PH12022550937A1 - Pharmaceutical composition comprising selexipag - Google Patents
Pharmaceutical composition comprising selexipagInfo
- Publication number
- PH12022550937A1 PH12022550937A1 PH1/2022/550937A PH12022550937A PH12022550937A1 PH 12022550937 A1 PH12022550937 A1 PH 12022550937A1 PH 12022550937 A PH12022550937 A PH 12022550937A PH 12022550937 A1 PH12022550937 A1 PH 12022550937A1
- Authority
- PH
- Philippines
- Prior art keywords
- selexipag
- pharmaceutical composition
- diphenylpyrazin
- butyloxy
- isopropylamino
- Prior art date
Links
- QXWZQTURMXZVHJ-UHFFFAOYSA-N selexipag Chemical compound C=1C=CC=CC=1C1=NC(N(CCCCOCC(=O)NS(C)(=O)=O)C(C)C)=CN=C1C1=CC=CC=C1 QXWZQTURMXZVHJ-UHFFFAOYSA-N 0.000 title abstract 5
- 229960003841 selexipag Drugs 0.000 title abstract 4
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Physiology (AREA)
- Nutrition Science (AREA)
- Pulmonology (AREA)
- Diabetes (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Dermatology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP2019078905 | 2019-10-23 | ||
| PCT/EP2020/079698 WO2021078835A1 (en) | 2019-10-23 | 2020-10-22 | Pharmaceutical composition comprising selexipag |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PH12022550937A1 true PH12022550937A1 (en) | 2023-06-14 |
Family
ID=75620412
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PH1/2022/550937A PH12022550937A1 (en) | 2019-10-23 | 2020-10-22 | Pharmaceutical composition comprising selexipag |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20220401441A1 (https=) |
| EP (1) | EP4048235A1 (https=) |
| JP (2) | JP7646646B2 (https=) |
| KR (1) | KR20220087443A (https=) |
| CN (1) | CN114555088A (https=) |
| AU (1) | AU2020369912A1 (https=) |
| BR (1) | BR112022007207A2 (https=) |
| CA (1) | CA3154802A1 (https=) |
| EC (1) | ECSP22040921A (https=) |
| IL (1) | IL292354A (https=) |
| JO (1) | JOP20220093A1 (https=) |
| MX (1) | MX2022004882A (https=) |
| PE (1) | PE20221455A1 (https=) |
| PH (1) | PH12022550937A1 (https=) |
| WO (1) | WO2021078835A1 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TR2022005274A1 (tr) * | 2022-04-05 | 2023-10-23 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Seleksi̇pag'in bi̇r kati di̇spersi̇yonunu i̇çeren bi̇r fi̇lm kapli tablet |
| TR2022005277A2 (tr) * | 2022-04-05 | 2023-10-23 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Yaş granülasyon i̇le i̇şlenmi̇ş seleksi̇pag i̇çeren bi̇r fi̇lm kapli tablet |
| TR2022005273A2 (tr) * | 2022-04-05 | 2023-10-23 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Seleksi̇pag i̇çeren bi̇r fi̇lm kapli tablet |
| TR2022020995A1 (tr) * | 2022-12-28 | 2024-07-22 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Seleksi̇pag i̇çeren bi̇r tablet formülasyonu |
| CN116392491A (zh) * | 2023-04-11 | 2023-07-07 | 广东省实验动物监测所 | 司来帕格的药物组合物及其制备方法 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI316055B (https=) | 2001-04-26 | 2009-10-21 | Nippon Shinyaku Co Ltd | |
| CN104761509A (zh) | 2008-02-28 | 2015-07-08 | 日本新药株式会社 | 纤维化抑制剂 |
