NO903113D0 - 2-IMINO 3-HETEROCYCLYLALKYL BENZOTIAZOLINE DERIVATIVES AND THEIR PREPARATION. - Google Patents

2-IMINO 3-HETEROCYCLYLALKYL BENZOTIAZOLINE DERIVATIVES AND THEIR PREPARATION.

Info

Publication number
NO903113D0
NO903113D0 NO903113A NO903113A NO903113D0 NO 903113 D0 NO903113 D0 NO 903113D0 NO 903113 A NO903113 A NO 903113A NO 903113 A NO903113 A NO 903113A NO 903113 D0 NO903113 D0 NO 903113D0
Authority
NO
Norway
Prior art keywords
preparation
benzotiazoline
heterocyclylalkyl
imino
derivatives
Prior art date
Application number
NO903113A
Other languages
Norwegian (no)
Other versions
NO175590B (en
NO903113L (en
NO175590C (en
Inventor
Patrick Jimonet
Joseph Le Blevec
Conception Nemecek
Original Assignee
Rhone Poulenc Sante
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR8909483A external-priority patent/FR2649704B1/en
Priority claimed from FR9005889A external-priority patent/FR2661910B1/en
Application filed by Rhone Poulenc Sante filed Critical Rhone Poulenc Sante
Publication of NO903113D0 publication Critical patent/NO903113D0/en
Publication of NO903113L publication Critical patent/NO903113L/en
Publication of NO175590B publication Critical patent/NO175590B/en
Publication of NO175590C publication Critical patent/NO175590C/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D277/82—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Steroid Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

Compounds of formula: <IMAGE> in which R1 denotes a substituted 1-piperazinyl, substituted 1,2,3,6-tetrahydro-1-pyridyl or substituted piperidino radical, R2 denotes a polyfluoroalkoxy radical and n is equal to 2 or 3, salts of these compounds with an acid, processes for their preparation and medications containing them.
NO903113A 1989-07-13 1990-07-12 Analogous Process for Preparation of 2-Imino-3-Heterocyclylalkylbenzothiazoline Derivatives and Their Preparation NO175590C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8909483A FR2649704B1 (en) 1989-07-13 1989-07-13 IMINO-2 ETHYL-3 BENZOTHIAZOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND MEDICINAL PRODUCTS CONTAINING THEM
FR9005889A FR2661910B1 (en) 1990-05-11 1990-05-11 IMINO-2 HETEROCYCLYLALKYL-3 BENZOTHIAZOLINE DERIVATIVES, THEIR PREPARATION AND THE MEDICINAL PRODUCTS CONTAINING THEM.

Publications (4)

Publication Number Publication Date
NO903113D0 true NO903113D0 (en) 1990-07-12
NO903113L NO903113L (en) 1991-01-14
NO175590B NO175590B (en) 1994-07-25
NO175590C NO175590C (en) 1994-11-02

Family

ID=26227474

Family Applications (1)

Application Number Title Priority Date Filing Date
NO903113A NO175590C (en) 1989-07-13 1990-07-12 Analogous Process for Preparation of 2-Imino-3-Heterocyclylalkylbenzothiazoline Derivatives and Their Preparation

Country Status (20)

Country Link
EP (1) EP0409692B1 (en)
JP (1) JPH0386871A (en)
AT (1) ATE102612T1 (en)
AU (1) AU624972B2 (en)
CA (1) CA2021031A1 (en)
CZ (1) CZ281164B6 (en)
DE (1) DE69007196T2 (en)
DK (1) DK0409692T3 (en)
ES (1) ES2062445T3 (en)
FI (1) FI93109C (en)
HU (1) HU210827B (en)
IE (1) IE63318B1 (en)
IL (1) IL95053A (en)
NO (1) NO175590C (en)
NZ (1) NZ234487A (en)
PL (2) PL164326B1 (en)
PT (1) PT94701B (en)
RU (1) RU1836368C (en)
SK (1) SK342590A3 (en)
YU (1) YU47723B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2674853B1 (en) * 1991-04-03 1995-01-20 Synthelabo PIPERIDINYLGUANIDINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION.
FR2678619B1 (en) * 1991-07-04 1993-09-17 Rhone Poulenc Rorer Sa DERIVATIVES OF 1,2,4-THIADIAZOLO [3,4-B] BENZOTHIAZOLE, THEIR PREPARATION AND THE MEDICINAL PRODUCTS CONTAINING THEM.
FR2696457B1 (en) * 1992-10-02 1994-11-25 Rhone Poulenc Rorer Sa Derivatives of 3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-dioxide, their preparation and the medicaments containing them.
CA2130096A1 (en) * 1992-04-15 1993-10-28 Jean-Claude Aloup 3,4-dihydro-2h-1,2,4-benzothiadiazine-1,1-dioxide-3-carboxylic acid derivatives; process for preparing the same and therapeutic agents containing them
US5889010A (en) * 1995-05-18 1999-03-30 Pfizer Inc. Benzimidazole derivatives having dopaminergic activity

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2631163B2 (en) * 1976-07-10 1978-06-29 Basf Ag, 6700 Ludwigshafen Process for the preparation of 2-iminobenzothiazoles
FR2492258A1 (en) * 1980-10-17 1982-04-23 Pharmindustrie NEW AMINO-2 TRIFLUOROMETHOXY-6 BENZOTHIAZOLE-BASED MEDICINAL PRODUCT
EP0375510B1 (en) * 1988-12-15 1992-11-11 Rhone-Poulenc Sante 2-imino-6-polyfluoroalcoxy-benzothiazole derivatives, process for their preparation and medicaments containing them
FR2649701B2 (en) * 1988-12-15 1991-11-22 Rhone Poulenc Sante IMINO-2 BENZOTHIAZOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM

Also Published As

Publication number Publication date
FI93109B (en) 1994-11-15
IL95053A0 (en) 1991-06-10
IE902551A1 (en) 1991-02-27
JPH0386871A (en) 1991-04-11
SK278908B6 (en) 1998-04-08
EP0409692A3 (en) 1991-03-27
DE69007196T2 (en) 1994-06-30
NZ234487A (en) 1992-04-28
HU904189D0 (en) 1990-12-28
HUT58732A (en) 1992-03-30
IL95053A (en) 1994-05-30
HU210827B (en) 1995-08-28
PL164326B1 (en) 1994-07-29
NO175590B (en) 1994-07-25
PT94701A (en) 1991-03-20
CZ342590A3 (en) 1996-01-17
FI903531A0 (en) 1990-07-12
NO903113L (en) 1991-01-14
CA2021031A1 (en) 1991-01-14
IE63318B1 (en) 1995-04-05
PL164152B1 (en) 1994-06-30
EP0409692A2 (en) 1991-01-23
FI93109C (en) 1995-02-27
EP0409692B1 (en) 1994-03-09
CZ281164B6 (en) 1996-07-17
DE69007196D1 (en) 1994-04-14
DK0409692T3 (en) 1994-04-05
PT94701B (en) 1997-03-31
ES2062445T3 (en) 1994-12-16
NO175590C (en) 1994-11-02
YU47723B (en) 1996-01-08
ATE102612T1 (en) 1994-03-15
SK342590A3 (en) 1998-04-08
AU5884790A (en) 1991-01-17
RU1836368C (en) 1993-08-23
AU624972B2 (en) 1992-06-25
YU133990A (en) 1992-07-20

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