PE50296A1 - Eter substituido con tiazol y oxazol biciclico - Google Patents
Eter substituido con tiazol y oxazol biciclicoInfo
- Publication number
- PE50296A1 PE50296A1 PE1995278667A PE27866795A PE50296A1 PE 50296 A1 PE50296 A1 PE 50296A1 PE 1995278667 A PE1995278667 A PE 1995278667A PE 27866795 A PE27866795 A PE 27866795A PE 50296 A1 PE50296 A1 PE 50296A1
- Authority
- PE
- Peru
- Prior art keywords
- oxazole
- tiazole
- eter
- bicycle
- substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Diabetes (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
SE REFIERE AL COMPUESTO DE FORMULA I DONDE: X e Y SON INDEPENDIENTEMENTE OXIGENO O AZUFRE, DE PREFERENCIA OXIGENO; Z ES -CR1R2 o -CR1R2CH2-, DE PREFERENCIA EL PRIMERO; R1 Y R2 SON INDEPENDIENTEMENTE H o ALQUILO INFERIOR, DE PREFERENCIA H o METILO; R3 ES FENILO, OPCIONALMENTE MONOSUSTITUIDO O DISUSTITUIDO POR HALO, ALQUILO INFERIOR, ALCOXI INFERIOR O TRIFLUOROMETILO, DE PREFERENCIA ES FENILO MONOSUSTITUIDO O DISUSTITUIDO POR CLORO, ESPECIALMENTE 4-CLORO o 3,4 DICLORO; R4 Y R5 SON INDEPENDIENTEMENTE HIDROGENO, HALO, ALQUILO INFERIOR, -COOR6 ENTRE OTROS; TAMBIEN SE REFIERE AL PROCEDIMIENTO DE OBTENCION QUE COMPRENDE: a) LA PREPARACION DE UN COMPUESTO DE FORMULA I DONDE R6 ES DIFERENTE DE HIDROGENO, HACIENDO REACCIONAR UN COMPUESTO DE FORMULA II CON UN COMPUESTO DE FORMULA III, DONDE R7 ES H o UN GRUPO PROTECTOR DE AMINA; O b) LA PREPARACION DE UN COMPUESTO DE FORMULA I DONDE R6 ES H, HIDROLIZANDO UN COMPUESTO DE FORMULA I EN LA CUAL R6 ES ALQUILO INFERIOR o TRIALQUILSILIL(INFERIOR)ALQUILO(INFERIOR) Y LUEGO RECUPERAR EL COMPUESTO RESULTANTE DE FORMULA I
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US30524994A | 1994-09-13 | 1994-09-13 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE50296A1 true PE50296A1 (es) | 1996-12-05 |
Family
ID=23180015
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE1995278667A PE50296A1 (es) | 1994-09-13 | 1995-09-11 | Eter substituido con tiazol y oxazol biciclico |
Country Status (26)
| Country | Link |
|---|---|
| EP (1) | EP0702015B1 (es) |
| JP (1) | JPH08109183A (es) |
| KR (1) | KR960010649A (es) |
| CN (1) | CN1130186A (es) |
| AT (1) | ATE158585T1 (es) |
| AU (1) | AU3055295A (es) |
| BR (1) | BR9504004A (es) |
| CA (1) | CA2157950A1 (es) |
| CO (1) | CO4410332A1 (es) |
| CZ (1) | CZ229595A3 (es) |
| DE (1) | DE69500758T2 (es) |
| DK (1) | DK0702015T3 (es) |
| ES (1) | ES2108550T3 (es) |
| FI (1) | FI954257A (es) |
| GR (1) | GR3025405T3 (es) |
| HU (1) | HUT73432A (es) |
| IL (1) | IL115235A0 (es) |
| MY (1) | MY132008A (es) |
| NO (1) | NO953569L (es) |
| NZ (1) | NZ272976A (es) |
| PE (1) | PE50296A1 (es) |
| PL (1) | PL310372A1 (es) |
| SI (1) | SI0702015T1 (es) |
| SK (1) | SK111195A3 (es) |
| TR (1) | TR199501115A2 (es) |
| ZA (1) | ZA957699B (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2002314744A1 (en) | 2001-04-17 | 2002-10-28 | Sepracor, Inc. | Thiazole and other heterocyclic ligands and use thereof |
| DE10333935A1 (de) * | 2003-07-25 | 2005-02-24 | Aventis Pharma Deutschland Gmbh | Neue bicyclische Cyanoheterocyclen, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| FR2858321B1 (fr) * | 2003-07-28 | 2006-01-20 | Servier Lab | Nouveaux derives d'oximes heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1249992A (en) * | 1983-11-10 | 1989-02-14 | Marcel Muller | Oxazolidines |
