PE20081463A1 - Formas salinas de compuestos de benzotienilo sustituido - Google Patents
Formas salinas de compuestos de benzotienilo sustituidoInfo
- Publication number
- PE20081463A1 PE20081463A1 PE2007001405A PE2007001405A PE20081463A1 PE 20081463 A1 PE20081463 A1 PE 20081463A1 PE 2007001405 A PE2007001405 A PE 2007001405A PE 2007001405 A PE2007001405 A PE 2007001405A PE 20081463 A1 PE20081463 A1 PE 20081463A1
- Authority
- PE
- Peru
- Prior art keywords
- methyl
- salt
- benzothynyl
- compounds
- alcoxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/60—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
SE REFIERE A FORMAS SALINAS DE UN COMPUESTO DE BENZOTIENILO SUSTITUIDO DE FORMUAL (I), EN DONDE R1 ES UNO O DOS HALOGENOS; R2 ES ALQUILO(C1-C4), ALCOXI (C1-C4), ALCOXI(C1-C4)CARBONILOXI-ALCOXI(C1-C4), ENTRE OTROS; DONDE LA FORMA SALINA ESTA SELECCIONADA DEL GRUPO QUE CONSISTE EN UNA FORMA MONO-SAL O DI-SAL, SELECCIONADA DE BENZATINA, t-BUTILAMINA, MAGNESIO, CALCIO, COLINA, CICLOHEXILAMINA, DIETANOLAMINA, ETILENDIAMINA, L-LISINA, NH3, HN4OH, N-METIL-D-GLUCAMINA, TRIS(HIDROXIMETIL)METILAMINA, ENTRE OTROS. SON SELECCIONADOS: SAL MONOCOLINA DE (E)-{(5-CLORO-BENZO[b]TIOFEN-3-IL)-[2-(3,4-DIFLUOR-FENIL)-VINILCARBAMOIL]-METIL}-METIL-FOSFINICO, SAL MONO COLINA DE ACIDO (E)-{(5-CLORO-BENZO[b]TIOFEN-3-IL)-[2-(3,5-DICLORO-FENIL)-VINILCARBAMOIL]-METIL}-FOSFONICO, ENTRE OTROS. TAMBIEN SE REFIERE A UN PROCEDIMIENTO DE PREPARACION, ESTOS COMPUESTOS SON INHIBIDORES DEL RECEPTOR DE QUINASA
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US85340706P | 2006-10-20 | 2006-10-20 |
Publications (1)
Publication Number | Publication Date |
---|---|
PE20081463A1 true PE20081463A1 (es) | 2008-10-18 |
Family
ID=39325140
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PE2007001405A PE20081463A1 (es) | 2006-10-20 | 2007-10-17 | Formas salinas de compuestos de benzotienilo sustituido |
Country Status (20)
Country | Link |
---|---|
US (1) | US20080097110A1 (es) |
EP (1) | EP2081430A4 (es) |
JP (1) | JP2010506933A (es) |
KR (1) | KR20090069331A (es) |
CN (1) | CN101583272A (es) |
AR (1) | AR063342A1 (es) |
AU (1) | AU2007309463A1 (es) |
BR (1) | BRPI0718168A2 (es) |
CA (1) | CA2667197A1 (es) |
CL (1) | CL2007003011A1 (es) |
EA (1) | EA200900574A1 (es) |
EC (1) | ECSP099267A (es) |
IL (1) | IL198224A0 (es) |
MX (1) | MX2009004206A (es) |
NI (1) | NI200900060A (es) |
NO (1) | NO20091971L (es) |
PE (1) | PE20081463A1 (es) |
TW (1) | TW200821291A (es) |
UY (1) | UY30648A1 (es) |
WO (1) | WO2008051489A2 (es) |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20020082421A1 (en) * | 2000-09-14 | 2002-06-27 | Abdel-Magid Ahmed F. | Novel solid salt forms of N-[2-[4-[2-(1- methylethoxy)phenyl]-1-piperazinyl]-2-oxo-1piperidineacetamide |
GB0314136D0 (en) * | 2003-06-18 | 2003-07-23 | Astrazeneca Ab | Therapeutic agents |
EA011745B1 (ru) * | 2004-01-23 | 2009-06-30 | Янссен Фармацевтика Н.В. | Новые ингибиторы химазы |
-
2007
- 2007-10-17 PE PE2007001405A patent/PE20081463A1/es not_active Application Discontinuation
- 2007-10-17 UY UY30648A patent/UY30648A1/es unknown
- 2007-10-19 TW TW096139087A patent/TW200821291A/zh unknown
- 2007-10-19 AR ARP070104638A patent/AR063342A1/es unknown
- 2007-10-19 BR BRPI0718168-0A patent/BRPI0718168A2/pt not_active IP Right Cessation
- 2007-10-19 AU AU2007309463A patent/AU2007309463A1/en not_active Abandoned
- 2007-10-19 CN CNA2007800476139A patent/CN101583272A/zh active Pending
- 2007-10-19 US US11/975,571 patent/US20080097110A1/en not_active Abandoned
- 2007-10-19 MX MX2009004206A patent/MX2009004206A/es not_active Application Discontinuation
- 2007-10-19 WO PCT/US2007/022370 patent/WO2008051489A2/en active Application Filing
- 2007-10-19 EP EP07861463A patent/EP2081430A4/en not_active Withdrawn
- 2007-10-19 CL CL200703011A patent/CL2007003011A1/es unknown
- 2007-10-19 JP JP2009533394A patent/JP2010506933A/ja not_active Withdrawn
- 2007-10-19 EA EA200900574A patent/EA200900574A1/ru unknown
- 2007-10-19 CA CA002667197A patent/CA2667197A1/en not_active Abandoned
- 2007-10-19 KR KR1020097009863A patent/KR20090069331A/ko not_active Application Discontinuation
-
2009
- 2009-04-19 IL IL198224A patent/IL198224A0/en unknown
- 2009-04-20 NI NI200900060A patent/NI200900060A/es unknown
- 2009-04-20 EC EC2009009267A patent/ECSP099267A/es unknown
- 2009-05-20 NO NO20091971A patent/NO20091971L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
NO20091971L (no) | 2009-05-20 |
KR20090069331A (ko) | 2009-06-30 |
EP2081430A4 (en) | 2010-11-10 |
EP2081430A2 (en) | 2009-07-29 |
CL2007003011A1 (es) | 2008-04-18 |
AR063342A1 (es) | 2009-01-21 |
BRPI0718168A2 (pt) | 2013-11-26 |
CN101583272A (zh) | 2009-11-18 |
WO2008051489A2 (en) | 2008-05-02 |
NI200900060A (es) | 2010-02-01 |
IL198224A0 (en) | 2009-12-24 |
MX2009004206A (es) | 2009-04-30 |
AU2007309463A1 (en) | 2008-05-02 |
JP2010506933A (ja) | 2010-03-04 |
ECSP099267A (es) | 2009-11-30 |
TW200821291A (en) | 2008-05-16 |
UY30648A1 (es) | 2008-05-02 |
CA2667197A1 (en) | 2008-05-02 |
WO2008051489A3 (en) | 2008-07-10 |
EA200900574A1 (ru) | 2009-10-30 |
US20080097110A1 (en) | 2008-04-24 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AR121612A2 (es) | Inhibidores de glucosilceramida sintasa | |
PE20142403A1 (es) | Compuestos inhibidores de beta-lactamasas | |
CO6400228A2 (es) | Sintesis de nucleosidos de purina | |
UY30084A1 (es) | Compuestos de piperazina con accion herbicida | |
GB201018916D0 (en) | Corrosion inhibition | |
UY38057A (es) | Inhibidores de sarcómero cardíaco | |
CY1121703T1 (el) | Ιατρικη χρηση του πολυμορφου a toy ibanδρονικου | |
EA201400138A1 (ru) | Пестицидные способы применения замещенных 3-пиридилтиазольных соединений и производных для борьбы с животными-вредителями ii | |
CO6761321A2 (es) | Pesticidas mesoionicos de pirido [1,2-a] pirimidina | |
PE20131047A1 (es) | Compuestos heterociclicos moduladores del acido urico | |
TW200640940A (en) | Ibandronate polymorph B | |
AR080827A1 (es) | Utilizacion del acido 4- fenil- butirico y/o de sus sales para el aumento de la tolerancia al estres en plantas | |
EA200900918A1 (ru) | Гетероароилзамещенные серинамиды | |
EA200700557A1 (ru) | Замещенные гетероароилом серин-амиды | |
MA41607A (fr) | Sels d'un inhibiteur de pi3k et procédés de préparation de ces sels | |
CL2008002922A1 (es) | Metodo para inhibir formacion y deposicion de incrustaciones en un proceso de desalinizacion que comprende agregar a una fuente acuosa salina, cantidad efectiva de una composicion de inhibidor de incrustaciones que incluye un copolimero de acido acrilico y acido 2-acrilamido-2-metilpropil sulfonico y acido fosfosuccinico oligomerico. | |
CO6351685A2 (es) | Metodo para controlar vegetacion mimosoideae no deseada | |
BR112014002612A2 (pt) | composições compreendendo monoésteres de isossorbida e hidroxipiridonas | |
ES2189464T3 (es) | Sales de nitrato como compuestos medicos. | |
BR112014002600A2 (pt) | composições compreendendo monoésteres e álcoois de isosorbida compreendendo pelo menos um grupo aromático | |
AR057909A1 (es) | Proceso para preparar montelukast y compuestos relacionados, que utiliza un compuesto intermediario derivado de un ester sulfonico. | |
AR061901A1 (es) | Proceso para la produccion de fosfatos metalicos nanofinos, fosfato nanofino producido mediante dicho proceso y su uso | |
AR069437A1 (es) | Bisfosfonatos de alquilo de 2 a 5 atomos de carbono - imidazol | |
UA109282C2 (xx) | Пестицидна суспензія на водній основі | |
AR075097A1 (es) | Sales y formas polimorficas cristalinas de [4-(6-fluoro-7-metilamino-2,4-dioxo-1,4-dihidro-2h-quinazolin-3-il)-fenil]-5-cloro-tiofen-2-il-sulfonil urea, composiciones farmaceuticas que las contiene, metodo para prepararlas y uso de las mismas en el tratamiento de enfermedades cardiovasculares asocia |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD | Application declared void or lapsed |