PL2477990T3 - Pochodne 5-fenylopirazolopirydyny, ich wytwarzanie oraz ich zastosowanie terapeutyczne - Google Patents
Pochodne 5-fenylopirazolopirydyny, ich wytwarzanie oraz ich zastosowanie terapeutyczneInfo
- Publication number
- PL2477990T3 PL2477990T3 PL10771159T PL10771159T PL2477990T3 PL 2477990 T3 PL2477990 T3 PL 2477990T3 PL 10771159 T PL10771159 T PL 10771159T PL 10771159 T PL10771159 T PL 10771159T PL 2477990 T3 PL2477990 T3 PL 2477990T3
- Authority
- PL
- Poland
- Prior art keywords
- phenyl
- preparation
- therapeutic use
- pyrazolopyridine derivatives
- pyrazolopyridine
- Prior art date
Links
- FXUDQKREGGIUQW-UHFFFAOYSA-N 5-phenyl-1h-pyrazolo[4,3-b]pyridine Chemical class N1=C2C=NNC2=CC=C1C1=CC=CC=C1 FXUDQKREGGIUQW-UHFFFAOYSA-N 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/06—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Anesthesiology (AREA)
- Addiction (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0956444A FR2950344B1 (fr) | 2009-09-18 | 2009-09-18 | Derives de 5-phenyl-pyrazolopyridine, leur preparation et leur aplication en therapeutique. |
| PCT/FR2010/051932 WO2011033230A1 (fr) | 2009-09-18 | 2010-09-17 | Dérivés de 5-phenyl-pyrazolopyridine, leur préparation et leur application en thérapeutique |
| EP10771159.0A EP2477990B1 (fr) | 2009-09-18 | 2010-09-17 | Dérivés de 5-phenyl-pyrazolopyridine, leur préparation et leur application en thérapeutique |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PL2477990T3 true PL2477990T3 (pl) | 2015-02-27 |
Family
ID=41572488
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL10771159T PL2477990T3 (pl) | 2009-09-18 | 2010-09-17 | Pochodne 5-fenylopirazolopirydyny, ich wytwarzanie oraz ich zastosowanie terapeutyczne |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US8618301B2 (pl) |
| EP (1) | EP2477990B1 (pl) |
| JP (1) | JP5616453B2 (pl) |
| AR (1) | AR078180A1 (pl) |
| CY (1) | CY1116581T1 (pl) |
| DK (1) | DK2477990T3 (pl) |
| ES (1) | ES2523505T3 (pl) |
| FR (1) | FR2950344B1 (pl) |
| HR (1) | HRP20141119T1 (pl) |
| JO (1) | JO3017B1 (pl) |
| PL (1) | PL2477990T3 (pl) |
| PT (1) | PT2477990E (pl) |
| SI (1) | SI2477990T1 (pl) |
| TW (1) | TWI464169B (pl) |
| UY (1) | UY32894A (pl) |
| WO (1) | WO2011033230A1 (pl) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2953520B1 (fr) * | 2009-12-04 | 2011-11-25 | Sanofi Aventis | Derives de diphenyl-pyrazolopyridines, leur preparation et leur application en therapeutique |
| JP2024525792A (ja) * | 2021-07-16 | 2024-07-12 | サノフイ | 治療に使用するための6H-イミダゾ[1,2-a]ピロロ[2,3-e]ピリジン誘導体 |
| EP4370518A1 (en) * | 2021-07-16 | 2024-05-22 | Sanofi | Imidazo[1,2-b][1,2,4]triazol derivatives for use in therapy |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2308457C2 (ru) * | 2001-04-27 | 2007-10-20 | Эйсай Ар Энд Ди Менеджмент Ко., Лтд. | Пиразоло [1, 5-а] пиридины и содержащие их лекарственные средства |
| AU2003220190A1 (en) * | 2002-03-13 | 2003-09-29 | Pharmacia & Upjohn Company Llc | Pyrazolo(1,5-a)pyridine derivatives as neurotransmitter modulators |
