PE20211752A1 - Formas y metodos de dosis para bupropion enantiomericamente enriquecido o puro - Google Patents

Formas y metodos de dosis para bupropion enantiomericamente enriquecido o puro

Info

Publication number
PE20211752A1
PE20211752A1 PE2020001272A PE2020001272A PE20211752A1 PE 20211752 A1 PE20211752 A1 PE 20211752A1 PE 2020001272 A PE2020001272 A PE 2020001272A PE 2020001272 A PE2020001272 A PE 2020001272A PE 20211752 A1 PE20211752 A1 PE 20211752A1
Authority
PE
Peru
Prior art keywords
bupropion
dosage forms
enantiomerically enriched
methods
enriched
Prior art date
Application number
PE2020001272A
Other languages
English (en)
Spanish (es)
Inventor
Herriot Tabuteau
Original Assignee
Axsome Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Axsome Therapeutics Inc filed Critical Axsome Therapeutics Inc
Publication of PE20211752A1 publication Critical patent/PE20211752A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Addiction (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PE2020001272A 2018-02-23 2019-02-25 Formas y metodos de dosis para bupropion enantiomericamente enriquecido o puro PE20211752A1 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201862634718P 2018-02-23 2018-02-23
US201962794469P 2019-01-18 2019-01-18
US201962809480P 2019-02-22 2019-02-22
PCT/US2019/019445 WO2019165379A1 (en) 2018-02-23 2019-02-25 Dosage forms and methods for enantiomerically enriched or pure bupropion

Publications (1)

Publication Number Publication Date
PE20211752A1 true PE20211752A1 (es) 2021-09-06

Family

ID=67688503

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2020001272A PE20211752A1 (es) 2018-02-23 2019-02-25 Formas y metodos de dosis para bupropion enantiomericamente enriquecido o puro

Country Status (19)

Country Link
EP (1) EP3755312A4 (enExample)
JP (3) JP2021513998A (enExample)
KR (3) KR20230075531A (enExample)
CN (2) CN112087999A (enExample)
AU (3) AU2019223187B2 (enExample)
BR (1) BR112020017179A2 (enExample)
CA (1) CA3092076A1 (enExample)
CL (1) CL2020002166A1 (enExample)
CR (1) CR20200415A (enExample)
EC (1) ECSP20060179A (enExample)
IL (2) IL313368A (enExample)
MA (1) MA51914A (enExample)
MX (2) MX2020008704A (enExample)
MY (1) MY202993A (enExample)
NI (1) NI202000056A (enExample)
NZ (1) NZ767378A (enExample)
PE (1) PE20211752A1 (enExample)
SG (1) SG11202008056SA (enExample)
WO (1) WO2019165379A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20230075531A (ko) * 2018-02-23 2023-05-31 액섬 테라퓨틱스, 인크. 거울상이성질체적으로 농후한 또는 순수한 부프로피온을 위한 투여 형태 및 방법
US11291639B2 (en) 2018-09-20 2022-04-05 Axsome Therapeutics, Inc. Dosage forms and methods for enantiomerically enriched or pure bupropion
US11660273B2 (en) 2018-09-20 2023-05-30 Axsome Therapeutics, Inc. Dosage forms and methods for enantiomerically enriched or pure bupropion
US11660274B2 (en) 2018-09-20 2023-05-30 Axsome Therapeutics, Inc. Dosage forms and methods for enantiomerically enriched or pure bupropion
EP4031121A4 (en) * 2019-09-20 2022-11-30 Axsome Therapeutics, Inc. DOSAGE FORMS AND METHODS FOR FORMING ENANTIOMERICALLY ENRICHED OR PURE BUPROPION
US12156914B2 (en) * 2022-06-30 2024-12-03 Axsome Therapeutics, Inc. Pharmaceutical compositions comprising bupropion and cysteine
US11717518B1 (en) 2022-06-30 2023-08-08 Antecip Bioventures Ii Llc Bupropion dosage forms with reduced food and alcohol dosing effects

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2483499A (en) * 1998-01-29 1999-08-16 Sepracor, Inc. Pharmaceutical uses of optically pure (+)-bupropion
US6337328B1 (en) * 1999-03-01 2002-01-08 Sepracor, Inc. Bupropion metabolites and methods of use
DK1575565T3 (da) * 2003-08-08 2010-04-12 Biovail Lab Int Srl Tablet med modificeret frigivelse af bupropion-hydrochlorid
WO2012118562A1 (en) * 2011-03-02 2012-09-07 Rhine Pharmaceuticals, Llc Compositions and methods for treating depression, adhd and other central nervous system disorders employing novel bupropion compounds, and methods for production and use of novel bupropion compounds and formulations
US9198905B2 (en) * 2013-11-05 2015-12-01 Antecip Bioventures Ii Llc Compositions and methods for reducing dextrorphan plasma levels and related pharmacodynamic effects
US9474731B1 (en) * 2013-11-05 2016-10-25 Antecip Bioventures Ii Llc Compositions and methods for increasing the metabolic lifetime of dextromethorphan and related pharmacodynamic effects
US10080727B2 (en) * 2013-11-05 2018-09-25 Antecip Bioventures Ii Llc Compositions and methods for increasing the metabolic lifetime of dextromethorphan and related pharmacodynamic effects
WO2015095713A1 (en) * 2013-12-20 2015-06-25 Deuterx, Llc Methods of treating neurological and other disorders using enantiopure deuterium-enriched bupropion
KR20230075531A (ko) * 2018-02-23 2023-05-31 액섬 테라퓨틱스, 인크. 거울상이성질체적으로 농후한 또는 순수한 부프로피온을 위한 투여 형태 및 방법

Also Published As

Publication number Publication date
WO2019165379A1 (en) 2019-08-29
NZ767378A (en) 2024-03-22
IL276871B1 (en) 2024-07-01
CL2020002166A1 (es) 2020-10-23
AU2024205858A1 (en) 2024-09-05
NI202000056A (es) 2021-01-11
KR20210003091A (ko) 2021-01-11
IL276871B2 (en) 2024-11-01
AU2022204521B2 (en) 2024-09-05
CN112087999A (zh) 2020-12-15
ECSP20060179A (es) 2020-12-31
AU2019223187B2 (en) 2022-07-28
MA51914A (fr) 2020-12-30
JP2024075655A (ja) 2024-06-04
AU2019223187A1 (en) 2020-09-17
EP3755312A4 (en) 2022-03-16
KR20240091043A (ko) 2024-06-21
KR20230075531A (ko) 2023-05-31
CR20200415A (es) 2021-02-03
JP2022153638A (ja) 2022-10-12
CA3092076A1 (en) 2019-08-29
AU2022204521A1 (en) 2022-07-21
MX2023009281A (es) 2023-08-17
BR112020017179A2 (pt) 2020-12-22
EP3755312A1 (en) 2020-12-30
MX2020008704A (es) 2020-12-07
SG11202008056SA (en) 2020-09-29
MY202993A (en) 2024-05-31
IL313368A (en) 2024-08-01
JP2021513998A (ja) 2021-06-03
IL276871A (en) 2020-10-29
CN120827545A (zh) 2025-10-24

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