PE20070229A1 - 7-AMINO-6-HETEROARYL-1,2,4-TRIAZOLO [1,5-a] PYRIMIDINE COMPOUNDS AND THEIR USE TO COMBAT DANGEROUS FUNGI - Google Patents

7-AMINO-6-HETEROARYL-1,2,4-TRIAZOLO [1,5-a] PYRIMIDINE COMPOUNDS AND THEIR USE TO COMBAT DANGEROUS FUNGI

Info

Publication number
PE20070229A1
PE20070229A1 PE2006000927A PE2006000927A PE20070229A1 PE 20070229 A1 PE20070229 A1 PE 20070229A1 PE 2006000927 A PE2006000927 A PE 2006000927A PE 2006000927 A PE2006000927 A PE 2006000927A PE 20070229 A1 PE20070229 A1 PE 20070229A1
Authority
PE
Peru
Prior art keywords
triazolo
heteroaryl
amino
pyrimidine
halogen
Prior art date
Application number
PE2006000927A
Other languages
Spanish (es)
Inventor
Oliver Wagner
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of PE20070229A1 publication Critical patent/PE20070229A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Abstract

SE REFIERE A COMPUESTOS DE 7-AMINO-6-HETEROARIL-1,2,4-TRIAZOLO[1,5-a] PIRIMIDINA DE FORMULA (I), EN DONDE HET ES HETEROARILO DE 5 MIEMBROS CON 2 ATOMOS DE N, SELECCIONADOS DE (1,2,3-), (1,2,4-), (1,3,4-), (1,2,5-) -TIADIAZOLILO, (1,2,4-), (1,3,4-), (1,2,5-) -OXADIAZOLILO, OPCIONALMENTE SUSTITUIDO POR L, DONDE L ES HALOGENO, CIANO, NITRO, ENTRE OTROS; R1 Y R2 SON INDEPENDIENTEMENTE H, ALQUILO(C1-C8), HALOALQUILO(C1-C8), ENTRE OTROS; O JUNTOS CON EL N, FORMAN UN HETEROCICLO DE 5 O 6 MIEMBROS OPCIONALMENTE SATURADO O AROMATICO CON HETEROATOMOS DE O, N O S, OPCIONALMENTE SUSTITUIDOS CON Ra; X ES H, HALOGENO, CIANO,ALCOXI(C1-C8), HALOGENO ALCOXI(C1-C8), ENTRE OTROS; Y ES H, HALOGENO, ALQUILO, ENTRE OTROS. SIENDO SELECCIONADO R-(5-CLORO-6-(5-METIL-[1,3,4]-TIADIAZOL-2-IL)-7-(1,2-DIMETILPROPILAMINO))-[1,2,4]-TRIAZOLO[1,5-a]PIRIMIDINA, 5-CLORO-6-(5-METIL-[1,3,4]-TIADIAZOL-2-IL)-7-(4-METILPIPERIDIN-1-IL)-[1,2,4]-TRIAZOLO[1,5-a]PIRIMIDINA. TAMBIEN SE REFIERE A UN PROCEDIMIENTO DE PREPARACION. ESTOS COMPUESTOS SON UTILES EN AGRICULTURA POR PRESETAR ACTIVIDAD FUNGICIDA CONTRA UN AMPLIO ESPECTRO DE HONGOS FITOPATOGENOSREFERS TO COMPOUNDS OF 7-AMINO-6-HETEROARYL-1,2,4-TRIAZOLO [1,5-a] PYRIMIDINE OF FORMULA (I), WHERE HET IS 5-MEMBER HETEROARILO WITH 2 N ATOMS, SELECTED FROM (1,2,3-), (1,2,4-), (1,3,4-), (1,2,5-) -TIADIAZOLYL, (1,2,4-), (1, 3,4-), (1,2,5-) -OXADIAZOLYL, OPTIONALLY SUBSTITUTED BY L, WHERE L IS HALOGEN, CYANE, NITRO, AMONG OTHERS; R1 AND R2 ARE INDEPENDENTLY H, ALKYL (C1-C8), HALOALKYL (C1-C8), AMONG OTHERS; OR TOGETHER WITH N, THEY FORM A 5 OR 6-MEMBER HETEROCICLE OPTIONALLY SATURATED OR AROMATIC WITH O, N OR S HETEROATOMS, OPTIONALLY SUBSTITUTED WITH Ra; X IS H, HALOGEN, CYANE, ALCOXY (C1-C8), HALOGEN ALCOXY (C1-C8), AMONG OTHERS; AND IT IS H, HALOGENO, RENT, AMONG OTHERS. BEING SELECTED R- (5-CHLORO-6- (5-METHYL- [1,3,4] -TIADIAZOL-2-IL) -7- (1,2-DIMETHYLPROPYLAMINE)) - [1,2,4] - TRIAZOLO [1,5-a] PYRIMIDINE, 5-CHLORO-6- (5-METHYL- [1,3,4] -TIADIAZOL-2-IL) -7- (4-METHYLPIPERIDIN-1-IL) - [1 , 2,4] -TRIAZOLO [1,5-a] PYRIMIDINE. IT ALSO REFERS TO A PREPARATION PROCEDURE. THESE COMPOUNDS ARE USEFUL IN AGRICULTURE BECAUSE THEY PRESET FUNGICIDAL ACTIVITY AGAINST A WIDE SPECTRUM OF PHYTOPATOGENIC FUNGI

PE2006000927A 2005-07-29 2006-07-31 7-AMINO-6-HETEROARYL-1,2,4-TRIAZOLO [1,5-a] PYRIMIDINE COMPOUNDS AND THEIR USE TO COMBAT DANGEROUS FUNGI PE20070229A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102005036319 2005-07-29

Publications (1)

Publication Number Publication Date
PE20070229A1 true PE20070229A1 (en) 2007-03-29

Family

ID=37402685

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2006000927A PE20070229A1 (en) 2005-07-29 2006-07-31 7-AMINO-6-HETEROARYL-1,2,4-TRIAZOLO [1,5-a] PYRIMIDINE COMPOUNDS AND THEIR USE TO COMBAT DANGEROUS FUNGI

Country Status (6)

Country Link
AR (1) AR055103A1 (en)
GT (1) GT200600344A (en)
PE (1) PE20070229A1 (en)
TW (1) TW200738721A (en)
UY (1) UY29707A1 (en)
WO (1) WO2007012642A1 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007101870A1 (en) * 2006-03-08 2007-09-13 Basf Se Substituted triazolopyrimidines, methods for the production thereof and use thereof for controlling parasitic fungi and agents containing the latter
AR081626A1 (en) 2010-04-23 2012-10-10 Cytokinetics Inc AMINO-PYRIDAZINIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM AND USE OF THE SAME TO TREAT CARDIAC AND SKELETIC MUSCULAR DISORDERS
AR081331A1 (en) 2010-04-23 2012-08-08 Cytokinetics Inc AMINO- PYRIMIDINES COMPOSITIONS OF THE SAME AND METHODS FOR THE USE OF THE SAME
US9133123B2 (en) 2010-04-23 2015-09-15 Cytokinetics, Inc. Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use
US8759380B2 (en) 2011-04-22 2014-06-24 Cytokinetics, Inc. Certain heterocycles, compositions thereof, and methods for their use

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL108731A (en) * 1993-03-04 1997-03-18 Shell Int Research 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
DE10063115A1 (en) * 2000-12-18 2002-06-27 Bayer Ag triazolopyrimidines
DE10328481A1 (en) * 2003-06-25 2005-01-13 Bayer Ag triazolopyrimidines

Also Published As

Publication number Publication date
AR055103A1 (en) 2007-08-08
WO2007012642A1 (en) 2007-02-01
GT200600344A (en) 2006-12-13
UY29707A1 (en) 2007-02-28
TW200738721A (en) 2007-10-16

