CL2007003011A1 - Forma salina de compuestos de benzotienilo sustituidos; procedimiento de preparacion; sal mono-colina de acido (e)-{(5-cloro-benzo[b]tiofen-3-il)-[2-(3,4-difluorfenil)-vinilcarbamoil]-metil}-metil-fosfinico. - Google Patents

Forma salina de compuestos de benzotienilo sustituidos; procedimiento de preparacion; sal mono-colina de acido (e)-{(5-cloro-benzo[b]tiofen-3-il)-[2-(3,4-difluorfenil)-vinilcarbamoil]-metil}-metil-fosfinico.

Info

Publication number
CL2007003011A1
CL2007003011A1 CL200703011A CL2007003011A CL2007003011A1 CL 2007003011 A1 CL2007003011 A1 CL 2007003011A1 CL 200703011 A CL200703011 A CL 200703011A CL 2007003011 A CL2007003011 A CL 2007003011A CL 2007003011 A1 CL2007003011 A1 CL 2007003011A1
Authority
CL
Chile
Prior art keywords
metil
benzotienyl
tiofen
carbamoil
difluorphenyl
Prior art date
Application number
CL200703011A
Other languages
English (en)
Inventor
Liugi Villani Frank J Anzalone
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of CL2007003011A1 publication Critical patent/CL2007003011A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/60Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CL200703011A 2006-10-20 2007-10-19 Forma salina de compuestos de benzotienilo sustituidos; procedimiento de preparacion; sal mono-colina de acido (e)-{(5-cloro-benzo[b]tiofen-3-il)-[2-(3,4-difluorfenil)-vinilcarbamoil]-metil}-metil-fosfinico. CL2007003011A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US85340706P 2006-10-20 2006-10-20

Publications (1)

Publication Number Publication Date
CL2007003011A1 true CL2007003011A1 (es) 2008-04-18

Family

ID=39325140

Family Applications (1)

Application Number Title Priority Date Filing Date
CL200703011A CL2007003011A1 (es) 2006-10-20 2007-10-19 Forma salina de compuestos de benzotienilo sustituidos; procedimiento de preparacion; sal mono-colina de acido (e)-{(5-cloro-benzo[b]tiofen-3-il)-[2-(3,4-difluorfenil)-vinilcarbamoil]-metil}-metil-fosfinico.

Country Status (20)

Country Link
US (1) US20080097110A1 (es)
EP (1) EP2081430A4 (es)
JP (1) JP2010506933A (es)
KR (1) KR20090069331A (es)
CN (1) CN101583272A (es)
AR (1) AR063342A1 (es)
AU (1) AU2007309463A1 (es)
BR (1) BRPI0718168A2 (es)
CA (1) CA2667197A1 (es)
CL (1) CL2007003011A1 (es)
EA (1) EA200900574A1 (es)
EC (1) ECSP099267A (es)
IL (1) IL198224A0 (es)
MX (1) MX2009004206A (es)
NI (1) NI200900060A (es)
NO (1) NO20091971L (es)
PE (1) PE20081463A1 (es)
TW (1) TW200821291A (es)
UY (1) UY30648A1 (es)
WO (1) WO2008051489A2 (es)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2001290743A1 (en) * 2000-09-14 2002-03-26 Ortho-Mcneil Pharmaceutical, Inc. Solid salt forms of n-(2-(4-(2-(1-methylethoxy)phenyl)-1-piperazinyl)ethyl)-2-oxo-1-piperidineacetamide
GB0314136D0 (en) * 2003-06-18 2003-07-23 Astrazeneca Ab Therapeutic agents
EP1716160B1 (en) * 2004-01-23 2010-12-29 Janssen Pharmaceutica NV Novel inhibitors of chymase

Also Published As

Publication number Publication date
IL198224A0 (en) 2009-12-24
PE20081463A1 (es) 2008-10-18
WO2008051489A2 (en) 2008-05-02
EA200900574A1 (ru) 2009-10-30
EP2081430A4 (en) 2010-11-10
NO20091971L (no) 2009-05-20
AU2007309463A1 (en) 2008-05-02
TW200821291A (en) 2008-05-16
CN101583272A (zh) 2009-11-18
JP2010506933A (ja) 2010-03-04
NI200900060A (es) 2010-02-01
MX2009004206A (es) 2009-04-30
EP2081430A2 (en) 2009-07-29
CA2667197A1 (en) 2008-05-02
WO2008051489A3 (en) 2008-07-10
AR063342A1 (es) 2009-01-21
UY30648A1 (es) 2008-05-02
BRPI0718168A2 (pt) 2013-11-26
KR20090069331A (ko) 2009-06-30
US20080097110A1 (en) 2008-04-24
ECSP099267A (es) 2009-11-30

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