| EP0590793B1 (en) * | 1992-08-31 | 1999-10-13 | Sankyo Company Limited | Oxazolidine derivatives having anti-diabetic and anti-obesity properties, their preparation and their therapeutic uses |
| US5321036A (en) * | 1993-02-10 | 1994-06-14 | Bristol-Myers Squibb Company | Thiazole and oxazole-based β3 adrenergic receptor agonists |
| KR0173145B1 (ko) * | 1993-04-07 | 1999-02-01 | 고바야시 유키오 | 티아졸리딘 유도체 및 이를 함유하는 약학적 조성물 |
-
1995
- 1995-09-06 SK SK1111-95A patent/SK111195A3/sk unknown
- 1995-09-07 CZ CZ952295A patent/CZ229595A3/cs unknown
- 1995-09-11 CA CA002157950A patent/CA2157950A1/en not_active Abandoned
- 1995-09-11 KR KR1019950029478A patent/KR960010649A/ko not_active Application Discontinuation
- 1995-09-11 JP JP7257240A patent/JPH08109183A/ja active Pending
- 1995-09-11 PE PE1995278667A patent/PE50296A1/es not_active Application Discontinuation
- 1995-09-11 AT AT95810561T patent/ATE158585T1/de not_active IP Right Cessation
- 1995-09-11 IL IL11523595A patent/IL115235A0/xx unknown
- 1995-09-11 AU AU30552/95A patent/AU3055295A/en not_active Abandoned
- 1995-09-11 DK DK95810561.1T patent/DK0702015T3/da active
- 1995-09-11 DE DE69500758T patent/DE69500758T2/de not_active Expired - Fee Related
- 1995-09-11 MY MYPI95002690A patent/MY132008A/en unknown
- 1995-09-11 ES ES95810561T patent/ES2108550T3/es not_active Expired - Lifetime
- 1995-09-11 FI FI954257A patent/FI954257A/fi not_active Application Discontinuation
- 1995-09-11 EP EP95810561A patent/EP0702015B1/en not_active Expired - Lifetime
- 1995-09-11 SI SI9530038T patent/SI0702015T1/xx unknown
- 1995-09-11 NO NO953569A patent/NO953569L/no unknown
- 1995-09-11 PL PL95310372A patent/PL310372A1/xx unknown
- 1995-09-11 NZ NZ272976A patent/NZ272976A/en unknown
- 1995-09-12 CN CN95115726A patent/CN1130186A/zh active Pending
- 1995-09-12 BR BR9504004A patent/BR9504004A/pt not_active Application Discontinuation
- 1995-09-12 CO CO95041744A patent/CO4410332A1/es unknown
- 1995-09-12 HU HU9502663A patent/HUT73432A/hu unknown
- 1995-09-12 TR TR95/01115A patent/TR199501115A2/xx unknown
- 1995-09-13 ZA ZA957699A patent/ZA957699B/xx unknown
-
1997
- 1997-11-19 GR GR970403050T patent/GR3025405T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI954257A0 (fi) | 1995-09-11 |
| NZ272976A (en) | 1996-09-25 |
| CZ229595A3 (en) | 1996-04-17 |
| CA2157950A1 (en) | 1996-03-14 |
| DE69500758T2 (de) | 1998-02-26 |
| JPH08109183A (ja) | 1996-04-30 |
| AU3055295A (en) | 1996-03-28 |
| EP0702015A1 (en) | 1996-03-20 |
| KR960010649A (ko) | 1996-04-20 |
| MY132008A (en) | 2007-09-28 |
| HUT73432A (en) | 1996-07-29 |
| NO953569D0 (no) | 1995-09-11 |
| PL310372A1 (en) | 1996-03-18 |
| BR9504004A (pt) | 1996-09-24 |
| CO4410332A1 (es) | 1997-01-09 |
| DK0702015T3 (da) | 1998-01-12 |
| IL115235A0 (en) | 1995-12-31 |
| TR199501115A2 (tr) | 1996-06-21 |
| DE69500758D1 (de) | 1997-10-30 |
| EP0702015B1 (en) | 1997-09-24 |
| HU9502663D0 (en) | 1995-11-28 |
| ATE158585T1 (de) | 1997-10-15 |
| ZA957699B (en) | 1997-03-13 |
| SI0702015T1 (en) | 1998-02-28 |
| CN1130186A (zh) | 1996-09-04 |
| SK111195A3 (en) | 1997-06-04 |
| ES2108550T3 (es) | 1997-12-16 |
| GR3025405T3 (en) | 1998-02-27 |
| FI954257A (fi) | 1996-03-14 |
| NO953569L (no) | 1996-03-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD | Application declared void or lapsed |