Similar Documents

Publication Publication Date Title
PE20100741A1 (en) COMPOUNDS DERIVED FROM 3,4-DIHYDROPYRIMIDE [4,5-d] PYRIMIDIN-2 (1H) -ONE AS KINASE INHIBITORS p38
PE20091833A1 (en) BRIDGED, BRIDGED BICYCLE SPIRO HETEROCYCLIC OR BICYCLE HETERO CYCLIC DERIVATIVES OF PIRAZOLO [1,5-A] PYRIMIDINES AS RAF KINASES INHIBITORS AND METHODS FOR THEIR PREPARATION
GEP20146030B (en) Organic compounds
PE20070229A1 (en) 7-AMINO-6-HETEROARYL-1,2,4-TRIAZOLO [1,5-a] PYRIMIDINE COMPOUNDS AND THEIR USE TO COMBAT DANGEROUS FUNGI
PE20091211A1 (en) PYRAZOLOPYRIMIDINE DERIVATIVES AS PDE9A MODULATORS
BRPI0611095B8 (en) pde1 inhibitor compounds, pharmaceutical composition comprising them, uses thereof as pde1 inhibitors for the treatment of related diseases such as parkinson's disease and cognitive impairment, and methods for producing said compounds
PE20100737A1 (en) NEW COMPOUNDS
Kashyap et al. Review on synthesis and various biological potential of thiazolopyrimidine derivatives
EA200600677A1 (en) 5,7-DIAMINOPIRAZOLO [4,3-D] Pyrimidines with PDE-5 inhibitory activity
PE20061354A1 (en) 2-AMINO-4-OXOBUTIL COMPOUNDS AS INHIBITORS OF DIPEPTIDYL PEPTIDES-IV
PE20091493A1 (en) PYRROLOPYRAZINE KINASE INHIBITORS
PE20081377A1 (en) THIAZOL COMPOUNDS PYRAZOLOPYRIMIDINE
PE20030155A1 (en) AZAINDOLS AS KINASE INHIBITORS
PE20081806A1 (en) IMIDAZO- AND SUBSTITUTE TRIAZOLOPYRIMIDINES
PE20091485A1 (en) PYROLO- [2,3-d] -PYRIMIDINE DERIVATIVES AS KINE INHIBITORS
PE20071104A1 (en) AMINOTETRAHYDROPYRANS AS INHIBITORS OF DIPEPTIDYL PEPTIDASE-IV (DPP-4)
PE20080315A1 (en) DERIVATIVES OF PIRAZOLO- [3,4-d] -PYRIMIDINES AS INHIBITORS OF KINASE PI-3
PE20090944A1 (en) BICYCLE PYRIMIDINES FUSED AS INHIBITORS OF THE PI3K / AKT VIA
PE20141023A1 (en) DERIVATIVES OF (1,2,4) TRIAZOLO [4,3-A] QUINOXALINE AS INHIBITORS OF PHOSPHODIESTERASES
PE20110582A1 (en) ARILCICLOHEXILETERES DE DIHIDRO-TETRAAZABENZOAZULENO
PE20081159A1 (en) INHIBITORS OF KINASES AND METHODS FOR THEIR USE
EA201070817A1 (en) IMIDAZO [1,2-α] PYRIDIN-2-CARBOXAMID DERIVATIVES, THEIR RECEIVING AND THEIR USE IN THERAPY
PE20071168A1 (en) COMPOUNDS DERIVED FROM 5,6-DIPHENYLFIDE [2,3-D] PYRIMIDINE AS NON-PROSTANOID ACTIVATORS OF THE IP RECEPTOR
PE20051165A1 (en) 5, 6-DIALKYL-7-AMINO-TRIAZOLOPYRIMIDINES COMPOUNDS
PE20060772A1 (en) 7-AMINO-6-HETARYL-1,2,4-TRIAZOLO [1,5-A] PYRIMIDINE COMPOUNDS TO COMBAT PHYTOPATOGENIC FUNGI

Legal Events

Date Code Title Description
FA Abandonment or withdrawal