NO20062187L - Furanderivat som EP4-reseptorantagonister - Google Patents
Furanderivat som EP4-reseptorantagonisterInfo
- Publication number
- NO20062187L NO20062187L NO20062187A NO20062187A NO20062187L NO 20062187 L NO20062187 L NO 20062187L NO 20062187 A NO20062187 A NO 20062187A NO 20062187 A NO20062187 A NO 20062187A NO 20062187 L NO20062187 L NO 20062187L
- Authority
- NO
- Norway
- Prior art keywords
- optionally substituted
- group
- alkyl
- receptor antagonists
- furan derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Det beskrives en forbindelse med formel (I) eller et salt, solvat eller kjemisk beskyttet derivat derav, der en av R2 og R5 er: (i) H eller en eventuelt substituert C1-4 alkyl gruppe; eller (ii) en eventuelt substituert C5-7 arylgruppe, og den andre av R2 og R5 er den andre gruppe; m og n kan være 0 eller 1 i det m + n = 1 eller 2, RN er H eller eventuelt substituert C1-4 alkyl, R3 er enten: (i) karboksy; (ii) en gruppe med formelen (II); (iii) en gruppe med formelen (III), der R eventuelt er substituert C1-7 alkyl, C5-20 aryl eller NRN3RN4 der RN3 og R N4 uavhengig er valgt blant eventuelt substituert C1-4 alkyl; eller (iv) tetrazol-5-yl.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0324269.0A GB0324269D0 (en) | 2003-10-16 | 2003-10-16 | EP4 receptor antagonists |
US51220003P | 2003-10-20 | 2003-10-20 | |
PCT/GB2004/004392 WO2005037812A1 (en) | 2003-10-16 | 2004-10-15 | Furan derivatives as ep4 receptor antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20062187L true NO20062187L (no) | 2006-07-07 |
Family
ID=34466432
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20062187A NO20062187L (no) | 2003-10-16 | 2006-05-15 | Furanderivat som EP4-reseptorantagonister |
Country Status (3)
Country | Link |
---|---|
KR (1) | KR20060097028A (no) |
DE (1) | DE602004018527D1 (no) |
NO (1) | NO20062187L (no) |
-
2004
- 2004-10-15 KR KR1020067009418A patent/KR20060097028A/ko active IP Right Grant
- 2004-10-15 DE DE602004018527T patent/DE602004018527D1/de active Active
-
2006
- 2006-05-15 NO NO20062187A patent/NO20062187L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
DE602004018527D1 (de) | 2009-01-29 |
KR20060097028A (ko) | 2006-09-13 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NO20092770L (no) | Nye aminopyrimidinderivater som PLK1-inhibitorer | |
ATE417841T1 (de) | Furanderivate als ep4-rezeptorantagonisten | |
NO20080717L (no) | Oksimderivat og fremgangsmate for fremstilling av dette | |
KR20050085991A (en) | Compounds exhibiting thrombopoietin receptor agonism | |
DE60222921D1 (de) | Amidderivate als inhibitoren der glycogensynthasekinase-3-beta | |
NO20063132L (no) | Naftyridinderivater og deres anvendelse som modulatorer av muskarinreceptorer | |
AP1902A (en) | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives and their use as antibacterials | |
WO2004035576A3 (en) | Pre-organized tricyclic integrase inhibitor compounds | |
TW200732329A (en) | Aryl-isoxazolo-4-yl-oxadiazole derivatives | |
NO331165B1 (no) | Derivater av dioksan-2-alkylkarbamater, fremgangsmate for fremstilling derav og anvendelse av de samme for fremstilling av medikamenter | |
TW200510326A (en) | Heterocyclic compounds and thrombopoietin receptor activators | |
HK1071565A1 (en) | 6,7-Dihydro-5H-pyrazolo Ä1,2-AÜ pyrazol-1-ones which control inflammatory cytokines | |
WO2008126732A1 (ja) | 縮合二環式ヘテロアリール誘導体 | |
WO2008051533A3 (en) | Benzimidazole compounds | |
WO2009116067A3 (en) | Novel derivatives of acyl cyanopyrrolidines | |
EP1364950A4 (en) | PYRIDOPYRIMIDINE OR NAPHTHYRIDINE DERIVATIVE | |
ATE259376T1 (de) | Heterozyklische verbindungen, ihre zwischenprodukte und elastase-inhibitoren | |
MY161992A (en) | Novel tetrahydroisoquinoline derivative | |
NO20063111L (no) | Fremgangsmate for fremstilling av tiazolpyrimidiner | |
WO2003072576A3 (en) | Oxazolidinone derivatives, processes for their preparation, and pharmaceutical compositions containing them | |
ATE449773T1 (de) | Homomorpholinoxazolidinone als antibakterielle mittel | |
NO20062187L (no) | Furanderivat som EP4-reseptorantagonister | |
RS54061B1 (en) | QUINOLINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONCERNING THEM, AND THEIR APPLICATIONS | |
MY139258A (en) | Carbamoyl-type benzofuran derivatives | |
WO2002098853A3 (en) | Inhibitors of cell proliferation, angiogenesis, fertility, and muscle contraction |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |