PT89657A - Processo de preparacao de derivados do imidazolo, dos seus intermediarios e de composicoes farmaceuticas contendo aqueles compostos - Google Patents

Processo de preparacao de derivados do imidazolo, dos seus intermediarios e de composicoes farmaceuticas contendo aqueles compostos

Info

Publication number
PT89657A
PT89657A PT89657A PT8965789A PT89657A PT 89657 A PT89657 A PT 89657A PT 89657 A PT89657 A PT 89657A PT 8965789 A PT8965789 A PT 8965789A PT 89657 A PT89657 A PT 89657A
Authority
PT
Portugal
Prior art keywords
imidazolo
intermediaries
pharmaceutical compositions
compositions containing
those compounds
Prior art date
Application number
PT89657A
Other languages
English (en)
Other versions
PT89657B (pt
Inventor
Mario Pinza
Carlo Farina
Alberto Cerri
Maria Teresa Riccaboni
Original Assignee
Isf Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Isf Spa filed Critical Isf Spa
Publication of PT89657A publication Critical patent/PT89657A/pt
Publication of PT89657B publication Critical patent/PT89657B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/30Oxygen or sulfur atoms
    • C07D233/32One oxygen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06139Dipeptides with the first amino acid being heterocyclic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Public Health (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pyrrole Compounds (AREA)
PT89657A 1988-02-08 1989-02-08 Processo de preparacao de derivados do imidazolo, dos seus intermediarios e de composicoes farmaceuticas contendo aqueles compostos PT89657B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT8819336A IT1233860B (it) 1988-02-08 1988-02-08 Derivati del peridroazacicloalca (1,2-a) imidazolo ad attivita' nootropa

Publications (2)

Publication Number Publication Date
PT89657A true PT89657A (pt) 1989-10-04
PT89657B PT89657B (pt) 1994-02-28

Family

ID=11156852

Family Applications (1)

Application Number Title Priority Date Filing Date
PT89657A PT89657B (pt) 1988-02-08 1989-02-08 Processo de preparacao de derivados do imidazolo, dos seus intermediarios e de composicoes farmaceuticas contendo aqueles compostos

Country Status (21)

Country Link
US (2) US5053422A (pt)
EP (1) EP0335483A3 (pt)
JP (1) JPH01246281A (pt)
KR (1) KR890013013A (pt)
CN (1) CN1036204A (pt)
AU (2) AU616240B2 (pt)
BR (1) BR8900541A (pt)
CA (1) CA1324378C (pt)
DD (2) DD291996A5 (pt)
DK (1) DK55089A (pt)
FI (1) FI890438A (pt)
HU (2) HU204794B (pt)
IT (1) IT1233860B (pt)
NO (1) NO168424C (pt)
NZ (1) NZ227833A (pt)
PL (1) PL158198B1 (pt)
PT (1) PT89657B (pt)
RO (4) RO105965B1 (pt)
RU (1) RU1799383C (pt)
ZA (1) ZA89894B (pt)
ZW (1) ZW1489A1 (pt)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9123641D0 (en) * 1991-11-07 1992-01-02 Isf Spa Process
TW304167B (pt) * 1995-01-30 1997-05-01 Lilly Co Eli
PE17897A1 (es) * 1995-02-17 1997-06-12 Lilly Co Eli Formulacion transdermica en parche del 3-(4-butiltio)-1,2,5-tiadiazol-3-il)-1-azabiciclo (2,2,2) octano
ZA964008B (en) * 1995-06-02 1997-07-11 Akzo Nobel Nv Imidazo[1,5a]pyridine derived serine protease inhibitors
JP3905409B2 (ja) 2002-04-10 2007-04-18 タレックス光学工業株式会社 光学レンズ成型用ポリウレタン樹脂組成物および耐衝撃性合成樹脂レンズ
ITMI20030573A1 (it) * 2003-03-24 2004-09-25 Nikem Research Srl Composti ad azione nootropica, loro preparazione,
ITMI20070770A1 (it) 2007-04-16 2008-10-17 Brane Discovery S R L Impiego di dimiracetam nel trattamento del dolore cronico
US9593209B2 (en) 2009-10-22 2017-03-14 Dow Corning Corporation Process for preparing clustered functional polyorganosiloxanes, and methods for their use
CN103052638B (zh) * 2010-07-26 2015-09-30 神经协调股份公司 制备地来西坦的方法
KR102172738B1 (ko) 2013-02-11 2020-11-02 다우 실리콘즈 코포레이션 클러스터형 작용성 폴리오르가노실록산, 이의 형성 방법, 및 이의 사용 방법
KR102192489B1 (ko) 2013-02-11 2020-12-17 다우 실리콘즈 코포레이션 열 전도성 열 라디칼 경화 실리콘 조성물을 형성하는 원 위치 방법
WO2014124389A1 (en) 2013-02-11 2014-08-14 Dow Corning Corporation Moisture-curable hot melt silicone adhesive compositions including an alkoxy-functional siloxane reactive resin
EP2954024B1 (en) 2013-02-11 2019-05-15 Dow Silicones Corporation Curable silicone compositions comprising clustered functional polyorganosiloxanes and silicone reactive diluents
KR102206708B1 (ko) 2013-02-11 2021-01-25 다우 실리콘즈 코포레이션 안정한 열 라디칼 경화성 실리콘 접착제 조성물
CN104968748B (zh) 2013-02-11 2017-03-29 道康宁公司 烷氧基官能化有机聚硅氧烷树脂和聚合物及其相关形成方法
US10370574B2 (en) 2013-02-11 2019-08-06 Dow Silicones Corporation Method for forming thermally conductive thermal radical cure silicone compositions
EP3196229B1 (en) 2015-11-05 2018-09-26 Dow Silicones Corporation Branched polyorganosiloxanes and related curable compositions, methods, uses and devices
JOP20190251A1 (ar) 2017-05-31 2019-10-21 Metys Pharmaceuticals AG تركيبات تآزرية تشتمل على (r)-ديميراسيتام (1) و(s)-ديميراسيتام (2) بنسبة غير راسيمية

