NO950501L - Process for Obtaining 3-α2 [4- (6-Fluoro-benzo [daisoxazol-3-yl) piperidin-1-yl] -ethyl-2-methyl-6,7,8,9-tetrahydro-4H-pyrido [1 2-aÅpyrimidin-4-one - Google Patents

Process for Obtaining 3-α2 [4- (6-Fluoro-benzo [daisoxazol-3-yl) piperidin-1-yl] -ethyl-2-methyl-6,7,8,9-tetrahydro-4H-pyrido [1 2-aÅpyrimidin-4-one

Info

Publication number
NO950501L
NO950501L NO950501A NO950501A NO950501L NO 950501 L NO950501 L NO 950501L NO 950501 A NO950501 A NO 950501A NO 950501 A NO950501 A NO 950501A NO 950501 L NO950501 L NO 950501L
Authority
NO
Norway
Prior art keywords
daisoxazol
aåpyrimidin
pyrido
piperidin
benzo
Prior art date
Application number
NO950501A
Other languages
Norwegian (no)
Other versions
NO306022B1 (en
NO950501D0 (en
Inventor
Pere Dalmases Barjoan
Francisco Marquillas Olondritz
Joan Huguet Clotet
Ana Bosch Rovira
Juan Carlos Del Castillo Nieto
Jose Maria Caldero Ges
Original Assignee
Vita Invest Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vita Invest Sa filed Critical Vita Invest Sa
Publication of NO950501D0 publication Critical patent/NO950501D0/en
Publication of NO950501L publication Critical patent/NO950501L/en
Publication of NO306022B1 publication Critical patent/NO306022B1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO950501A 1994-02-11 1995-02-09 Process for obtaining 3- {2- [4- (6-fluoro-benzo [d] isoxazol-3-yl) piperidin-1-yl] ethyl} -2-methyl-6,7,8,9-tetrahydro -4H-pyrido [1,2-a] pyrimidin-4-one NO306022B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES09400252A ES2074966B1 (en) 1994-02-11 1994-02-11 PROCEDURE FOR OBTAINING 3- (2- (4- (6-FLUORO-BENZO (D) ISOXAZOL-3-IL) PIPERIDIN-1-IL) -ETIL) -2-METHYL-6,7,8,9- TETRAHIDRO-4H-PIRIDO- (1,2-A) PIRIMIDIN-4-ONA.

Publications (3)

Publication Number Publication Date
NO950501D0 NO950501D0 (en) 1995-02-09
NO950501L true NO950501L (en) 1995-08-14
NO306022B1 NO306022B1 (en) 1999-09-06

Family

ID=8285178

Family Applications (1)

Application Number Title Priority Date Filing Date
NO950501A NO306022B1 (en) 1994-02-11 1995-02-09 Process for obtaining 3- {2- [4- (6-fluoro-benzo [d] isoxazol-3-yl) piperidin-1-yl] ethyl} -2-methyl-6,7,8,9-tetrahydro -4H-pyrido [1,2-a] pyrimidin-4-one

Country Status (14)

Country Link
KR (1) KR100221108B1 (en)
AT (1) AT405401B (en)
CZ (1) CZ286398B6 (en)
EG (1) EG20877A (en)
ES (1) ES2074966B1 (en)
FI (1) FI110000B (en)
GR (1) GR1002344B (en)
HU (1) HU222110B1 (en)
IS (1) IS1766B (en)
NO (1) NO306022B1 (en)
PL (1) PL181420B1 (en)
PT (1) PT101654B (en)
RU (1) RU2123004C1 (en)
SK (1) SK281752B6 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2101646B1 (en) * 1995-04-12 1998-04-01 Ferrer Int NEW COMPOUND DERIVED FROM CHROMENE.
ES2144355B1 (en) * 1997-12-30 2001-01-01 Ferrer Int COMPOUNDS DERIVED FROM THE CHROME.
EP1280804B1 (en) * 2000-05-05 2004-04-14 RPG Life Sciences Limited A process for the preparation of anti-psychotic 3- 2- 4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4h-pyrido 1,2,-a]pyrimidin-4-one
CA2419314C (en) 2000-08-14 2006-07-11 Teva Pharmaceutical Industries Ltd. Preparation of risperidone
KR20040034996A (en) 2002-10-18 2004-04-29 한미약품 주식회사 Improved method for the preparation of risperidone
WO2004043923A1 (en) 2002-11-13 2004-05-27 Synthon B.V. Process for making risperidone and intermediates therefor
BRPI0809837A2 (en) * 2007-04-19 2014-11-11 Youxin Li "COMPOSITION FOR TREATING MENTAL DISORDERS, BALANCE OF COMPOSITE FOR TREATING MENTAL DISORDERS, PHARMACEUTICAL COMPOSITION AND USE OF COMPOSITE FOR TREATING MENTAL DISORDERS"

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4352811A (en) * 1981-11-12 1982-10-05 Hoechst-Roussel Pharmaceuticals Inc. 3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles
US4804663A (en) * 1985-03-27 1989-02-14 Janssen Pharmaceutica N.V. 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
US4980365A (en) * 1987-07-13 1990-12-25 Hoechst-Roussel Pharmaceuticals Inc. N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents

Also Published As

Publication number Publication date
FI110000B (en) 2002-11-15
RU95101859A (en) 1997-03-20
KR950032196A (en) 1995-12-20
ES2074966A1 (en) 1995-09-16
PL181420B1 (en) 2001-07-31
NO306022B1 (en) 1999-09-06
HUT70169A (en) 1995-09-28
PT101654A (en) 1995-09-12
AT405401B (en) 1999-08-25
SK281752B6 (en) 2001-07-10
NO950501D0 (en) 1995-02-09
IS4259A (en) 1995-08-12
CZ286398B6 (en) 2000-04-12
CZ32995A3 (en) 1995-09-13
RU2123004C1 (en) 1998-12-10
ES2074966B1 (en) 1996-06-16
HU9500418D0 (en) 1995-03-28
IS1766B (en) 2001-03-15
FI950579A (en) 1995-08-12
GR1002344B (en) 1996-05-24
FI950579A0 (en) 1995-02-10
SK15695A3 (en) 1995-10-11
PT101654B (en) 2002-01-30
HU222110B1 (en) 2003-04-28
EG20877A (en) 2000-05-31
PL307200A1 (en) 1995-08-21
ATA24995A (en) 1998-12-15
KR100221108B1 (en) 1999-09-15

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