PL3470400T3 - Krystaliczne postacie ozanimodu i chlorowodorku ozanimodu oraz sposoby ich otrzymywania - Google Patents

Krystaliczne postacie ozanimodu i chlorowodorku ozanimodu oraz sposoby ich otrzymywania

Info

Publication number
PL3470400T3
PL3470400T3 PL17812728.8T PL17812728T PL3470400T3 PL 3470400 T3 PL3470400 T3 PL 3470400T3 PL 17812728 T PL17812728 T PL 17812728T PL 3470400 T3 PL3470400 T3 PL 3470400T3
Authority
PL
Poland
Prior art keywords
ozanimod
processes
preparation
crystalline forms
hydrochloride
Prior art date
Application number
PL17812728.8T
Other languages
English (en)
Inventor
Minhua Chen
Yanfeng Zhang
Xiaoting ZHAI
Kaiqiang YAN
Chaohui YANG
Xiaoyu Zhang
Original Assignee
Receptos Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=60663299&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL3470400(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Receptos Llc filed Critical Receptos Llc
Publication of PL3470400T3 publication Critical patent/PL3470400T3/pl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurosurgery (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Hospice & Palliative Care (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PL17812728.8T 2016-06-14 2017-06-14 Krystaliczne postacie ozanimodu i chlorowodorku ozanimodu oraz sposoby ich otrzymywania PL3470400T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN201610416179 2016-06-14
CN201610493910 2016-06-29
PCT/CN2017/088314 WO2017215617A1 (zh) 2016-06-14 2017-06-14 奥扎莫德的晶型、其盐酸盐的晶型及其制备方法

Publications (1)

Publication Number Publication Date
PL3470400T3 true PL3470400T3 (pl) 2025-08-04

Family

ID=60663299

Family Applications (1)

Application Number Title Priority Date Filing Date
PL17812728.8T PL3470400T3 (pl) 2016-06-14 2017-06-14 Krystaliczne postacie ozanimodu i chlorowodorku ozanimodu oraz sposoby ich otrzymywania

Country Status (15)

Country Link
US (2) US11111223B2 (pl)
EP (2) EP3470400B1 (pl)
CN (2) CN114957157A (pl)
DK (1) DK3470400T5 (pl)
ES (1) ES3022204T3 (pl)
FI (1) FI3470400T3 (pl)
HR (1) HRP20250558T1 (pl)
HU (1) HUE072197T2 (pl)
LT (1) LT3470400T (pl)
PL (1) PL3470400T3 (pl)
PT (1) PT3470400T (pl)
RS (1) RS66905B1 (pl)
SI (1) SI3470400T1 (pl)
SM (1) SMT202500228T1 (pl)
WO (1) WO2017215617A1 (pl)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES3022204T3 (en) 2016-06-14 2025-05-28 Receptos Llc Crystalline forms of ozanimod and ozanimod hydrochloride, and processes for preparation thereof
US11028060B2 (en) 2016-08-19 2021-06-08 Receptos Llc Crystalline forms of ozanimod and processes for preparation thereof
WO2018050091A1 (zh) 2016-09-14 2018-03-22 苏州科睿思制药有限公司 奥扎莫德盐酸盐的晶型及其制备方法
MA48798B1 (fr) * 2017-05-22 2023-10-31 Egyt Gyogyszervegyeszeti Gyar Procédé de production d'ozanimod
CN109280035B (zh) * 2017-07-19 2023-06-09 广东东阳光药业有限公司 奥扎莫德的多晶型及其制备方法
EP3677575A4 (en) 2017-08-31 2020-07-15 Crystal Pharmaceutical (Suzhou) Co., Ltd. CRYSTALLINE FORM OF OZANIMODHYDROCHLORIDE AND PRODUCTION METHOD THEREFOR
CN107840830A (zh) * 2017-09-20 2018-03-27 广东东阳光药业有限公司 盐酸奥扎莫德无水晶型i
WO2019094409A1 (en) 2017-11-07 2019-05-16 Teva Pharmaceuticals International Gmbh Salts and solid state forms of ozanimod
WO2020152718A1 (en) * 2019-01-25 2020-07-30 Mylan Laboratories Limited Polymorphic forms 5-[3-[(1s)-2,3-dihydro-1-[(2-hydroxyethyl) amino]-1h-inden-4-yl]-1,2,4-oxadiazol-5-yl]-2-(1-methylethoxy)benzonitrile
EP3999495A1 (en) 2019-07-16 2022-05-25 Synthon B.V. Improved process for preparing ozanimod
EP4126826A1 (en) * 2020-04-02 2023-02-08 Synthon B.V. Crystalline form of ozanimod hydrochloride
WO2023152767A1 (en) 2022-02-11 2023-08-17 Mylan Laboratories Limited Polymorphic forms of ozanimod hydrochloride
WO2024246174A1 (en) 2023-05-31 2024-12-05 Química Sintética, S.A. Amorphous and crystalline form of ozanimod hydrochloride

