NO993928L - Farmasöytisk blanding for oral administrasjon av heterosykliske forbindelser i form av kvaternær ammonium - Google Patents

Farmasöytisk blanding for oral administrasjon av heterosykliske forbindelser i form av kvaternær ammonium

Info

Publication number
NO993928L
NO993928L NO993928A NO993928A NO993928L NO 993928 L NO993928 L NO 993928L NO 993928 A NO993928 A NO 993928A NO 993928 A NO993928 A NO 993928A NO 993928 L NO993928 L NO 993928L
Authority
NO
Norway
Prior art keywords
pharmaceutical composition
weight
quaternary ammonium
oral administration
heterocyclic compounds
Prior art date
Application number
NO993928A
Other languages
English (en)
Other versions
NO993928D0 (no
Inventor
Jean-Claude Gautier
Xavier Boulenc
Regine Bellamy
Bernard Abramovici
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Publication of NO993928D0 publication Critical patent/NO993928D0/no
Publication of NO993928L publication Critical patent/NO993928L/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)

Abstract

Oppfinnelsen angår et farmasøytisk preparat for oral administrering av heterocykliske forbindelser i form av kvaternært ammonium, inneholdende aktivt prinsipp hydrofilt løsemiddel anionisk overflateaktivt middel polysorbat 80 makrogoglycerid QS opptil 0,1 tiM5vekt% O til 60 vekt% O til 5 vekt% O til 5 vekt% 100vekt%, forutsatt at minst en bestanddel valgt fra det hydrofile løsemiddel og anioniske overflateaktive middel er til stede.
NO993928A 1997-02-17 1999-08-16 Farmasöytisk blanding for oral administrasjon av heterosykliske forbindelser i form av kvaternær ammonium NO993928L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9701825A FR2759584B1 (fr) 1997-02-17 1997-02-17 Composition pharmaceutique pour l'administration orale de composes heterocycliques sous forme ammonium quaternaire
PCT/FR1998/000298 WO1998035662A1 (fr) 1997-02-17 1998-02-17 Composition pharmaceutique pour l'administration orale de composes heterocycliques sous forme ammonium quaternaire

Publications (2)

Publication Number Publication Date
NO993928D0 NO993928D0 (no) 1999-08-16
NO993928L true NO993928L (no) 1999-08-16

Family

ID=9503804

Family Applications (1)

Application Number Title Priority Date Filing Date
NO993928A NO993928L (no) 1997-02-17 1999-08-16 Farmasöytisk blanding for oral administrasjon av heterosykliske forbindelser i form av kvaternær ammonium

Country Status (11)

Country Link
EP (1) EP0969825A1 (no)
JP (1) JP2001511795A (no)
AR (1) AR011805A1 (no)
AU (1) AU6404998A (no)
BR (1) BR9807694A (no)
CA (1) CA2281560A1 (no)
FR (1) FR2759584B1 (no)
HR (1) HRP980075A2 (no)
NO (1) NO993928L (no)
WO (1) WO1998035662A1 (no)
ZA (1) ZA981289B (no)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102188424B (zh) * 2011-03-23 2013-03-27 浙江理工大学 Sr140333的抗血癌作用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2676055B1 (fr) * 1991-05-03 1993-09-03 Sanofi Elf Composes polycycliques amines et leurs enantiomeres, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2676054B1 (fr) * 1991-05-03 1993-09-03 Sanofi Elf Nouveaux composes n-alkylenepiperidino et leurs enantiomeres, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2688219B1 (fr) * 1992-03-03 1994-07-08 Sanofi Elf Sels d'ammonium quaternaires de composes aromatiques amines, leur preparation et compositions pharmaceutiques les contenant.
FR2696178B1 (fr) * 1992-09-30 1994-12-30 Sanofi Elf Amides basiques quaternaires, procédé pour leur préparation et compositions pharmaceutiques en contenant.
FR2717804B1 (fr) * 1994-03-25 1996-06-21 Sanofi Sa Sels de composés hétéroaromatiques azotés substitués, procédé pour leur préparation et compositions pharmaceutiques en contenant.
CN1067385C (zh) * 1994-08-25 2001-06-20 默里尔药物公司 用于治疗变应性疾病的新的取代的哌啶类化合物
FR2725986B1 (fr) * 1994-10-21 1996-11-29 Adir Nouveaux derives de piperidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2725900B1 (fr) * 1994-10-21 1997-07-18 Sanofi Sa Utilisation d'antagonistes des recepteurs nk1 pour la preparation de medicaments a action cardioregulatrice
FR2729951B1 (fr) * 1995-01-30 1997-04-18 Sanofi Sa Nouveaux composes heterocycliques, procede pour leur preparation et compositions pharmaceutiques en contenant
FR2729954B1 (fr) * 1995-01-30 1997-08-01 Sanofi Sa Composes heterocycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant

Also Published As

Publication number Publication date
EP0969825A1 (fr) 2000-01-12
NO993928D0 (no) 1999-08-16
WO1998035662A1 (fr) 1998-08-20
HRP980075A2 (en) 1998-10-31
AR011805A1 (es) 2000-09-13
JP2001511795A (ja) 2001-08-14
FR2759584A1 (fr) 1998-08-21
ZA981289B (en) 1998-08-26
FR2759584B1 (fr) 1999-06-11
BR9807694A (pt) 2000-03-21
AU6404998A (en) 1998-09-08
CA2281560A1 (en) 1998-08-20

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