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3334099A (en) * 1965-03-31 1967-08-01 Sandoz Ag Novel pyrrolo-diazepines, pyrrolo-imidazolidines, and pyrrolo-pyrimidines
FR2358891A1 (fr) * 1976-07-22 1978-02-17 Yamanouchi Pharma Co Ltd Composes heterocycliques contenant un azote, utilise comme agents analgesiques et anti-inflammatoires
US4372966A (en) * 1980-09-15 1983-02-08 Warner-Lambert Company Use of dihydro-1H-pyrrolizine-3,5(2H,6H)-dione as a cognition activator
US4582838A (en) * 1984-08-24 1986-04-15 Warner-Lambert Company Derivatives of dihydro-1H-pyrrolo[1,2-c]imidazol-3,5-dione as cognition activators
US4677098A (en) * 1985-11-22 1987-06-30 Warner-Lambert Company Substituted dihydro-1H-pyrolizine-3,5(2H,6H)-diones
JPS62289581A (ja) * 1986-06-09 1987-12-16 Idemitsu Kosan Co Ltd イミダゾピロリンジオン誘導体,その製造方法およびそれを有効成分とする除草剤
JPS62292783A (ja) * 1986-06-12 1987-12-19 Idemitsu Kosan Co Ltd イミダゾピロリンジオン誘導体,その製造方法およびそれを有効成分として含有する除草剤

Also Published As

Publication number Publication date
CN1036204A (zh) 1989-10-11
EP0335483A3 (en) 1991-12-18
DK55089A (da) 1989-08-09
IT8819336A0 (it) 1988-02-08
AU616240B2 (en) 1991-10-24
EP0335483A2 (en) 1989-10-04
ZW1489A1 (en) 1989-08-02
DD291996A5 (de) 1991-07-18
DD283393A5 (de) 1990-10-10
AU2969289A (en) 1989-08-10
JPH01246281A (ja) 1989-10-02
HU204794B (en) 1992-02-28
NO168424B (no) 1991-11-11
NO890515D0 (no) 1989-02-07
RU1799383C (ru) 1993-02-28
ZA89894B (en) 1991-10-30
PT89657B (pt) 1994-02-28
BR8900541A (pt) 1989-10-03
FI890438A0 (fi) 1989-01-30
IT1233860B (it) 1992-04-21
HU203104B (en) 1991-05-28
CA1324378C (en) 1993-11-16
PL158198B1 (pl) 1992-08-31
DK55089D0 (da) 1989-02-07
FI890438A (fi) 1989-08-09
RO105965B1 (ro) 1993-01-30
KR890013013A (ko) 1989-09-20
HUT53363A (en) 1990-10-28
NO890515L (no) 1989-08-09
NO168424C (no) 1992-02-19
RO105964B1 (ro) 1993-01-30
AU7947991A (en) 1991-09-12
HU904864D0 (en) 1991-01-28
RO104070B1 (en) 1993-07-20
US5053422A (en) 1991-10-01
NZ227833A (en) 1991-09-25
US5130319A (en) 1992-07-14
RO105963B1 (ro) 1993-01-30

