NZ561710A - Alpha aminoacid ester-drug conjugates hydrolysable by carboxylesterase - Google Patents

Alpha aminoacid ester-drug conjugates hydrolysable by carboxylesterase

Info

Publication number
NZ561710A
NZ561710A NZ561710A NZ56171006A NZ561710A NZ 561710 A NZ561710 A NZ 561710A NZ 561710 A NZ561710 A NZ 561710A NZ 56171006 A NZ56171006 A NZ 56171006A NZ 561710 A NZ561710 A NZ 561710A
Authority
NZ
New Zealand
Prior art keywords
inhibitor
amino acid
conjugate
ester
enzyme
Prior art date
Application number
NZ561710A
Other languages
English (en)
Inventor
Alan Hornsby Davidson
Alan Hastings Drummond
Lindsey Ann Needham
Original Assignee
Chroma Therapeutics Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chroma Therapeutics Ltd filed Critical Chroma Therapeutics Ltd
Priority claimed from PCT/GB2006/001635 external-priority patent/WO2006117567A2/en
Publication of NZ561710A publication Critical patent/NZ561710A/en

Links

Landscapes

  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicinal Preparation (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
NZ561710A 2005-05-05 2006-05-04 Alpha aminoacid ester-drug conjugates hydrolysable by carboxylesterase NZ561710A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0509226A GB0509226D0 (en) 2005-05-05 2005-05-05 Enzyme and receptor modulation
US68054205P 2005-05-13 2005-05-13
PCT/GB2006/001635 WO2006117567A2 (en) 2005-05-05 2006-05-04 Alpha aminoacid ester-drug conjugates hydrolysable by carboxylesterase

Publications (1)

Publication Number Publication Date
NZ561710A true NZ561710A (en) 2010-08-27

Family

ID=34685158

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ561710A NZ561710A (en) 2005-05-05 2006-05-04 Alpha aminoacid ester-drug conjugates hydrolysable by carboxylesterase

Country Status (10)

Country Link
CN (1) CN101171039B (zh)
CA (1) CA2836827C (zh)
DK (1) DK1877098T3 (zh)
ES (2) ES2415244T3 (zh)
GB (1) GB0509226D0 (zh)
NZ (1) NZ561710A (zh)
PT (1) PT1877098E (zh)
SG (1) SG2014007512A (zh)
SI (1) SI1877098T1 (zh)
ZA (1) ZA200708283B (zh)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1231919B1 (en) * 1999-09-08 2015-09-30 Sloan-Kettering Institute For Cancer Research Derivatives of 1-amino-1-(hetero)arylaminocarbonyl-6-hydroxyaminocarbonylhexane useful in the treatment of tumors
WO2005037272A1 (en) * 2003-10-22 2005-04-28 Arpida A/S Benzimidazole derivatives and use thereof as peptide deformylase inhibitors

Also Published As

Publication number Publication date
ZA200708283B (en) 2008-10-29
ES2577433T3 (es) 2016-07-14
PT1877098E (pt) 2013-07-31
CA2836827A1 (en) 2006-11-09
CN101171039B (zh) 2013-01-23
SI1877098T1 (sl) 2013-08-30
CN101171039A (zh) 2008-04-30
SG2014007512A (en) 2014-03-28
CA2836827C (en) 2016-05-03
GB0509226D0 (en) 2005-06-15
DK1877098T3 (da) 2013-07-08
ES2415244T3 (es) 2013-07-24

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