| JP4890439B2 (ja) * | 2005-03-07 | 2012-03-07 | 杏林製薬株式会社 | ピラゾロピリジン−4−イルピリダジノン誘導体とその付加塩及びそれらを有効成分とするpde阻害剤 |
| FR2906250B1 (fr) * | 2006-09-22 | 2008-10-31 | Sanofi Aventis Sa | Derives de 2-aryl-6phenyl-imidazo(1,2-a) pyridines, leur preparation et leur application en therapeutique |
| MX2009006706A (es) * | 2006-12-22 | 2009-07-02 | Astex Therapeutics Ltd | Compuestos heterociclicos biciclicos como inhibidores del receptor del factor de crecimiento de fibroblastos. |
| MX2009006704A (es) * | 2006-12-22 | 2009-06-30 | Astex Therapeutics Ltd | Derivados de amina triciclicos como inhibidores de proteina de tirosina cinasa. |
| FR2925900B1 (fr) * | 2008-01-02 | 2011-03-04 | Sanofi Aventis | DERIVES DE N-PHENYL-IMIDAZO°1,2-a!PYRIDINE-2-CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE |
| FR2928922B1 (fr) * | 2008-03-21 | 2010-04-23 | Sanofi Aventis | Derives de 2-aryl-6-phenyl-imidazo°1,2-a!pyridines polysubstitues, leur preparation et leur application en therapeutique |
| FR2953520B1 (fr) * | 2009-12-04 | 2011-11-25 | Sanofi Aventis | Derives de diphenyl-pyrazolopyridines, leur preparation et leur application en therapeutique |
-
2009
- 2009-09-18 FR FR0956444A patent/FR2950344B1/fr not_active Expired - Fee Related
-
2010
- 2010-09-16 AR ARP100103375A patent/AR078180A1/es unknown
- 2010-09-16 JO JOP/2010/0315A patent/JO3017B1/ar active
- 2010-09-17 DK DK10771159.0T patent/DK2477990T3/en active
- 2010-09-17 PL PL10771159T patent/PL2477990T3/pl unknown
- 2010-09-17 HR HRP20141119AT patent/HRP20141119T1/hr unknown
- 2010-09-17 SI SI201030792T patent/SI2477990T1/sl unknown
- 2010-09-17 UY UY0001032894A patent/UY32894A/es not_active Application Discontinuation
- 2010-09-17 ES ES10771159.0T patent/ES2523505T3/es active Active
- 2010-09-17 US US13/496,118 patent/US8618301B2/en not_active Expired - Fee Related
- 2010-09-17 TW TW099131736A patent/TWI464169B/zh not_active IP Right Cessation
- 2010-09-17 JP JP2012529329A patent/JP5616453B2/ja not_active Expired - Fee Related
- 2010-09-17 WO PCT/FR2010/051932 patent/WO2011033230A1/fr not_active Ceased
- 2010-09-17 EP EP10771159.0A patent/EP2477990B1/fr not_active Not-in-force
- 2010-09-17 PT PT107711590T patent/PT2477990E/pt unknown
-
2014
- 2014-11-20 CY CY20141100967T patent/CY1116581T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2011033230A1 (fr) | 2011-03-24 |
| US20130023554A1 (en) | 2013-01-24 |
| CY1116581T1 (el) | 2018-03-07 |
| TWI464169B (zh) | 2014-12-11 |
| JO3017B1 (ar) | 2016-09-05 |
| TW201118093A (en) | 2011-06-01 |
| UY32894A (es) | 2011-04-29 |
| AR078180A1 (es) | 2011-10-19 |
| ES2523505T3 (es) | 2014-11-26 |
| FR2950344A1 (fr) | 2011-03-25 |
| JP2013505227A (ja) | 2013-02-14 |
| HRP20141119T1 (hr) | 2015-01-30 |
| PT2477990E (pt) | 2014-11-27 |
| EP2477990A1 (fr) | 2012-07-25 |
| US8618301B2 (en) | 2013-12-31 |
| EP2477990B1 (fr) | 2014-08-20 |
| JP5616453B2 (ja) | 2014-10-29 |
| SI2477990T1 (sl) | 2014-12-31 |
| DK2477990T3 (en) | 2014-12-01 |
| FR2950344B1 (fr) | 2011-11-25 |
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