PT89370A - Processo para a preparacao de compostos derivados de mercapto-imidazolinas, dos seus intermedarios e de composicoes farmaceuticas contendo aqueles derivados - Google Patents

Processo para a preparacao de compostos derivados de mercapto-imidazolinas, dos seus intermedarios e de composicoes farmaceuticas contendo aqueles derivados

Info

Publication number
PT89370A
PT89370A PT89370A PT8937088A PT89370A PT 89370 A PT89370 A PT 89370A PT 89370 A PT89370 A PT 89370A PT 8937088 A PT8937088 A PT 8937088A PT 89370 A PT89370 A PT 89370A
Authority
PT
Portugal
Prior art keywords
imidazolines
mercapto
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
PT89370A
Other languages
English (en)
Inventor
Lawrence Ivan Kruse
Stephen Torey Ross
Thomas Brent Leonard
Original Assignee
Smithkline Beckman Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beckman Corp filed Critical Smithkline Beckman Corp
Publication of PT89370A publication Critical patent/PT89370A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/30Oxygen or sulfur atoms
    • C07D233/42Sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C333/00Derivatives of thiocarbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C333/14Dithiocarbamic acids; Derivatives thereof
    • C07C333/16Salts of dithiocarbamic acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT89370A 1987-12-31 1988-12-30 Processo para a preparacao de compostos derivados de mercapto-imidazolinas, dos seus intermedarios e de composicoes farmaceuticas contendo aqueles derivados PT89370A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/140,053 US4876266A (en) 1987-12-31 1987-12-31 1-aralkyl-2-mercaptoimidazolines as DBH inhibitors

Publications (1)

Publication Number Publication Date
PT89370A true PT89370A (pt) 1989-12-29

Family

ID=22489533

Family Applications (1)

Application Number Title Priority Date Filing Date
PT89370A PT89370A (pt) 1987-12-31 1988-12-30 Processo para a preparacao de compostos derivados de mercapto-imidazolinas, dos seus intermedarios e de composicoes farmaceuticas contendo aqueles derivados

Country Status (7)

Country Link
US (1) US4876266A (pt)
EP (1) EP0329900A1 (pt)
JP (1) JPH03501728A (pt)
AU (1) AU2911389A (pt)
PT (1) PT89370A (pt)
WO (1) WO1989006126A1 (pt)
ZA (1) ZA889708B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3821464A1 (de) * 1988-06-25 1989-12-28 Degussa Verfahren zur herstellung substituierter organyloxysilylfunktioneller, cyclischer thioharnstoffe und diese verbindungen
CA2518941C (en) * 2003-03-19 2011-06-14 Maschinenfabrik Reinhausen Gmbh Pressure-relief valve
DE10312177B3 (de) * 2003-03-19 2004-06-17 Maschinenfabrik Reinhausen Gmbh Druckentlastungsventil
WO2013134047A2 (en) 2012-03-07 2013-09-12 The Mclean Hospital Corporation Aminoquinoline derivatives and uses thereof
EP3138863A1 (de) * 2015-09-01 2017-03-08 Sika Technology AG Emissionsarme epoxidharz-zusammensetzung

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2839561A (en) * 1955-02-10 1958-06-17 Bayer Ag Dithiocarbonic acid esters and production
BE688585A (pt) * 1965-10-21 1967-04-20
GB1261345A (en) * 1968-03-07 1972-01-26 Ici Ltd Sulphur-containing benzyl derivatives and pesticidal compositions containing them
BE787477A (fr) * 1971-08-12 1973-02-12 Bayer Ag 1-phenyl-2-imino-imidazolidines, leur procede de preparation etleur application comme repulsifs a l'egard des oiseaux
DE2259627A1 (de) * 1972-12-06 1974-06-12 Hoechst Ag Imidazolyl-(2)-thio-alkansaeureester und verfahren zu ihrer herstellung
US4284641A (en) * 1977-08-26 1981-08-18 Burroughs Wellcome Co. Pharmaceutically active imidazole derivatives
GB2096987B (en) * 1981-04-22 1984-04-04 Farmos Oy Substituted imidazole and imidazole derivatives and their preparation and use
US4532331A (en) * 1983-04-12 1985-07-30 Smithkline Beckman Corporation 1-Benzyl-2-aminomethyl imidazole derivatives
PT78388B (en) * 1983-04-12 1986-09-15 Smithkline Beckman Corp Dopamine-beta-hydroxylase inhibitors
JPS614038A (ja) * 1984-06-18 1986-01-09 Asahi Chem Ind Co Ltd 新規な感光性組成物

Also Published As

Publication number Publication date
JPH03501728A (ja) 1991-04-18
US4876266A (en) 1989-10-24
EP0329900A1 (en) 1989-08-30
ZA889708B (en) 1989-12-27
AU2911389A (en) 1989-08-01
WO1989006126A1 (en) 1989-07-13

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Legal Events

Date Code Title Description
FC3A Refusal

Effective date: 19940721