NZ326039A - Process for making 3,4-dihydro-pyrimidin-2(1h)-one derivatives - Google Patents

Process for making 3,4-dihydro-pyrimidin-2(1h)-one derivatives

Info

Publication number
NZ326039A
NZ326039A NZ326039A NZ32603996A NZ326039A NZ 326039 A NZ326039 A NZ 326039A NZ 326039 A NZ326039 A NZ 326039A NZ 32603996 A NZ32603996 A NZ 32603996A NZ 326039 A NZ326039 A NZ 326039A
Authority
NZ
New Zealand
Prior art keywords
pyrimidin
dihydro
derivatives
making
Prior art date
Application number
NZ326039A
Other languages
English (en)
Inventor
Essa H Hu
Daniel R Sidler
Ulf H Dolling
Michael A Patane
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9617968.4A external-priority patent/GB9617968D0/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of NZ326039A publication Critical patent/NZ326039A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/20—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D239/22—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
NZ326039A 1995-12-14 1996-12-12 Process for making 3,4-dihydro-pyrimidin-2(1h)-one derivatives NZ326039A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US864195P 1995-12-14 1995-12-14
GBGB9617968.4A GB9617968D0 (en) 1996-08-28 1996-08-28 Process for making dihydropyrimidinones
PCT/US1996/019651 WO1997021687A1 (en) 1995-12-14 1996-12-12 Process for making dihydropyrimidinones

Publications (1)

Publication Number Publication Date
NZ326039A true NZ326039A (en) 1999-08-30

Family

ID=26309937

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ326039A NZ326039A (en) 1995-12-14 1996-12-12 Process for making 3,4-dihydro-pyrimidin-2(1h)-one derivatives

Country Status (11)

Country Link
EP (1) EP0882026A4 (xx)
JP (1) JP2000501734A (xx)
KR (1) KR19990072125A (xx)
AU (1) AU705409B2 (xx)
BR (1) BR9611933A (xx)
CA (1) CA2238924A1 (xx)
CZ (1) CZ184098A3 (xx)
NZ (1) NZ326039A (xx)
PL (1) PL327147A1 (xx)
SK (1) SK77398A3 (xx)
WO (1) WO1997021687A1 (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2297889A1 (en) * 1997-08-05 1999-02-18 Norihiro Ikemoto Alpha 1a adrenergic receptor antagonist
US6207444B1 (en) 1997-08-05 2001-03-27 Merck & Co., Inc. Enzymatic process of making alpha 1a adrenergic receptor antagonists using protease
WO2003006439A1 (en) 2001-07-13 2003-01-23 Astrazeneca Uk Limited Preparation of aminopyrimidine compounds
AU2003237544A1 (en) 2002-06-17 2003-12-31 Vittal Mallya Scientific Research Foundation Substituted dihydropyrimidines and dihydropyrimidinethiones as calcium channel blockers
AU2003270562B2 (en) 2002-09-12 2010-09-16 Diakron Pharmaceuticals, Inc. Calcium channel blockers
DK1578731T3 (da) 2002-12-16 2010-02-15 Astrazeneca Uk Ltd Fremgangsmåde til fremstilling af pyrimidinforbindelser
GB0428328D0 (en) 2004-12-24 2005-02-02 Astrazeneca Uk Ltd Chemical process
CN105037277B (zh) * 2015-07-09 2017-12-01 华南理工大学 一种3，4‑二氢嘧啶酮/硫酮类杂环化合物的合成方法
CN105233870A (zh) * 2015-09-24 2016-01-13 齐鲁工业大学 具有催化二氢嘧啶酮类化合物的吡啶乙烯配位聚合物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS60214778A (ja) * 1984-03-08 1985-10-28 Suntory Ltd Ν置換３，４−ジヒドロピリミジン誘導体ならびにその製造法および用途
US4675321A (en) * 1986-02-07 1987-06-23 Merck & Co., Inc. Substituted pyrimidines useful as calcium channel blockers
US5459145A (en) * 1988-01-19 1995-10-17 Pfizer Inc. Calcium independent camp phosphodiesterase inhibitor antidepressant
CZ279305B6 (cs) * 1992-01-24 1995-04-12 Lonza A.G. Kyseliny 2-halogen pyrimidin-4-karboxylové, způsob jejich přípravy a jejich použití pro přípravu derivátů substituovaných pyrimidinů-4-karboxylový ch kyselin

Also Published As

Publication number Publication date
AU705409B2 (en) 1999-05-20
BR9611933A (pt) 1999-03-02
AU1331697A (en) 1997-07-03
PL327147A1 (en) 1998-11-23
CA2238924A1 (en) 1997-06-19
KR19990072125A (ko) 1999-09-27
JP2000501734A (ja) 2000-02-15
WO1997021687A1 (en) 1997-06-19
SK77398A3 (en) 1999-02-11
EP0882026A1 (en) 1998-12-09
MX9804766A (es) 1998-10-31
EP0882026A4 (en) 1999-04-07
CZ184098A3 (cs) 1998-11-11

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