NO874374L - PREPARATION OF PEPTIDE AMINOAL CYLAMIDES AND PEPTIDE HYDRAZIDES BY THE PHASE PHASE METHOD. - Google Patents

PREPARATION OF PEPTIDE AMINOAL CYLAMIDES AND PEPTIDE HYDRAZIDES BY THE PHASE PHASE METHOD.

Info

Publication number
NO874374L
NO874374L NO874374A NO874374A NO874374L NO 874374 L NO874374 L NO 874374L NO 874374 A NO874374 A NO 874374A NO 874374 A NO874374 A NO 874374A NO 874374 L NO874374 L NO 874374L
Authority
NO
Norway
Prior art keywords
peptide
phase
cylamides
aminoal
preparation
Prior art date
Application number
NO874374A
Other languages
Norwegian (no)
Other versions
NO172895B (en
NO874374D0 (en
NO172895C (en
Inventor
Gerhard Breipohl
Jochen Knolle
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of NO874374D0 publication Critical patent/NO874374D0/en
Publication of NO874374L publication Critical patent/NO874374L/en
Publication of NO172895B publication Critical patent/NO172895B/en
Publication of NO172895C publication Critical patent/NO172895C/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/58—Atrial natriuretic factor complex; Atriopeptin; Atrial natriuretic peptide [ANP]; Cardionatrin; Cardiodilatin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C07K1/042—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers characterised by the nature of the carrier
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Endocrinology (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Cardiology (AREA)
  • Analytical Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pyrane Compounds (AREA)

Abstract

Compounds of the formula I <IMAGE> in which A is hydrogen or an amino protective group, B is an amino acid residue, X is alkylene or aralkylene, Y<1>, Y<2>, Y<3> and Y<4> are identical or different and are hydrogen, methyl, methoxy or nitro, V is hydrogen or a carboxyl protective group, W is -[CH2]n- or -O-[CH2]n-, m is 0 or 1, n is 0 to 6 and p is 0 to 5, are prepared as described and used in the solid-phase synthesis.
NO874374A 1986-10-21 1987-10-20 PEPTID AMINOAL CYLAMIDS, THEIR USE FOR PREPARATION OF PEPTIDES, AND A PROCEDURE FOR THE PREPARATION OF SUCH PEPTIDES NO172895C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19863635670 DE3635670A1 (en) 1986-10-21 1986-10-21 SYNTHESIS OF PEPTIDE-AMINOALKYLAMIDES AND PEPTIDYHYDRAZIDES BY MEANS OF THE SOLID PHASE METHOD

Publications (4)

Publication Number Publication Date
NO874374D0 NO874374D0 (en) 1987-10-20
NO874374L true NO874374L (en) 1988-04-22
NO172895B NO172895B (en) 1993-06-14
NO172895C NO172895C (en) 1993-09-22

Family

ID=6312082

Family Applications (1)

Application Number Title Priority Date Filing Date
NO874374A NO172895C (en) 1986-10-21 1987-10-20 PEPTID AMINOAL CYLAMIDS, THEIR USE FOR PREPARATION OF PEPTIDES, AND A PROCEDURE FOR THE PREPARATION OF SUCH PEPTIDES

Country Status (18)

Country Link
EP (1) EP0264802B1 (en)
JP (1) JP2540564B2 (en)
KR (1) KR960013073B1 (en)
AT (1) ATE83244T1 (en)
AU (1) AU595390B2 (en)
CA (1) CA1340421C (en)
DE (2) DE3635670A1 (en)
DK (1) DK175126B1 (en)
ES (1) ES2052535T3 (en)
FI (1) FI88031C (en)
GR (1) GR3007231T3 (en)
HU (1) HU197719B (en)
IE (1) IE60864B1 (en)
IL (1) IL84195A (en)
NO (1) NO172895C (en)
NZ (1) NZ222204A (en)
PT (1) PT85952B (en)
ZA (1) ZA877862B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3926822A1 (en) 1989-08-14 1991-02-21 Hoechst Ag PEPTIDES WITH BRADYKININ ANTAGONISTIC EFFECT
EP0376218B1 (en) * 1988-12-27 1999-02-24 Perseptive Biosystems, Inc. Racemization free attachment of amino acids to solid phase
DE4408533A1 (en) 1994-03-14 1995-09-28 Hoechst Ag PNA synthesis using a base-labile amino protecting group
SI0946478T1 (en) * 1996-12-19 2007-06-30 Aventis Pharma Inc Process for the solid phase synthesis of aldehydes, ketones and hydroxamic acid compounds
GB9727123D0 (en) * 1997-12-22 1998-02-25 Int Centre Genetic Eng & Bio Synthesis of diamines
US6852789B2 (en) * 2002-02-15 2005-02-08 Degussa - Ag Glycols starting materials containing dispersed superfine ceramic powder coagulates capable of forming polyester molded bodies having high mechanical strength and transparency

