PL4038052T3 - Antagoniści receptora ep4 prostaglandyny e2 (pge2) - Google Patents

Antagoniści receptora ep4 prostaglandyny e2 (pge2)

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Publication number
PL4038052T3
PL4038052T3 PL20785746.7T PL20785746T PL4038052T3 PL 4038052 T3 PL4038052 T3 PL 4038052T3 PL 20785746 T PL20785746 T PL 20785746T PL 4038052 T3 PL4038052 T3 PL 4038052T3
Authority
PL
Poland
Prior art keywords
pge2
prostaglandin
receptor antagonists
antagonists
receptor
Prior art date
Application number
PL20785746.7T
Other languages
English (en)
Inventor
Anne-Laure Blayo
Ismet Dorange
Gaël HOMMET
Baptiste Manteau
Stanislas Mayer
Stephan Schann
Original Assignee
Domain Therapeutics
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Domain Therapeutics filed Critical Domain Therapeutics
Publication of PL4038052T3 publication Critical patent/PL4038052T3/pl

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    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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    • C07D311/94—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings
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CA2473778A1 (en) * 2002-02-08 2003-08-14 Merck & Co., Inc. N-biphenylmethyl aminocycloalkanecarboxamide derivatives
KR100707123B1 (ko) * 2003-07-02 2007-04-16 그뤼넨탈 게엠베하 바닐로이드 수용체의 길항제로서 강력한 진통효과를나타내는 4-(메틸설포닐아미노)페닐 동족체 및 이를함유하는 약학적 조성물
CA2565813C (en) * 2004-05-04 2010-10-26 Pfizer Inc. Substituted methyl aryl or heteroaryl amide compounds
JP2009503078A (ja) * 2005-08-02 2009-01-29 メルク エンド カムパニー インコーポレーテッド アンドロゲン受容体モジュレーターとしてのｎ−（ピリジン−４−イル）−２−フェニルブタンアミド
WO2008016676A2 (en) * 2006-08-02 2008-02-07 Cytokinetics, Incorporated Certain chemical entities, compositions, and methods
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