PL3169666T3 - Podstawione pochodne azaspiro(4,5)dekanu - Google Patents
Podstawione pochodne azaspiro(4,5)dekanuInfo
- Publication number
- PL3169666T3 PL3169666T3 PL15738274T PL15738274T PL3169666T3 PL 3169666 T3 PL3169666 T3 PL 3169666T3 PL 15738274 T PL15738274 T PL 15738274T PL 15738274 T PL15738274 T PL 15738274T PL 3169666 T3 PL3169666 T3 PL 3169666T3
- Authority
- PL
- Poland
- Prior art keywords
- decane derivatives
- substituted azaspiro
- azaspiro
- substituted
- decane
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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- A—HUMAN NECESSITIES
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/541—Non-condensed thiazines containing further heterocyclic rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C—CHEMISTRY; METALLURGY
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- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
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- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Neurology (AREA)
- Neurosurgery (AREA)
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- Pain & Pain Management (AREA)
- Addiction (AREA)
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- Diabetes (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14002439 | 2014-07-15 | ||
| PCT/EP2015/001445 WO2016008582A1 (en) | 2014-07-15 | 2015-07-14 | Substituted azaspiro(4.5)decane derivatives |
| EP15738274.8A EP3169666B1 (en) | 2014-07-15 | 2015-07-14 | Substituted azaspiro(4.5)decane derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PL3169666T3 true PL3169666T3 (pl) | 2019-03-29 |
Family
ID=51211484
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL15738274T PL3169666T3 (pl) | 2014-07-15 | 2015-07-14 | Podstawione pochodne azaspiro(4,5)dekanu |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US10214520B2 (pl) |
| EP (1) | EP3169666B1 (pl) |
| JP (1) | JP6509321B2 (pl) |
| CN (1) | CN106660954A (pl) |
| AU (1) | AU2015291467B2 (pl) |
| BR (1) | BR112017000762A2 (pl) |
| CA (1) | CA2955071A1 (pl) |
| CY (1) | CY1120812T1 (pl) |
| DK (1) | DK3169666T3 (pl) |
| EA (1) | EA201790185A1 (pl) |
| ES (1) | ES2686326T3 (pl) |
| HR (1) | HRP20181112T1 (pl) |
| HU (1) | HUE040133T2 (pl) |
| LT (1) | LT3169666T (pl) |
| MX (1) | MX2017000520A (pl) |
| PL (1) | PL3169666T3 (pl) |
| PT (1) | PT3169666T (pl) |
| RS (1) | RS57732B1 (pl) |
| SI (1) | SI3169666T1 (pl) |
| WO (1) | WO2016008582A1 (pl) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
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| WO2019152688A1 (en) * | 2018-01-31 | 2019-08-08 | Aptinyx Inc. | Spiro-lactam nmda receptor modulators and uses thereof |
| CN111518016B (zh) * | 2018-06-01 | 2022-02-25 | 厦门宝太生物科技股份有限公司 | 一种csf1r抑制剂中间体及其制备方法 |
| CN111848423B (zh) * | 2019-04-30 | 2022-10-14 | 尚科生物医药(上海)有限公司 | 3-氧代环丁基氨基甲酸叔丁酯的制备方法 |
| CN112679405B (zh) * | 2019-10-17 | 2023-12-15 | 南京富润凯德生物医药有限公司 | 一种(s)-7-氧杂-2-氮杂螺[4.5]癸烷衍生物的制备方法 |
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-
2015
- 2015-07-14 DK DK15738274.8T patent/DK3169666T3/en active
- 2015-07-14 CN CN201580038275.7A patent/CN106660954A/zh active Pending
- 2015-07-14 RS RS20181037A patent/RS57732B1/sr unknown
- 2015-07-14 HR HRP20181112TT patent/HRP20181112T1/hr unknown
- 2015-07-14 PT PT15738274T patent/PT3169666T/pt unknown
- 2015-07-14 MX MX2017000520A patent/MX2017000520A/es unknown
- 2015-07-14 LT LTEP15738274.8T patent/LT3169666T/lt unknown
- 2015-07-14 EA EA201790185A patent/EA201790185A1/ru unknown
- 2015-07-14 JP JP2017502138A patent/JP6509321B2/ja not_active Expired - Fee Related
- 2015-07-14 BR BR112017000762A patent/BR112017000762A2/pt not_active Application Discontinuation
- 2015-07-14 WO PCT/EP2015/001445 patent/WO2016008582A1/en not_active Ceased
- 2015-07-14 CA CA2955071A patent/CA2955071A1/en not_active Abandoned
- 2015-07-14 SI SI201530319T patent/SI3169666T1/en unknown
- 2015-07-14 HU HUE15738274A patent/HUE040133T2/hu unknown
- 2015-07-14 EP EP15738274.8A patent/EP3169666B1/en not_active Not-in-force
- 2015-07-14 PL PL15738274T patent/PL3169666T3/pl unknown
- 2015-07-14 ES ES15738274T patent/ES2686326T3/es active Active
- 2015-07-14 US US15/326,138 patent/US10214520B2/en not_active Expired - Fee Related
- 2015-07-14 AU AU2015291467A patent/AU2015291467B2/en not_active Ceased
-
2018
- 2018-09-04 CY CY181100914T patent/CY1120812T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN106660954A (zh) | 2017-05-10 |
| LT3169666T (lt) | 2018-08-10 |
| BR112017000762A2 (pt) | 2017-11-21 |
| MX2017000520A (es) | 2017-05-01 |
| DK3169666T3 (en) | 2018-07-30 |
| EP3169666B1 (en) | 2018-06-06 |
| WO2016008582A1 (en) | 2016-01-21 |
| ES2686326T3 (es) | 2018-10-17 |
| AU2015291467A1 (en) | 2017-03-09 |
| JP2017520601A (ja) | 2017-07-27 |
| EP3169666A1 (en) | 2017-05-24 |
| CY1120812T1 (el) | 2019-12-11 |
| JP6509321B2 (ja) | 2019-05-08 |
| US20170210734A1 (en) | 2017-07-27 |
| CA2955071A1 (en) | 2016-01-21 |
| US10214520B2 (en) | 2019-02-26 |
| EA201790185A1 (ru) | 2017-07-31 |
| HUE040133T2 (hu) | 2019-02-28 |
| SI3169666T1 (en) | 2018-08-31 |
| WO2016008582A8 (en) | 2016-03-24 |
| AU2015291467B2 (en) | 2019-01-24 |
| RS57732B1 (sr) | 2018-12-31 |
| PT3169666T (pt) | 2018-10-19 |
| HRP20181112T1 (hr) | 2018-09-21 |
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