PL3826686T3 - Stabilne, stężone roztwory kompleksów radionuklidów - Google Patents

Stabilne, stężone roztwory kompleksów radionuklidów

Info

Publication number
PL3826686T3
PL3826686T3 PL18783136.7T PL18783136T PL3826686T3 PL 3826686 T3 PL3826686 T3 PL 3826686T3 PL 18783136 T PL18783136 T PL 18783136T PL 3826686 T3 PL3826686 T3 PL 3826686T3
Authority
PL
Poland
Prior art keywords
radionuclid
complexes
stable
concentrated solutions
concentrated
Prior art date
Application number
PL18783136.7T
Other languages
English (en)
Inventor
Daniela Chicco
Donato BARBATO
Francesco DE PALO
Lorenza Fugazza
Maurizio Mariani
Giovanni TESORIERE
Clementina BRAMBATI
Original Assignee
Advanced Accelerator Applications S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/IB2018/055575 external-priority patent/WO2020021310A1/en
Priority claimed from US16/045,484 external-priority patent/US20200030465A1/en
Application filed by Advanced Accelerator Applications S.A. filed Critical Advanced Accelerator Applications S.A.
Publication of PL3826686T3 publication Critical patent/PL3826686T3/pl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/12Preparations containing radioactive substances for use in therapy or testing in vivo characterised by a special physical form, e.g. emulsion, microcapsules, liposomes, characterized by a special physical form, e.g. emulsions, dispersions, microcapsules
    • A61K51/121Solutions, i.e. homogeneous liquid formulation
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12Carboxylic acids; Salts or anhydrides thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183Amino acids, e.g. glycine, EDTA or aspartame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/22Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/0474Organic compounds complexes or complex-forming compounds, i.e. wherein a radioactive metal (e.g. 111In3+) is complexed or chelated by, e.g. a N2S2, N3S, NS3, N4 chelating group
    • A61K51/0478Organic compounds complexes or complex-forming compounds, i.e. wherein a radioactive metal (e.g. 111In3+) is complexed or chelated by, e.g. a N2S2, N3S, NS3, N4 chelating group complexes from non-cyclic ligands, e.g. EDTA, MAG3
    • A61K51/048DTPA (diethylenetriamine tetraacetic acid)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/0474Organic compounds complexes or complex-forming compounds, i.e. wherein a radioactive metal (e.g. 111In3+) is complexed or chelated by, e.g. a N2S2, N3S, NS3, N4 chelating group
    • A61K51/0482Organic compounds complexes or complex-forming compounds, i.e. wherein a radioactive metal (e.g. 111In3+) is complexed or chelated by, e.g. a N2S2, N3S, NS3, N4 chelating group chelates from cyclic ligands, e.g. DOTA
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/08Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/08Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins
    • A61K51/083Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins the peptide being octreotide or a somatostatin-receptor-binding peptide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/08Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins
    • A61K51/088Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins conjugates with carriers being peptides, polyamino acids or proteins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Optics & Photonics (AREA)
  • Physics & Mathematics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Dispersion Chemistry (AREA)
  • Dermatology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Peptides Or Proteins (AREA)
PL18783136.7T 2018-07-25 2018-09-25 Stabilne, stężone roztwory kompleksów radionuklidów PL3826686T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
PCT/IB2018/055575 WO2020021310A1 (en) 2018-07-25 2018-07-25 Stable, concentrated radionuclide complex solutions
US16/045,484 US20200030465A1 (en) 2018-07-25 2018-07-25 Stable, concentrated radionuclide complex solutions
PCT/IB2018/057415 WO2020021322A1 (en) 2018-07-25 2018-09-25 Stable, concentrated radionuclide complex solutions

Publications (1)

Publication Number Publication Date
PL3826686T3 true PL3826686T3 (pl) 2025-09-22

Family

ID=63794577

Family Applications (1)

Application Number Title Priority Date Filing Date
PL18783136.7T PL3826686T3 (pl) 2018-07-25 2018-09-25 Stabilne, stężone roztwory kompleksów radionuklidów

Country Status (23)

