PL3880675T3 - Związki antybiotykowe, sposoby ich wytwarzania, kompozycje farmaceutyczne zawierające te związki oraz ich zastosowanie - Google Patents

Związki antybiotykowe, sposoby ich wytwarzania, kompozycje farmaceutyczne zawierające te związki oraz ich zastosowanie

Info

Publication number
PL3880675T3
PL3880675T3 PL19805569.1T PL19805569T PL3880675T3 PL 3880675 T3 PL3880675 T3 PL 3880675T3 PL 19805569 T PL19805569 T PL 19805569T PL 3880675 T3 PL3880675 T3 PL 3880675T3
Authority
PL
Poland
Prior art keywords
compounds
manufacturing
methods
pharmaceutical compositions
compositions containing
Prior art date
Application number
PL19805569.1T
Other languages
English (en)
Inventor
Vincent Gerusz
Vasileios TATSIS
Mihiro Sunose
Juan Bravo
Terry Finn
Danig Pohin
Pierre-Michel REGENASS
Original Assignee
Debiopharm International Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Debiopharm International Sa filed Critical Debiopharm International Sa
Publication of PL3880675T3 publication Critical patent/PL3880675T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/499Spiro-condensed pyrazines or piperazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/20Spiro-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PL19805569.1T 2018-11-12 2019-11-11 Związki antybiotykowe, sposoby ich wytwarzania, kompozycje farmaceutyczne zawierające te związki oraz ich zastosowanie PL3880675T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP18205619 2018-11-12
EP18213016 2018-12-17
PCT/EP2019/080903 WO2020099341A1 (en) 2018-11-12 2019-11-11 Antibiotic compounds, methods of manufacturing the same, pharmaceutical compositions containing the same and uses thereof

Publications (1)

Publication Number Publication Date
PL3880675T3 true PL3880675T3 (pl) 2025-02-10

Family

ID=68610175

Family Applications (1)

Application Number Title Priority Date Filing Date
PL19805569.1T PL3880675T3 (pl) 2018-11-12 2019-11-11 Związki antybiotykowe, sposoby ich wytwarzania, kompozycje farmaceutyczne zawierające te związki oraz ich zastosowanie

Country Status (26)

Country Link
US (1) US20230035837A1 (pl)
EP (1) EP3880675B1 (pl)
JP (1) JP2022506957A (pl)
KR (1) KR102872166B1 (pl)
CN (1) CN113272302B (pl)
AU (1) AU2019380568B2 (pl)
BR (1) BR112021009106A2 (pl)
CA (1) CA3119390A1 (pl)
CL (2) CL2021001244A1 (pl)
DK (1) DK3880675T3 (pl)
ES (1) ES3009675T3 (pl)
FI (1) FI3880675T3 (pl)
HU (1) HUE069513T2 (pl)
IL (2) IL311894A (pl)
LT (1) LT3880675T (pl)
MX (2) MX2021005535A (pl)
PH (1) PH12021551058A1 (pl)
PL (1) PL3880675T3 (pl)
RS (1) RS66257B1 (pl)
SG (1) SG11202104863RA (pl)
SI (1) SI3880675T1 (pl)
SM (1) SMT202400519T1 (pl)
TN (1) TN2021000092A1 (pl)
UA (1) UA129248C2 (pl)
WO (1) WO2020099341A1 (pl)
ZA (1) ZA202103516B (pl)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL293980A (en) 2019-12-19 2022-08-01 Debiopharm Int Sa New compounds and their use
WO2022187329A1 (en) * 2021-03-03 2022-09-09 The Board Of Trustees Of The University Of Illinois Fabi inhibitors for gram-negative pathogens
CA3223459A1 (en) 2021-06-23 2022-12-29 Vincent Gerusz Novel compounds and their use
WO2025073269A1 (zh) * 2023-10-07 2025-04-10 广州白云山医药集团股份有限公司白云山制药总厂 一种FabI酶抑制剂及其应用
WO2025078209A1 (en) 2023-10-09 2025-04-17 Debiopharm International S.A. Antibiotic compounds for treating bacterial infections

