NZ530211A - D-threo methylphenidate substantially free of the L-threo form to treat fatigue, neurobehavioral slowing and other cogitative disorders exacerbated by treatments associated with cancer therapy - Google Patents
D-threo methylphenidate substantially free of the L-threo form to treat fatigue, neurobehavioral slowing and other cogitative disorders exacerbated by treatments associated with cancer therapyInfo
- Publication number
- NZ530211A NZ530211A NZ530211A NZ53021102A NZ530211A NZ 530211 A NZ530211 A NZ 530211A NZ 530211 A NZ530211 A NZ 530211A NZ 53021102 A NZ53021102 A NZ 53021102A NZ 530211 A NZ530211 A NZ 530211A
- Authority
- NZ
- New Zealand
- Prior art keywords
- threo
- methylphenidate
- treatment
- oncological condition
- substantially free
- Prior art date
Links
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Classifications
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- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/34—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
- C12P17/00—Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms
- C12P17/10—Nitrogen as only ring hetero atom
- C12P17/12—Nitrogen as only ring hetero atom containing a six-membered hetero ring
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- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
- C12P41/00—Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture
- C12P41/006—Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture by reactions involving C-N bonds, e.g. nitriles, amides, hydantoins, carbamates, lactames, transamination reactions, or keto group formation from racemic mixtures
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
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- Chemical Kinetics & Catalysis (AREA)
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- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Epidemiology (AREA)
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- Biochemistry (AREA)
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- Endocrinology (AREA)
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- Cardiology (AREA)
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- Hematology (AREA)
- Heart & Thoracic Surgery (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| NZ565754A NZ565754A (en) | 2001-07-12 | 2002-07-11 | Methods for treatment of cognitive and menopausal disorders with D-threo methylphenidate |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/903,803 US6486177B2 (en) | 1995-12-04 | 2001-07-12 | Methods for treatment of cognitive and menopausal disorders with D-threo methylphenidate |
| PCT/US2002/022039 WO2003005962A2 (en) | 2001-07-12 | 2002-07-11 | Methods for treatment of cognitive and menopausal disorders with d-threo methylphenidate |
Publications (1)
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| NZ530211A true NZ530211A (en) | 2008-04-30 |
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| NZ530211A NZ530211A (en) | 2001-07-12 | 2002-07-11 | D-threo methylphenidate substantially free of the L-threo form to treat fatigue, neurobehavioral slowing and other cogitative disorders exacerbated by treatments associated with cancer therapy |
| NZ565754A NZ565754A (en) | 2001-07-12 | 2002-07-11 | Methods for treatment of cognitive and menopausal disorders with D-threo methylphenidate |
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| NZ565754A NZ565754A (en) | 2001-07-12 | 2002-07-11 | Methods for treatment of cognitive and menopausal disorders with D-threo methylphenidate |
Country Status (10)
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| EP (1) | EP1411943A4 (https=) |
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| KR (1) | KR20040029360A (https=) |
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| CA (1) | CA2453510C (https=) |
| IL (1) | IL159313A0 (https=) |
| MX (1) | MXPA04000249A (https=) |
| NZ (2) | NZ530211A (https=) |
| WO (1) | WO2003005962A2 (https=) |
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| WO1997003671A1 (en) | 1995-07-14 | 1997-02-06 | Medeva Europe Limited | Composition comprising d-threo-methylphenidate and another drug |
