PT89657A - Processo de preparacao de derivados do imidazolo, dos seus intermediarios e de composicoes farmaceuticas contendo aqueles compostos - Google Patents
Processo de preparacao de derivados do imidazolo, dos seus intermediarios e de composicoes farmaceuticas contendo aqueles compostosInfo
- Publication number
- PT89657A PT89657A PT89657A PT8965789A PT89657A PT 89657 A PT89657 A PT 89657A PT 89657 A PT89657 A PT 89657A PT 8965789 A PT8965789 A PT 8965789A PT 89657 A PT89657 A PT 89657A
- Authority
- PT
- Portugal
- Prior art keywords
- imidazolo
- intermediaries
- pharmaceutical compositions
- compositions containing
- those compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/30—Oxygen or sulfur atoms
- C07D233/32—One oxygen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Biochemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biophysics (AREA)
- Public Health (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT8819336A IT1233860B (it) | 1988-02-08 | 1988-02-08 | Derivati del peridroazacicloalca (1,2-a) imidazolo ad attivita' nootropa |
Publications (2)
Publication Number | Publication Date |
---|---|
PT89657A true PT89657A (pt) | 1989-10-04 |
PT89657B PT89657B (pt) | 1994-02-28 |
Family
ID=11156852
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT89657A PT89657B (pt) | 1988-02-08 | 1989-02-08 | Processo de preparacao de derivados do imidazolo, dos seus intermediarios e de composicoes farmaceuticas contendo aqueles compostos |
Country Status (21)
Country | Link |
---|---|
US (2) | US5053422A (pt) |
EP (1) | EP0335483A3 (pt) |
JP (1) | JPH01246281A (pt) |
KR (1) | KR890013013A (pt) |
CN (1) | CN1036204A (pt) |
AU (2) | AU616240B2 (pt) |
BR (1) | BR8900541A (pt) |
CA (1) | CA1324378C (pt) |
DD (2) | DD291996A5 (pt) |
DK (1) | DK55089A (pt) |
FI (1) | FI890438A (pt) |
HU (2) | HU204794B (pt) |
IT (1) | IT1233860B (pt) |
NO (1) | NO168424C (pt) |
NZ (1) | NZ227833A (pt) |
PL (1) | PL158198B1 (pt) |
PT (1) | PT89657B (pt) |
RO (4) | RO105965B1 (pt) |
RU (1) | RU1799383C (pt) |
ZA (1) | ZA89894B (pt) |
ZW (1) | ZW1489A1 (pt) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9123641D0 (en) * | 1991-11-07 | 1992-01-02 | Isf Spa | Process |
TW304167B (pt) * | 1995-01-30 | 1997-05-01 | Lilly Co Eli | |
PE17897A1 (es) * | 1995-02-17 | 1997-06-12 | Lilly Co Eli | Formulacion transdermica en parche del 3-(4-butiltio)-1,2,5-tiadiazol-3-il)-1-azabiciclo (2,2,2) octano |
ZA964008B (en) * | 1995-06-02 | 1997-07-11 | Akzo Nobel Nv | Imidazo[1,5a]pyridine derived serine protease inhibitors |
JP3905409B2 (ja) | 2002-04-10 | 2007-04-18 | タレックス光学工業株式会社 | 光学レンズ成型用ポリウレタン樹脂組成物および耐衝撃性合成樹脂レンズ |
ITMI20030573A1 (it) * | 2003-03-24 | 2004-09-25 | Nikem Research Srl | Composti ad azione nootropica, loro preparazione, |
ITMI20070770A1 (it) | 2007-04-16 | 2008-10-17 | Brane Discovery S R L | Impiego di dimiracetam nel trattamento del dolore cronico |
US9593209B2 (en) | 2009-10-22 | 2017-03-14 | Dow Corning Corporation | Process for preparing clustered functional polyorganosiloxanes, and methods for their use |
CN103052638B (zh) * | 2010-07-26 | 2015-09-30 | 神经协调股份公司 | 制备地来西坦的方法 |
KR102172738B1 (ko) | 2013-02-11 | 2020-11-02 | 다우 실리콘즈 코포레이션 | 클러스터형 작용성 폴리오르가노실록산, 이의 형성 방법, 및 이의 사용 방법 |
KR102192489B1 (ko) | 2013-02-11 | 2020-12-17 | 다우 실리콘즈 코포레이션 | 열 전도성 열 라디칼 경화 실리콘 조성물을 형성하는 원 위치 방법 |
WO2014124389A1 (en) | 2013-02-11 | 2014-08-14 | Dow Corning Corporation | Moisture-curable hot melt silicone adhesive compositions including an alkoxy-functional siloxane reactive resin |
EP2954024B1 (en) | 2013-02-11 | 2019-05-15 | Dow Silicones Corporation | Curable silicone compositions comprising clustered functional polyorganosiloxanes and silicone reactive diluents |
