PT89997A - Processo para a preparacao de derivados 1-carbonil de 4-aril-4-arilxipiperidinas e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de derivados 1-carbonil de 4-aril-4-arilxipiperidinas e de composicoes farmaceuticas que os contem

Info

Publication number
PT89997A
PT89997A PT89997A PT8999789A PT89997A PT 89997 A PT89997 A PT 89997A PT 89997 A PT89997 A PT 89997A PT 8999789 A PT8999789 A PT 8999789A PT 89997 A PT89997 A PT 89997A
Authority
PT
Portugal
Prior art keywords
arylipiperidines
aryl
contain
pharmaceutical compositions
carbonyl derivatives
Prior art date
Application number
PT89997A
Other languages
English (en)
Inventor
Grover Cleveland Helsley
Larry Davis
Gordom Edward Olsen
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of PT89997A publication Critical patent/PT89997A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/52Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT89997A 1988-03-14 1989-03-13 Processo para a preparacao de derivados 1-carbonil de 4-aril-4-arilxipiperidinas e de composicoes farmaceuticas que os contem PT89997A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/167,929 US4853384A (en) 1988-03-14 1988-03-14 1-carbonyl derivatives of 4-aryl-4-aryloxypiperidines

Publications (1)

Publication Number Publication Date
PT89997A true PT89997A (pt) 1989-11-10

Family

ID=22609403

Family Applications (1)

Application Number Title Priority Date Filing Date
PT89997A PT89997A (pt) 1988-03-14 1989-03-13 Processo para a preparacao de derivados 1-carbonil de 4-aril-4-arilxipiperidinas e de composicoes farmaceuticas que os contem

Country Status (5)

Country Link
US (1) US4853384A (pt)
EP (1) EP0333025A1 (pt)
JP (1) JPH01275558A (pt)
DK (1) DK120989A (pt)
PT (1) PT89997A (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GEP20094676B (en) * 2003-07-24 2009-05-10 Euro Celtique Sa Piperidine compounds and pharmaceutical compositions containing them
WO2007044804A2 (en) * 2005-10-11 2007-04-19 Chemocentryx, Inc. Piperidine derivatives and methods of use

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2850500A (en) * 1958-09-02 Chjchzcoochj
GB1280699A (en) * 1968-12-23 1972-07-05 Robins Co Inc A H 0-substituted-4-phenoxypiperidines
US3996366A (en) * 1973-11-19 1976-12-07 The Boots Company Limited Thio derivatives of imidazol-1-yl carboxamides
US4333942A (en) * 1979-08-03 1982-06-08 Byk Gulden Lomberg Chemische Fabrik Gmbh Anti-depressant and analgesic 4-phenoxypiperidines
US4330546A (en) * 1979-09-14 1982-05-18 John Wyeth & Brother Limited 3-Aryl-3-aryloxypropylamines
GB2060619B (en) * 1979-09-14 1983-06-08 Wyeth John & Brother Ltd 4-aryl-4-aryloxypiperidines

Also Published As

Publication number Publication date
JPH01275558A (ja) 1989-11-06
EP0333025A1 (en) 1989-09-20
US4853384A (en) 1989-08-01
DK120989D0 (da) 1989-03-13
DK120989A (da) 1989-09-15

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Legal Events

Date Code Title Description
FC3A Refusal

Effective date: 19940427