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL2291080T3 (pl) 2008-05-14 2015-12-31 Scripps Research Inst Nowe modulatory receptorów sfingozyno-1-fosforanu
DK2913326T3 (da) 2008-05-14 2020-08-17 Scripps Research Inst Hidtil ukendte modulatorer af sphingosinphosphatreceptorer
CA2780772C (en) * 2009-11-13 2018-01-16 Receptos, Inc. Selective sphingosine 1 phosphate receptor modulators and methods of chiral synthesis
EP3062792A1 (en) 2013-11-01 2016-09-07 Celgene International II Sarl Selective sphingosine 1 phosphate receptor modulators and combination therapy therewith
CA2981743A1 (en) * 2015-04-06 2016-10-13 Auspex Pharmaceuticals, Inc. Deuterium-substituted oxadiazoles
ES3022204T3 (en) 2016-06-14 2025-05-28 Receptos Llc Crystalline forms of ozanimod and ozanimod hydrochloride, and processes for preparation thereof
US11028060B2 (en) 2016-08-19 2021-06-08 Receptos Llc Crystalline forms of ozanimod and processes for preparation thereof
WO2018050091A1 (zh) 2016-09-14 2018-03-22 苏州科睿思制药有限公司 奥扎莫德盐酸盐的晶型及其制备方法
CN108137516A (zh) 2016-09-14 2018-06-08 杭州领业医药科技有限公司 奥扎莫德的晶型、其制备方法及药物组合物
US20200031784A1 (en) * 2017-04-07 2020-01-30 Solipharma Llc Ozanimod addition salt crystal, preparation method, pharmaceutical composition, and uses
EP3677575A4 (en) 2017-08-31 2020-07-15 Crystal Pharmaceutical (Suzhou) Co., Ltd. CRYSTALLINE FORM OF OZANIMODHYDROCHLORIDE AND PRODUCTION METHOD THEREFOR
CN107840830A (zh) 2017-09-20 2018-03-27 广东东阳光药业有限公司 盐酸奥扎莫德无水晶型i

Also Published As

Publication number Publication date
PT3470400T (pt) 2025-04-29
HUE072197T2 (hu) 2025-10-28
CN109219597A (zh) 2019-01-15
CN114957157A (zh) 2022-08-30
HRP20250558T1 (hr) 2025-07-04
DK3470400T3 (da) 2025-06-16
SMT202500228T1 (it) 2025-07-22
FI3470400T3 (fi) 2025-06-13
US20190337908A1 (en) 2019-11-07
LT3470400T (lt) 2025-07-10
EP3470400B1 (en) 2025-04-02
RS66905B1 (sr) 2025-07-31
WO2017215617A1 (zh) 2017-12-21
ES3022204T3 (en) 2025-05-28
EP3470400A1 (en) 2019-04-17
EP4566676A3 (en) 2025-11-05
US20200157065A1 (en) 2020-05-21
DK3470400T5 (da) 2025-06-30
EP4566676A2 (en) 2025-06-11
US11680050B2 (en) 2023-06-20
SI3470400T1 (sl) 2025-09-30
US11111223B2 (en) 2021-09-07
EP3470400A4 (en) 2019-04-17

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