Country Link
EP (7) EP4541380B1 (pl)
JP (3) JP7402218B2 (pl)
KR (2) KR102865113B1 (pl)
CN (5) CN120860270A (pl)
AU (6) AU2018433575B2 (pl)
BR (1) BR112021001148A2 (pl)
CA (1) CA3153630A1 (pl)
CO (1) CO2021000506A2 (pl)
DE (3) DE202018007006U1 (pl)
DK (5) DK3826686T3 (pl)
ES (1) ES3038413T3 (pl)
FI (5) FI4545101T3 (pl)
HR (1) HRP20250912T1 (pl)
HU (1) HUE072720T2 (pl)
IL (4) IL319542A (pl)
LT (5) LT4541379T (pl)
MX (2) MX2021000805A (pl)
PL (1) PL3826686T3 (pl)
PT (5) PT4545101T (pl)
RS (2) RS67667B1 (pl)
SG (1) SG11202100645XA (pl)
SI (1) SI3826686T1 (pl)
WO (1) WO2020021322A1 (pl)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11541134B1 (en) 2021-08-02 2023-01-03 Rayzebio, Inc. Stabilized compositions of radionuclides and uses thereof
JPWO2023100852A1 (pl) * 2021-11-30 2023-06-08
KR20240146015A (ko) * 2022-02-04 2024-10-07 어드밴스드 엑셀러레이터 어플리케이션즈 방사성 핵종 복합체의 대규모 합성 방법
CN114404618A (zh) * 2022-03-28 2022-04-29 北京先通国际医药科技股份有限公司 放射性药物水溶液及其用途
CN114404619A (zh) * 2022-03-28 2022-04-29 北京先通国际医药科技股份有限公司 放射性药物水溶液及其制备方法和用途
CN116920129A (zh) * 2022-04-02 2023-10-24 北京先通国际医药科技股份有限公司 放射性药物水溶液及其制备方法和用途
WO2026006569A1 (en) * 2024-06-27 2026-01-02 Curium Us Llc 177lutetium-dota-tate formulations

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2779780A (en) 1955-03-01 1957-01-29 Du Pont 1, 4-diamino-2, 3-dicyano-1, 4-bis (substituted mercapto) butadienes and their preparation
US4261989A (en) 1979-02-19 1981-04-14 Kaken Chemical Co. Ltd. Geldanamycin derivatives and antitumor drug
EP0647450A1 (en) 1993-09-09 1995-04-12 BEHRINGWERKE Aktiengesellschaft Improved prodrugs for enzyme mediated activation
US6066309A (en) * 1996-02-02 2000-05-23 Rhomed Incorporated Post-labeling stabilization of radiolabeled proteins and peptides
EP1143957A3 (en) 1998-12-16 2002-02-27 Warner-Lambert Company Treatment of arthritis with mek inhibitors
CA2416685C (en) 2000-07-19 2008-10-07 Warner-Lambert Company Oxygenated esters of 4-iodo phenylamino benzhydroxamic acids
US6995162B2 (en) 2001-01-12 2006-02-07 Amgen Inc. Substituted alkylamine derivatives and methods of use
JP4547911B2 (ja) 2002-02-01 2010-09-22 アリアド・ファーマシューティカルズ・インコーポレイテッド リン含有化合物およびその用途
WO2003076424A1 (en) 2002-03-08 2003-09-18 Eisai Co. Ltd. Macrocyclic compounds useful as pharmaceuticals
DE60330227D1 (de) 2002-03-13 2010-01-07 Array Biopharma Inc N3-alkylierte benzimidazol-derivate als mek-hemmer
TWI275390B (en) 2002-04-30 2007-03-11 Wyeth Corp Process for the preparation of 7-substituted-3- quinolinecarbonitriles
JP5139678B2 (ja) * 2003-07-24 2013-02-06 ブラッコ・イメージング・ソシエタ・ペル・アチオニ 安定な放射性医薬品組成物およびその製法
ES2481402T3 (es) 2005-07-21 2014-07-30 Ardea Biosciences, Inc. Inhibidores de N-(arilamino)sulfonamida de MEK
WO2008009444A1 (en) 2006-07-19 2008-01-24 Van Dulmen, Adrianus, A. Use of ethanol for stabilizing a single-vial liquid formulation of a radiolabeled peptide
JP7242538B2 (ja) * 2016-11-04 2023-03-20 クラリティー・ファーマシューティカルズ・リミテッド 放射線治療及び画像診断のための製剤
US10596276B2 (en) 2018-07-25 2020-03-24 Advanced Accelerator Applications (Italy) S.R.L. Stable, concentrated radionuclide complex solutions

