

Family Applications (1)

Application Number Title Priority Date Filing Date
RO7593489A RO72980A (en) 1974-08-02 1975-07-25 PROCESS FOR PREPARING DERIVATIVES OF 3-TRIAZINYL-TOMOTIL-PHYALOSPORINE

Country Status (22)

Country Link
JP (1) JPS6123195B2 (en)
AR (1) AR210998A1 (en)
AT (1) AT347580B (en)
BG (1) BG26395A3 (en)
CA (1) CA1100129A (en)
CH (1) CH616683A5 (en)
CS (1) CS189716B2 (en)
DD (1) DD121114A5 (en)
DE (1) DE2534071A1 (en)
DK (1) DK343275A (en)
FR (1) FR2280381A1 (en)
GB (1) GB1521073A (en)
HU (1) HU174130B (en)
IE (1) IE41590B1 (en)
IL (1) IL47802A (en)
NL (1) NL7509053A (en)
PH (1) PH16078A (en)
PL (1) PL95607B1 (en)
RO (1) RO72980A (en)
SE (1) SE426830B (en)
SU (1) SU755200A3 (en)
YU (1) YU197075A (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4348518A (en) 1974-05-05 1982-09-07 Hoffmann-La Roche Inc. Cephalosporins
JPS50141233U (en) * 1974-05-08 1975-11-20
NZ186610A (en) * 1977-03-07 1979-11-01 Lilly Co Eli Preparing of cephalosporins where the acetoxy group is displaced by a sulphur nucleophile
NL7805715A (en) * 1977-06-03 1978-12-05 Hoffmann La Roche METHOD FOR PREPARING ACYL DERIVATIVES.
US4200745A (en) * 1977-12-20 1980-04-29 Eli Lilly And Company 7[2-(2-Aminothiazol-4-yl)-2-alkoxyimino]acetamido 3[4-alkyl-5-oxo-6-hydroxy-3,4 dihydro 1,2,4-triazin 3-yl]thio methyl cephalosporins
MC1259A1 (en) * 1978-05-30 1980-01-14 Hoffmann La Roche ACYL DERIVATIVES
DK225179A (en) 1978-06-22 1979-12-23 Chugai Pharmaceutical Co Ltd PROCEDURE FOR PREPARING CEPHALOSPORINE DERIVATIVES
NO782998L (en) * 1978-07-19 1980-01-22 Hoffmann La Roche CEPHALOSPORINESTERS AND EATERS.
NL8100089A (en) 1980-01-17 1981-08-17 Rhone Poulenc Ind NEW THIOLS AND THEIR PREPARATION.
FR2474030A1 (en) * 1980-01-17 1981-07-24 Rhone Poulenc Ind 2-Mercapto-1,2,4-triazine, 1,3,4-triazole or tetrazole derivs. - useful as intermediates for antibacterial cephalosporin(s)
FR2494278A1 (en) * 1980-11-20 1982-05-21 Rhone Poulenc Ind NEW DERIVATIVES OF CEPHALOSPORIN, THEIR PREPARATIONS AND THE MEDICINAL PRODUCTS CONTAINING THEM

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5116436B1 (en) * 1971-05-31 1976-05-24

Also Published As

Publication number Publication date
IE41590L (en) 1976-02-02
GB1521073A (en) 1978-08-09
PL95607B1 (en) 1977-10-31
PH16078A (en) 1983-06-20
CS189716B2 (en) 1979-04-30
JPS5139693A (en) 1976-04-02
DD121114A5 (en) 1976-07-12
IE41590B1 (en) 1980-02-13
SE426830B (en) 1983-02-14
BG26395A3 (en) 1979-03-15
SE7508570L (en) 1976-02-03
CH616683A5 (en) 1980-04-15
FR2280381B1 (en) 1979-08-10
NL7509053A (en) 1976-02-04
IL47802A0 (en) 1975-10-15
CA1100129A (en) 1981-04-28
DE2534071A1 (en) 1976-02-12
FR2280381A1 (en) 1976-02-27
AT347580B (en) 1979-01-10
IL47802A (en) 1980-05-30
SU755200A3 (en) 1980-08-07
HU174130B (en) 1979-11-28
DK343275A (en) 1976-02-03
YU197075A (en) 1982-05-31
JPS6123195B2 (en) 1986-06-04
AR210998A1 (en) 1977-10-14
ATA594075A (en) 1976-11-15

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