PT86642A - Arylthiadiazolylsulfonamides and derivatives a process for thir preparation and their use as medicaments - Google Patents

Arylthiadiazolylsulfonamides and derivatives a process for thir preparation and their use as medicaments

Info

Publication number
PT86642A
PT86642A PT86642A PT8664288A PT86642A PT 86642 A PT86642 A PT 86642A PT 86642 A PT86642 A PT 86642A PT 8664288 A PT8664288 A PT 8664288A PT 86642 A PT86642 A PT 86642A
Authority
PT
Portugal
Prior art keywords
arylthiadiazolylsulfonamides
thir
medicines
derivatives
preparation
Prior art date
Application number
PT86642A
Other languages
English (en)
Other versions
PT86642B (pt
Inventor
John Joseph Tegeler
Kirk David Shoger
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of PT86642A publication Critical patent/PT86642A/pt
Publication of PT86642B publication Critical patent/PT86642B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/081,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT86642A 1987-01-29 1988-01-27 Processo para a preparacao de ariltiadiazolilsulfonamidas e seus derivados e de composicoes farmaceuticas que os contem PT86642B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/008,225 US4758578A (en) 1987-01-29 1987-01-29 Arylthiadiazolylsulfonamides, pharmaceutical compositions and use

Publications (2)

Publication Number Publication Date
PT86642A true PT86642A (pt) 1988-02-01
PT86642B PT86642B (pt) 1992-01-31

Family

ID=21730449

Family Applications (1)

Application Number Title Priority Date Filing Date
PT86642A PT86642B (pt) 1987-01-29 1988-01-27 Processo para a preparacao de ariltiadiazolilsulfonamidas e seus derivados e de composicoes farmaceuticas que os contem

Country Status (6)

Country Link
US (1) US4758578A (pt)
EP (1) EP0276822A1 (pt)
JP (1) JPS63192764A (pt)
DK (1) DK42888A (pt)
IE (1) IE880233L (pt)
PT (1) PT86642B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5104887A (en) * 1983-02-04 1992-04-14 University Of Iowa Research Foundation Topical ophthalmic imino substituted 2-imino-3-methyl-delta4-1,3,4-thiadiazoline-5-sulfonamides carbonic anhydrase inhibitors
NZ231534A (en) * 1988-11-29 1992-02-25 Warner Lambert Co 3,5-di-t-butyl-4-hydroxyphenyl-triazoles, oxadiazoles and thiadiazoles; anti-inflammatory compositions
US5256680A (en) * 1988-11-29 1993-10-26 Warner-Lambert Company 3,5-di-tertiary-butyl-4-hydroxyphenyl-1,3,4-thiadiazoles, and oxadiazoles and 3,5-di-tertiary-butyl-4-hydroxy-phenyl-1,2,4-thiadazoles, oxadiazoles and triazoles as antiinflammatory agents
US5155122A (en) * 1988-11-29 1992-10-13 Warner-Lambert Company 3,5-di-tertiary-butyl-4-hydroxyphenyl-1,3,4-thiadiazoles, and oxadiazoles and 3,5-di-tertiary-butyl-4-hydroxy-phenyl-1,2,4-thiadazoles, oxadiazoles and triazoles as antiinflammatory agents
DE19847823A1 (de) * 1998-10-16 2000-04-20 Aventis Pharma Gmbh Substituierte Thiadiazolsulfonamide

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3899502A (en) * 1973-05-14 1975-08-12 Monsanto Co 1,2,4-Thiadiazol-3,5-diyl-sulfenamides
DE2452618A1 (de) * 1974-11-06 1976-05-13 Merck Patent Gmbh Sulfenamide

Also Published As

Publication number Publication date
IE880233L (en) 1988-07-29
US4758578A (en) 1988-07-19
DK42888A (da) 1988-07-30
DK42888D0 (da) 1988-01-28
JPS63192764A (ja) 1988-08-10
PT86642B (pt) 1992-01-31
EP0276822A1 (en) 1988-08-03

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Legal Events

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Effective date: 19930131