| WO2009154246A1 (ja) | 2008-06-19 | 2009-12-23 | 日本新薬株式会社 | 勃起不全治療剤 |
| WO2009157397A1 (ja) | 2008-06-23 | 2009-12-30 | 日本新薬株式会社 | 非ステロイド性抗炎症剤投与に伴う腸管傷害治療剤 |
| HRP20151443T1 (hr) | 2008-06-23 | 2016-01-29 | Nippon Shinyaku Co., Ltd. | Terapijsko sredstvo protiv stenoze kralježniäśnog kanala |
| CN102065864B (zh) | 2008-06-23 | 2012-11-21 | 日本新药株式会社 | 炎性肠病治疗剂 |
| LT2447254T (lt) | 2009-06-26 | 2018-01-10 | Nippon Shinyaku Co., Ltd. | Kristalai |
| WO2011024874A1 (ja) | 2009-08-26 | 2011-03-03 | 日本新薬株式会社 | 塩基付加塩 |
| HK1198358A1 (en) | 2011-08-12 | 2015-04-10 | Ascendis Pharma A/S | Sustained release composition of prostacyclin |
| EP2913047B1 (en) | 2012-10-29 | 2019-05-08 | Cardio Incorporated | Pulmonary disease-specific therapeutic agent |
| PT4331607T (pt) * | 2015-12-02 | 2025-05-22 | Nippon Shinyaku Co Ltd | Composição farmacêutica sólida que contém 2-{4-[n-(5,6-difenilpirazin-2-il)-n-isopropilamino]butiloxi}-n-(metil-sulfonil)acetamida |
| JOP20190204A1 (ar) | 2017-03-08 | 2019-09-05 | Actelion Pharmaceuticals Ltd | تركيبة صيدلانية تشتمل على سيليكسيباغ |
| TW201936175A (zh) * | 2018-02-21 | 2019-09-16 | 日商日本新藥股份有限公司 | 粒狀組合物、粒狀組合物之製造方法、及粒狀組合物之溶出性改善方法 |
| JP2022532076A (ja) * | 2019-05-06 | 2022-07-13 | アクテリオン ファーマシューティカルズ リミテッド | サルコイドーシス関連肺高血圧症の治療方法 |
-
2020
- 2020-10-22 CN CN202080071283.2A patent/CN114555088A/zh active Pending
- 2020-10-22 PH PH1/2022/550937A patent/PH12022550937A1/en unknown
- 2020-10-22 CA CA3154802A patent/CA3154802A1/en active Pending
- 2020-10-22 EP EP20792448.1A patent/EP4048235A1/en active Pending
- 2020-10-22 PE PE2022000625A patent/PE20221455A1/es unknown
- 2020-10-22 KR KR1020227012736A patent/KR20220087443A/ko not_active Withdrawn
- 2020-10-22 MX MX2022004882A patent/MX2022004882A/es unknown
- 2020-10-22 JP JP2022523448A patent/JP7646646B2/ja active Active
- 2020-10-22 WO PCT/EP2020/079698 patent/WO2021078835A1/en not_active Ceased
- 2020-10-22 IL IL292354A patent/IL292354A/en unknown
- 2020-10-22 JO JOP/2022/0093A patent/JOP20220093A1/ar unknown
- 2020-10-22 BR BR112022007207A patent/BR112022007207A2/pt not_active IP Right Cessation
- 2020-10-22 AU AU2020369912A patent/AU2020369912A1/en active Pending
- 2020-10-22 US US17/770,155 patent/US20220401441A1/en not_active Abandoned
-
2022
- 2022-05-20 EC ECSENADI202240921A patent/ECSP22040921A/es unknown
-
2025
- 2025-03-04 JP JP2025033867A patent/JP2025074286A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| EP4048235A1 (en) | 2022-08-31 |
| ECSP22040921A (es) | 2022-06-30 |
| BR112022007207A2 (pt) | 2022-07-26 |
| JP2022553313A (ja) | 2022-12-22 |
| WO2021078835A1 (en) | 2021-04-29 |
| MX2022004882A (es) | 2022-08-04 |
| CA3154802A1 (en) | 2021-04-29 |
| CN114555088A (zh) | 2022-05-27 |
| KR20220087443A (ko) | 2022-06-24 |
| PE20221455A1 (es) | 2022-09-21 |
| JP2025074286A (ja) | 2025-05-13 |
| JP7646646B2 (ja) | 2025-03-17 |
| JOP20220093A1 (ar) | 2023-01-30 |
| AU2020369912A1 (en) | 2022-04-14 |
| US20220401441A1 (en) | 2022-12-22 |
| IL292354A (en) | 2022-06-01 |
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