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6921763B2 (en) 1999-09-17 2005-07-26 Abbott Laboratories Pyrazolopyrimidines as therapeutic agents
DE60017180T2 (de) * 1999-10-08 2005-12-08 Affinium Pharmaceuticals, Inc., Toronto Fab i inhibitoren
CA2444597A1 (en) * 2001-04-06 2002-10-06 Affinium Pharmaceuticals, Inc. Fab i inhibitors
CA2519429C (en) * 2003-03-17 2013-08-06 Affinium Pharmaceuticals, Inc. Pharmaceutical compositions comprising inhibitors of fab i and further antibiotics
US8450307B2 (en) * 2004-06-04 2013-05-28 Affinium Pharmaceuticals, Inc. Therapeutic agents, and methods of making and using the same
CN101415701A (zh) * 2005-12-05 2009-04-22 Affinium医药公司 作为fabi抑制剂的杂环丙烯酰胺化合物和抗菌剂
EP1973902A2 (en) 2005-12-05 2008-10-01 Affinium Pharmaceuticals, Inc. 3-heterocyclylacrylamide compounds as fabi inhibitors and antibacterial agents
US7601716B2 (en) 2006-05-01 2009-10-13 Cephalon, Inc. Pyridopyrazines and derivatives thereof as ALK and c-Met inhibitors
WO2008009122A1 (en) 2006-07-20 2008-01-24 Affinium Pharmaceuticals, Inc. Acrylamide derivatives as fab i inhibitors
EP2125802A4 (en) 2007-02-16 2014-08-20 Debiopharm Int Sa SALTS, PRODRUGS AND POLYMORPHES OF FAB I INHIBITORS
JO3611B1 (ar) 2011-08-10 2020-08-27 Janssen Sciences Ireland Uc سايكلو بنتا (سي (بيرول 4,3 ثاني هيدرو 1 hمستبدله [8,1] نافثيريدينونات مضادة للجراثيم
WO2013042035A1 (en) 2011-09-19 2013-03-28 Vitas Pharma Research Private Limited Heterocyclic compounds as inhibitors of fatty acid biosynthesis for bacterial infections
EP2785715A1 (en) 2011-12-02 2014-10-08 Aurigene Discovery Technologies Limited Substituted pyridine derivatives as fabi inhibitors
DK2861608T3 (da) * 2012-06-19 2019-06-24 Debiopharm Int Sa Prodrug-derivater af (e)-n-methyl-n-((3-methylbenzofuran-2-yl)methyl)-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)acrylamid
JP6250667B2 (ja) * 2012-08-10 2017-12-20 ヤンセン・サイエンシズ・アイルランド・ユーシー 新しい抗菌化合物
US9951056B2 (en) 2013-09-30 2018-04-24 Beijing Innocare Pharma Tech Co., Ltd. Substituted nicotinamide inhibitors of BTK and their preparation and use in the treatment of cancer, inflammation and autoimmune disease

Also Published As

Publication number Publication date
CL2022003703A1 (es) 2023-06-09
FI3880675T3 (fi) 2024-12-09
ZA202103516B (en) 2025-11-26
AU2019380568B2 (en) 2024-08-15
AU2019380568A1 (en) 2021-06-17
UA129248C2 (uk) 2025-02-26
CN113272302A (zh) 2021-08-17
IL282950A (en) 2021-06-30
JP2022506957A (ja) 2022-01-17
RS66257B1 (sr) 2024-12-31
HUE069513T2 (hu) 2025-03-28
MX2024010625A (es) 2024-09-05
KR102872166B1 (ko) 2025-10-15
BR112021009106A2 (pt) 2021-08-10
PH12021551058A1 (en) 2021-11-22
SG11202104863RA (en) 2021-06-29
LT3880675T (lt) 2024-12-27
WO2020099341A1 (en) 2020-05-22
CL2021001244A1 (es) 2021-11-19
IL311894A (en) 2024-06-01
NZ776487A (en) 2024-10-25
SMT202400519T1 (it) 2025-01-14
CA3119390A1 (en) 2020-05-22
EP3880675A1 (en) 2021-09-22
DK3880675T3 (da) 2024-12-02
TN2021000092A1 (en) 2023-01-05
SI3880675T1 (sl) 2025-02-28
CN113272302B (zh) 2024-08-13
MX2021005535A (es) 2021-09-08
EP3880675B1 (en) 2024-11-06
ES3009675T3 (en) 2025-03-31
US20230035837A1 (en) 2023-02-02
KR20210093292A (ko) 2021-07-27

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