Also Published As

Publication number Publication date
AU2018433575A1 (en) 2021-02-11
CN112584875A (zh) 2021-03-30
EP4541379B1 (en) 2025-11-19
AU2025204901B2 (en) 2025-09-18
EP3826686A1 (en) 2021-06-02
EP4545100A3 (en) 2025-07-23
IL280314A (en) 2021-03-25
BR112021001148A2 (pt) 2021-04-20
FI4541379T3 (fi) 2026-02-17
IL313560A (en) 2024-08-01
DK4541379T3 (da) 2026-02-02
FI4545101T3 (fi) 2026-02-24
PT4545101T (pt) 2026-02-24
DK3826686T3 (da) 2025-08-25
LT4541379T (lt) 2026-02-10
EP4541380B1 (en) 2025-12-10
EP4541381A3 (en) 2025-07-23
LT4545101T (lt) 2026-03-10
DE202018006567U1 (de) 2021-02-22
CA3153630A1 (en) 2020-01-30
EP4541380A2 (en) 2025-04-23
LT3826686T (lt) 2025-08-25
JP2023117417A (ja) 2023-08-23
JP7402218B2 (ja) 2023-12-20
AU2022203683A1 (en) 2022-06-16
RS67667B1 (sr) 2026-02-27
SG11202100645XA (en) 2021-02-25
JP7796696B2 (ja) 2026-01-09
EP4640241A3 (en) 2025-12-10
PT4541380T (pt) 2026-02-24
KR20250017751A (ko) 2025-02-04
CN121081692A (zh) 2025-12-09
KR20240033296A (ko) 2024-03-12
FI4545100T3 (fi) 2026-03-02
KR20210035855A (ko) 2021-04-01
EP4545101B1 (en) 2025-12-10
FI3826686T3 (fi) 2025-08-20
EP3826686B1 (en) 2025-05-21
AU2024201217A1 (en) 2024-03-14
IL313560B2 (en) 2025-11-01
AU2024201217B2 (en) 2025-02-27
IL313560B1 (en) 2025-07-01
PT4545100T (pt) 2026-02-16
AU2022203683B2 (en) 2023-12-21
CO2021000506A2 (es) 2021-04-19
HRP20250912T1 (hr) 2025-09-26
AU2025202231A1 (en) 2025-04-17
CN120860270A (zh) 2025-10-31
DE202018007007U1 (de) 2025-10-08
PT3826686T (pt) 2025-08-04
RS67034B1 (sr) 2025-08-29
IL319542A (en) 2025-05-01
EP4640241A2 (en) 2025-10-29
EP4545101A2 (en) 2025-04-30
DK4545100T3 (da) 2026-02-23
AU2025204901A1 (en) 2025-07-17
LT4545100T (lt) 2026-02-25
EP4545101A3 (en) 2025-07-23
EP4541381A2 (en) 2025-04-23
EP4541381B1 (en) 2026-02-04
LT4541380T (lt) 2026-03-10
ES3038413T3 (en) 2025-10-13
KR102643582B1 (ko) 2024-03-05
EP4541379A2 (en) 2025-04-23
KR102865113B1 (ko) 2025-09-26
FI4541380T3 (fi) 2026-03-02
DK4541380T3 (da) 2026-02-23
AU2025220852A1 (en) 2025-09-11
CN120860272A (zh) 2025-10-31
CN120860271A (zh) 2025-10-31
AU2018433575B2 (en) 2022-07-07
IL319541B2 (en) 2026-01-01
DE202018007006U1 (de) 2025-10-08
MX2025012060A (es) 2025-11-03
EP4541380A3 (en) 2025-07-23
MX2021000805A (es) 2021-05-12
JP2022501313A (ja) 2022-01-06
IL319541A (en) 2025-05-01
IL319541B1 (en) 2025-09-01
EP4545100B1 (en) 2025-12-10
WO2020021322A1 (en) 2020-01-30
HUE072720T2 (hu) 2025-12-28
EP4541379A3 (en) 2025-07-23
JP2025111424A (ja) 2025-07-30
DK4545101T3 (da) 2026-03-02
SI3826686T1 (sl) 2025-09-30
PT4541379T (pt) 2026-01-29
AU2025220852B2 (en) 2025-10-23
EP4545100A2 (en) 2025-04-30

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