Similar Documents

Publication Publication Date Title
PT91042A (pt) Processo de preparacao de derivados da pirimidina fundidos, dos seus intermediarios e de composicoes farmaceuticas
PT90893A (pt) Processo de preparacao de derivados da pirimidina, de seus intermediarios e de composicoes farmaceuticas que os contem
PT89657A (pt) Processo de preparacao de derivados do imidazolo, dos seus intermediarios e de composicoes farmaceuticas contendo aqueles compostos
PT82623B (pt) Processo para a preparacao de analogos imidazolicos de mevalonolactona e dos seus derivados
PT89793A (pt) Processo de preparacao de derivados de quinolina substituidos e de composicoes farmaceuticas que os contem
PT93241A (pt) Processo de preparacao de derivados de piperidina e de composicoes farmaceuticas que os contem
PT83608B (pt) Processo de preparacao de derivados da paroxetina
PT91099A (pt) Processo de preparacao de peptidos de ligacao a proteases de retroviros, dos seus intermediarios e de composicoes farmaceuticas
PT91299A (pt) Processo para a preparacao de aminometiltetralinas substituidas e de seus analogos heterociclicos
PT84790B (pt) Processo de preparacao de derivados de amino-tiazol e de amino-oxazole e de composicoes farmaceuticas contendo-os
BR9609420A (pt) Derivados de 4-fenilaminotiazol seu processo de preparação e as composições farmacêuticas contendo os mesmos
PT82985A (pt) Process for the preparation of distamycin derivatives and of pharmaceutical compositions containing the same
PT91098A (pt) Processo de preparacao de derivados de (aza)naftalenossultame
PT83896B (pt) Processo para a preparacao de novos conjugados da vinblastina e dos seus derivados, e de composicoes farmaceuticas que os contem
PT83998B (pt) Processo de preparacao de novos derivados azaciclicos e de composicoes farmaceuticas que os contem
PT89789A (pt) Processo de preparacao de novos derivados substituidos da quinolina e de composicoes farmaceuticas contendo tais derivados
PT81760B (pt) Processo para a preparacao de compostos de podofilotoxina e seus derivados e de composicoes farmaceuticas contendo os mesmos
PT81029B (pt) Processo para a preparacao de derivados de flavanona com efeito antialergico e aplicacao dos mesmos para a preparacao de composicoes farmaceuticas com efeito antialergico
PT89616A (pt) Processo para a preparacao de composicoes artropodicidas contendo misturas sinergicas de derivados piretroides e butoxido de piperonilo
PT83173B (pt) Processo de preparacao de novos derivados de beta-lactama e seus intermediarios
PT88202A (pt) Processo para a preparacao dos compostos de 1-fenil-3-(1-piperazinil)-1h-indazol e seus intermediarios e de composicoes farmaceuticas que os contem
PT82319B (pt) Processo de preparacao de derivados de indeno e de naftaleno e de composicoes farmceuticas que os contem
PT87024A (pt) Process for the preparation of propiolophenone derivatives and of pharmaceutical compositions containing the same
IT1208807B (it) Derivati di 1 3 ossazolidin 2 one e procedimenti per la loro preparazione
PT89790A (pt) Processo de preparacao de derivados da quinolina substituidos e de composicoes farmaceuticas que os contem

Legal Events

Date Code Title Description
FG3A Patent granted, date of granting

Effective date: 19930809