| US5837284A (en) * | 1995-12-04 | 1998-11-17 | Mehta; Atul M. | Delivery of multiple doses of medications |
| US5922736A (en) * | 1995-12-04 | 1999-07-13 | Celegene Corporation | Chronic, bolus administration of D-threo methylphenidate |
| US6486177B2 (en) * | 1995-12-04 | 2002-11-26 | Celgene Corporation | Methods for treatment of cognitive and menopausal disorders with D-threo methylphenidate |
| US6962997B1 (en) * | 1997-05-22 | 2005-11-08 | Celgene Corporation | Process and intermediates for resolving piperidyl acetamide steroisomers |
| WO2001097806A1 (en) * | 2000-06-20 | 2001-12-27 | Herbst Arthur L | Cox-2 inhibitors and the prevention of the side effects of radiation therapy |
| FR2823975B1 (fr) * | 2001-04-27 | 2003-05-30 | Sanofi Synthelabo | Nouvelle utilisation de pyridoindolone |
| ATE526988T1 (de) * | 2003-10-08 | 2011-10-15 | Mallinckrodt Llc | Methylphenidat-lösung und relevante verabreichungs- und herstellungsverfahren |
| US20050239830A1 (en) * | 2004-04-26 | 2005-10-27 | Vikram Khetani | Methods of diminishing co-abuse potential |
| WO2006012476A2 (en) * | 2004-07-22 | 2006-02-02 | Wyeth | Method for treating nervous system disorders and conditions |
| MX2007000851A (es) * | 2004-07-22 | 2007-03-26 | Wyeth Corp | Procedimiento para el tratamiento de trastornos y dolencias del sistema nervioso. |
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| CN102488652B (zh) | 2006-03-16 | 2014-06-18 | 特瑞斯制药股份有限公司 | 含有药物-离子交换树脂复合物的经修饰释放的制剂 |
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| KR101312286B1 (ko) * | 2012-11-26 | 2013-09-27 | (주)비씨월드제약 | 즉시방출 및 조절방출 특성을 갖고 d-트레오-메틸페니데이트를 포함하는 약학 조성물 |
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2001
- 2001-07-12 US US09/903,803 patent/US6486177B2/en not_active Expired - Fee Related
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2002
- 2002-07-11 NZ NZ530211A patent/NZ530211A/en not_active IP Right Cessation
- 2002-07-11 AU AU2002318302A patent/AU2002318302B2/en not_active Ceased
- 2002-07-11 MX MXPA04000249A patent/MXPA04000249A/es active IP Right Grant
- 2002-07-11 JP JP2003511771A patent/JP2005520780A/ja active Pending
- 2002-07-11 KR KR10-2004-7000312A patent/KR20040029360A/ko not_active Ceased
- 2002-07-11 EP EP02748129A patent/EP1411943A4/en not_active Withdrawn
- 2002-07-11 CA CA2453510A patent/CA2453510C/en not_active Expired - Fee Related
- 2002-07-11 WO PCT/US2002/022039 patent/WO2003005962A2/en not_active Ceased
- 2002-07-11 NZ NZ565754A patent/NZ565754A/en not_active IP Right Cessation
- 2002-07-11 IL IL15931302A patent/IL159313A0/xx unknown
- 2002-07-16 US US10/195,974 patent/US7115631B2/en not_active Expired - Fee Related
-
2004
- 2004-04-08 US US10/820,397 patent/US20040204456A1/en not_active Abandoned
-
2006
- 2006-04-11 US US11/402,385 patent/US20060183774A1/en not_active Abandoned
-
2009
- 2009-12-17 US US12/640,734 patent/US20100093797A1/en not_active Abandoned
-
2011
- 2011-06-30 US US13/172,977 patent/US20110257227A1/en not_active Abandoned
-
2012
- 2012-10-26 US US13/661,472 patent/US20130053414A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2003005962A2 (en) | 2003-01-23 |
| US20020198234A1 (en) | 2002-12-26 |
| US20060183774A1 (en) | 2006-08-17 |
| US20040204456A1 (en) | 2004-10-14 |
| EP1411943A4 (en) | 2005-09-28 |
| MXPA04000249A (es) | 2004-05-04 |
| CA2453510C (en) | 2012-03-20 |
| US20130053414A1 (en) | 2013-02-28 |
| CA2453510A1 (en) | 2003-01-23 |
| NZ565754A (en) | 2009-05-31 |
| EP1411943A2 (en) | 2004-04-28 |
| US20020022640A1 (en) | 2002-02-21 |
| WO2003005962A3 (en) | 2003-06-12 |
| AU2002318302B2 (en) | 2007-03-15 |
| JP2005520780A (ja) | 2005-07-14 |
| IL159313A0 (en) | 2004-06-01 |
| US20100093797A1 (en) | 2010-04-15 |
| KR20040029360A (ko) | 2004-04-06 |
| US7115631B2 (en) | 2006-10-03 |
| US20110257227A1 (en) | 2011-10-20 |
| US6486177B2 (en) | 2002-11-26 |
| AU2002318302C1 (en) | 2003-01-29 |
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| RENW | Renewal (renewal fees accepted) | ||
| PSEA | Patent sealed | ||
| RENW | Renewal (renewal fees accepted) | ||
| LAPS | Patent lapsed |