KR102206708B1 (ko) | 2013-02-11 | 2021-01-25 | 다우 실리콘즈 코포레이션 | 안정한 열 라디칼 경화성 실리콘 접착제 조성물 |
CN104968748B (zh) | 2013-02-11 | 2017-03-29 | 道康宁公司 | 烷氧基官能化有机聚硅氧烷树脂和聚合物及其相关形成方法 |
US10370574B2 (en) | 2013-02-11 | 2019-08-06 | Dow Silicones Corporation | Method for forming thermally conductive thermal radical cure silicone compositions |
EP3196229B1 (en) | 2015-11-05 | 2018-09-26 | Dow Silicones Corporation | Branched polyorganosiloxanes and related curable compositions, methods, uses and devices |
JOP20190251A1 (ar) | 2017-05-31 | 2019-10-21 | Metys Pharmaceuticals AG | تركيبات تآزرية تشتمل على (r)-ديميراسيتام (1) و(s)-ديميراسيتام (2) بنسبة غير راسيمية |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3334099A (en) * | 1965-03-31 | 1967-08-01 | Sandoz Ag | Novel pyrrolo-diazepines, pyrrolo-imidazolidines, and pyrrolo-pyrimidines |
FR2358891A1 (fr) * | 1976-07-22 | 1978-02-17 | Yamanouchi Pharma Co Ltd | Composes heterocycliques contenant un azote, utilise comme agents analgesiques et anti-inflammatoires |
US4372966A (en) * | 1980-09-15 | 1983-02-08 | Warner-Lambert Company | Use of dihydro-1H-pyrrolizine-3,5(2H,6H)-dione as a cognition activator |
US4582838A (en) * | 1984-08-24 | 1986-04-15 | Warner-Lambert Company | Derivatives of dihydro-1H-pyrrolo[1,2-c]imidazol-3,5-dione as cognition activators |
US4677098A (en) * | 1985-11-22 | 1987-06-30 | Warner-Lambert Company | Substituted dihydro-1H-pyrolizine-3,5(2H,6H)-diones |
JPS62289581A (ja) * | 1986-06-09 | 1987-12-16 | Idemitsu Kosan Co Ltd | イミダゾピロリンジオン誘導体,その製造方法およびそれを有効成分とする除草剤 |
JPS62292783A (ja) * | 1986-06-12 | 1987-12-19 | Idemitsu Kosan Co Ltd | イミダゾピロリンジオン誘導体,その製造方法およびそれを有効成分として含有する除草剤 |
-
1988
- 1988-02-08 IT IT8819336A patent/IT1233860B/it active
-
1989
- 1989-01-30 FI FI890438A patent/FI890438A/fi not_active Application Discontinuation
- 1989-02-02 NZ NZ227833A patent/NZ227833A/xx unknown
- 1989-02-03 BR BR898900541A patent/BR8900541A/pt unknown
- 1989-02-03 ZW ZW14/89A patent/ZW1489A1/xx unknown
- 1989-02-04 CN CN89101740A patent/CN1036204A/zh active Pending
- 1989-02-06 DD DD89337916A patent/DD291996A5/de not_active IP Right Cessation
- 1989-02-06 CA CA000590213A patent/CA1324378C/en not_active Expired - Lifetime
- 1989-02-06 EP EP19890301123 patent/EP0335483A3/en not_active Ceased
- 1989-02-06 US US07/307,012 patent/US5053422A/en not_active Expired - Lifetime
- 1989-02-06 ZA ZA89894A patent/ZA89894B/xx unknown
- 1989-02-06 DD DD89325551A patent/DD283393A5/de not_active IP Right Cessation
- 1989-02-07 RU SU894613489A patent/RU1799383C/ru active
- 1989-02-07 HU HU904864A patent/HU204794B/hu not_active IP Right Cessation
- 1989-02-07 HU HU89574A patent/HU203104B/hu not_active IP Right Cessation
- 1989-02-07 NO NO890515A patent/NO168424C/no unknown
- 1989-02-07 PL PL1989277610A patent/PL158198B1/pl unknown
- 1989-02-07 DK DK055089A patent/DK55089A/da not_active Application Discontinuation
- 1989-02-07 AU AU29692/89A patent/AU616240B2/en not_active Ceased
- 1989-02-08 KR KR1019890001446A patent/KR890013013A/ko not_active Application Discontinuation
- 1989-02-08 RO RO145765A patent/RO105965B1/ro unknown
- 1989-02-08 PT PT89657A patent/PT89657B/pt active IP Right Grant
- 1989-02-08 RO RO145763A patent/RO105963B1/ro unknown
- 1989-02-08 RO RO138146A patent/RO104070B1/ro unknown
- 1989-02-08 RO RO145764A patent/RO105964B1/ro unknown
- 1989-02-08 JP JP1029571A patent/JPH01246281A/ja active Pending
-
1991
- 1991-03-15 US US07/669,806 patent/US5130319A/en not_active Expired - Lifetime
- 1991-07-01 AU AU79479/91A patent/AU7947991A/en not_active Abandoned
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG3A | Patent granted, date of granting |
Effective date: 19930809 |