PE20001598A1 - Derivados de n-[2-(4-aminofenil)etil]-2,3-dihidro-1,4-benzodioxin-2-metanamina - Google Patents
Derivados de n-[2-(4-aminofenil)etil]-2,3-dihidro-1,4-benzodioxin-2-metanaminaInfo
- Publication number
- PE20001598A1 PE20001598A1 PE2000000275A PE0002752000A PE20001598A1 PE 20001598 A1 PE20001598 A1 PE 20001598A1 PE 2000000275 A PE2000000275 A PE 2000000275A PE 0002752000 A PE0002752000 A PE 0002752000A PE 20001598 A1 PE20001598 A1 PE 20001598A1
- Authority
- PE
- Peru
- Prior art keywords
- benzodioxin
- dihydro
- derivatives
- ethyl
- alcoxycarbonylmethyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
- C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
- C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D319/20—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
SE REFIERE A DERIVADOS DE N-[2-(4-AMINOFENIL)ETIL]-2,3-DIHIDRO-1,4-BENZODIOXIN-2-METANAMINA DE FORMULA I, DONDE: X ES H, HALOGENO, CIANO, NITRO, OH, ALQUILO C1-C4, FENILO, TIENILO, TIENILMETOXI, ALCOXI C1-C4, CICLOALQUILMETOXI C3-C6, FENILMETOXI, ALCOXICARBONILO C1-C4, ALCOXICARBONILMETILO C1-C4, PIRROLIDIN-1-ILCARBONILO, CARBAMOILO, ENTRE OTROS; R1 ES H, METILO; R2 ES ALCANOILO C1-C4, FENILALCANOILO C1-C4, METOXIACETILO, CICLOALQUILCARBONILO C3-C6, BENZOILO OPCIONALMENTE SUSTITUIDO CON HALOGENO, ALQUILO C1-C4, ALCOXI C1-C4, ENTRE OTROS; NR1R2 ES 2-OXO-4,5-DIHIDROOXAZOLIDIN-3-ILO. LOS COMPUESTOS DE FORMULA I TIENEN AFINIDAD POR LOS RECEPTORES DOPAMINERGICOS DE TIPO D3, AFINIDAD MODERADA DE TIPO D2 Y 5-HT1A Y PUEDEN SER UTILES PARA EL TRATAMIENTO DE PSICOSIS, ESQUIZOFRENIA, ANSIEDAD, PANICO, FOBIAS, TRASTORNOS OBSESIVO COMPULSIVOS
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9903936A FR2791675B1 (fr) | 1999-03-30 | 1999-03-30 | Derives de n-[2-(4-aminophenyl) ethyl] -2,3-dihydro-1,4- benzodioxinne-2-methanamine, leur preparation et leur application en therapeutique |
Publications (1)
Publication Number | Publication Date |
---|---|
PE20001598A1 true PE20001598A1 (es) | 2001-04-01 |
Family
ID=9543788
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PE2000000275A PE20001598A1 (es) | 1999-03-30 | 2000-03-30 | Derivados de n-[2-(4-aminofenil)etil]-2,3-dihidro-1,4-benzodioxin-2-metanamina |
Country Status (6)
Country | Link |
---|---|
AU (1) | AU3660700A (es) |
CO (1) | CO5170535A1 (es) |
FR (1) | FR2791675B1 (es) |
PE (1) | PE20001598A1 (es) |
UY (1) | UY26085A1 (es) |
WO (1) | WO2000058301A1 (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0117396D0 (en) | 2001-07-17 | 2001-09-05 | Glaxo Group Ltd | Chemical compounds |
GB0308208D0 (en) | 2003-04-09 | 2003-05-14 | Glaxo Group Ltd | Chemical compounds |
PA8663501A1 (es) | 2005-02-17 | 2006-11-09 | Wyeth Wyeth | Derivados de indol, benzotiofeno, benzofurano e indeno cicloalquilcondensados |
TW200716595A (en) | 2005-04-22 | 2007-05-01 | Wyeth Corp | Chromane and chromene derivatives and uses thereof |
JP2008538575A (ja) * | 2005-04-22 | 2008-10-30 | ワイス | ベンゾジオキサンおよびベンゾジオキソラン誘導体ならびにそれらの使用 |
AR060493A1 (es) * | 2006-04-18 | 2008-06-18 | Wyeth Corp | Derivados de benzodioxano y benzodioxolano. procesos de obtencion. |
TW200823187A (en) * | 2006-10-24 | 2008-06-01 | Wyeth Corp | Benzodioxane derivatives and uses thereof |
CA2722986A1 (en) | 2008-04-29 | 2009-11-05 | Nsab, Filial Af Neurosearch Sweden Ab, Sverige | Modulators of dopamine neurotransmission |
CA2722978A1 (en) | 2008-04-29 | 2009-11-05 | Nsab, Filial Af Neurosearch Sweden Ab, Sverige | Modulators of dopamine neurotransmission |
EP2271635A1 (en) * | 2008-04-29 | 2011-01-12 | NSAB, Filial af NeuroSearch Sweden AB, Sverige | Modulators of dopamine neurotransmission |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NL281245A (es) * | 1962-07-20 | |||
CA1147342A (en) * | 1977-10-12 | 1983-05-31 | Kazuo Imai | Process of producing novel phenylethanolamine derivatives |
-
1999
- 1999-03-30 FR FR9903936A patent/FR2791675B1/fr not_active Expired - Fee Related
-
2000
- 2000-03-27 WO PCT/FR2000/000762 patent/WO2000058301A1/fr active Application Filing
- 2000-03-27 AU AU36607/00A patent/AU3660700A/en not_active Abandoned
- 2000-03-29 CO CO00022433A patent/CO5170535A1/es not_active Application Discontinuation
- 2000-03-29 UY UY26085A patent/UY26085A1/es unknown
- 2000-03-30 PE PE2000000275A patent/PE20001598A1/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO2000058301A1 (fr) | 2000-10-05 |
UY26085A1 (es) | 2000-10-31 |
AU3660700A (en) | 2000-10-16 |
CO5170535A1 (es) | 2002-06-27 |
FR2791675A1 (fr) | 2000-10-06 |
FR2791675B1 (fr) | 2001-05-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Grant, registration | ||
FD | Application declared void or lapsed |