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4108846A (en) * 1977-02-01 1978-08-22 Hoffmann-La Roche Inc. Solid phase synthesis with base N alpha-protecting group cleavage

Also Published As

Publication number Publication date
KR960013073B1 (en) 1996-09-30
FI874586A0 (en) 1987-10-19
GR3007231T3 (en) 1993-07-30
NZ222204A (en) 1989-10-27
DE3783009D1 (en) 1993-01-21
DK548287D0 (en) 1987-10-20
PT85952B (en) 1990-07-31
FI88031B (en) 1992-12-15
JP2540564B2 (en) 1996-10-02
ZA877862B (en) 1988-04-22
IL84195A0 (en) 1988-03-31
PT85952A (en) 1987-11-01
DE3635670A1 (en) 1988-04-28
IE872821L (en) 1988-04-21
AU595390B2 (en) 1990-03-29
DK548287A (en) 1988-04-22
NO172895B (en) 1993-06-14
IE60864B1 (en) 1994-08-24
CA1340421C (en) 1999-03-09
AU7993587A (en) 1988-04-28
ATE83244T1 (en) 1992-12-15
KR880005147A (en) 1988-06-28
DK175126B1 (en) 2004-06-07
EP0264802B1 (en) 1992-12-09
NO874374D0 (en) 1987-10-20
JPS63104951A (en) 1988-05-10
EP0264802A2 (en) 1988-04-27
FI874586A (en) 1988-04-22
FI88031C (en) 1993-03-25
HUT46706A (en) 1988-11-28
ES2052535T3 (en) 1994-07-16
NO172895C (en) 1993-09-22
HU197719B (en) 1989-05-29
EP0264802A3 (en) 1989-07-26
IL84195A (en) 1992-08-18

Similar Documents

Publication Publication Date Title
HUP9902576A1 (en) Novel erythromycin derivatives, method for preparing them, and use thereof as drugs
ATE69239T1 (en) OLIGOPEPTIDYLNITRILE DERIVATIVES, AGENTS CONTAINING THEM, PROCESSES FOR THEIR PREPARATION AND THEIR USE.
PL263885A1 (en) Method of obtaining novel derivatives of dihydrobenzofurane and chromate carbonamide
IL83141A0 (en) Solutions of oxazophorins having improved stability and their preparation
NO874374D0 (en) PREPARATION OF PEPTIDE AMINOAL CYLAMIDES AND PEPTIDE HYDRAZIDES BY THE PHASE PHASE METHOD.
DE58905462D1 (en) Enzyme-inhibiting amino acid derivatives, processes for their preparation, compositions containing them and their use.
IE850116L (en) Aspartic acid derivatives
DE68907746T2 (en) Benzhydrylamine derivatives.
ZA90866B (en) Cycloaminoalkoxyphenyl derivatives,a process for their preparation as well as the compositions containing them
EP0252030A3 (en) Derivatives of l-amino acyl l-carnitine, process for their preparation and pharmaceutical compositions having hepatoprotecting activity containing same
ES471606A2 (en) Preparation of benzylidene derivatives
JPS57175150A (en) Synthesis of dipeptide containing methylene group
ATE137741T1 (en) AMINO ACID DERIVATIVES FOR PEPTIDE SYNTHESIS
KR860003254A (en) Method for preparing octahydroindolo [2,3-a] quinolizine-1-yl-alkane carboxylic acid amide and acid addition salts thereof
JPS55145695A (en) Novel mixed acid anhydride
NO975150L (en) Process for the preparation of enantiomeric forms of aminoalkylaminophenylpropanoic acid

Legal Events

Date Code Title Description
MK1K Patent expired