NO158505C - ANALOGY PROCEDURE FOR THE PREPARATION OF A THERAPEUTIC ACTIVE 7BETA-SUBSTITUTED MALONAMIDO-1-OXADADIA 7ALFA-METOXY-3- (1-METHYLTETRAZOL-5-YL) -TYOMETHYL CEPHALOSPORIN. - Google Patents

ANALOGY PROCEDURE FOR THE PREPARATION OF A THERAPEUTIC ACTIVE 7BETA-SUBSTITUTED MALONAMIDO-1-OXADADIA 7ALFA-METOXY-3- (1-METHYLTETRAZOL-5-YL) -TYOMETHYL CEPHALOSPORIN.

Info

Publication number
NO158505C
NO158505C NO771023A NO771023A NO158505C NO 158505 C NO158505 C NO 158505C NO 771023 A NO771023 A NO 771023A NO 771023 A NO771023 A NO 771023A NO 158505 C NO158505 C NO 158505C
Authority
NO
Norway
Prior art keywords
tyomethyl
oxadadia
7alfa
malonamido
7beta
Prior art date
Application number
NO771023A
Other languages
Norwegian (no)
Other versions
NO771023L (en
NO158505B (en
Inventor
Masayuki Narisada
Wataru Nagata
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP3340176A external-priority patent/JPS52122386A/en
Priority claimed from JP5029576A external-priority patent/JPS52133997A/en
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of NO771023L publication Critical patent/NO771023L/en
Publication of NO158505B publication Critical patent/NO158505B/en
Publication of NO158505C publication Critical patent/NO158505C/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D505/00Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
NO771023A 1976-03-25 1977-03-23 ANALOGY PROCEDURE FOR THE PREPARATION OF A THERAPEUTIC ACTIVE 7BETA-SUBSTITUTED MALONAMIDO-1-OXADADIA 7ALFA-METOXY-3- (1-METHYLTETRAZOL-5-YL) -TYOMETHYL CEPHALOSPORIN. NO158505C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP3340176A JPS52122386A (en) 1976-03-25 1976-03-25 Cephalosporin analogous compounds as antibacterials
JP5029576A JPS52133997A (en) 1976-04-30 1976-04-30 Cephalosporin antibiotics

Publications (3)

Publication Number Publication Date
NO771023L NO771023L (en) 1977-09-27
NO158505B NO158505B (en) 1988-06-13
NO158505C true NO158505C (en) 1988-09-21

Family

ID=26372085

Family Applications (2)

Application Number Title Priority Date Filing Date
NO771023A NO158505C (en) 1976-03-25 1977-03-23 ANALOGY PROCEDURE FOR THE PREPARATION OF A THERAPEUTIC ACTIVE 7BETA-SUBSTITUTED MALONAMIDO-1-OXADADIA 7ALFA-METOXY-3- (1-METHYLTETRAZOL-5-YL) -TYOMETHYL CEPHALOSPORIN.
NO862107A NO862107L (en) 1976-03-25 1986-05-28 ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE CEPHALOSPORINE DERIVATIVES.

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO862107A NO862107L (en) 1976-03-25 1986-05-28 ANALOGICAL PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE CEPHALOSPORINE DERIVATIVES.

Country Status (19)

Country Link
AR (1) AR224606A1 (en)
BG (1) BG31074A3 (en)
CY (1) CY1158A (en)
DD (1) DD129792A5 (en)
DE (1) DE2713370C2 (en)
DK (1) DK161331C (en)
ES (5) ES457174A1 (en)
GR (1) GR61146B (en)
HK (1) HK46882A (en)
HU (1) HU172720B (en)
IE (1) IE44794B1 (en)
IL (1) IL51743A (en)
MX (1) MX4348E (en)
NO (2) NO158505C (en)
NZ (1) NZ183687A (en)
PT (1) PT66346B (en)
RO (2) RO71742A (en)
SE (1) SE443143B (en)
YU (2) YU44038B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1557552A (en) * 1977-02-15 1979-12-12 Shionogi & Co 1 oxadethiacepham compounds
US4252953A (en) * 1979-05-01 1981-02-24 Eli Lilly And Company Antibiotic crystalline epimer
JPS60123490A (en) * 1983-12-07 1985-07-02 Shionogi & Co Ltd Malonyloxacephem carboxylic acid derivative

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL178005C (en) * 1972-11-06 1986-01-02 Merck & Co Inc METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION WITH ANTIBACTERIAL ACTION, AND METHOD FOR PREPARING A CEPHALOSPORINE ANTIBIOTIC.
US3962232A (en) * 1973-11-05 1976-06-08 Eli Lilly And Company 7-methoxycephalosporins
GB1449420A (en) * 1973-11-26 1976-09-15 Sankyo Co 7alpha-methoxycephalosporing derivatives

Also Published As

Publication number Publication date
DK131277A (en) 1977-09-26
ES457174A1 (en) 1978-08-16
YU44038B (en) 1990-02-28
YU44039B (en) 1990-02-28
YU173783A (en) 1983-12-31
DE2713370A1 (en) 1977-09-29
DK161331B (en) 1991-06-24
RO78228A (en) 1982-02-01
SE443143B (en) 1986-02-17
MX4348E (en) 1982-04-05
CY1158A (en) 1983-01-28
IE44794B1 (en) 1982-04-07
NO862107L (en) 1977-09-27
SE7703325L (en) 1977-09-26
DK161331C (en) 1991-12-09
RO71742A (en) 1982-02-26
YU173883A (en) 1983-12-31
ES469284A1 (en) 1978-11-16
BG31074A3 (en) 1981-10-15
IL51743A (en) 1980-10-26
DE2713370C2 (en) 1994-04-21
PT66346A (en) 1977-04-01
NZ183687A (en) 1979-01-11
ES469285A1 (en) 1979-09-16
ES469286A1 (en) 1979-09-16
AR224606A1 (en) 1981-12-30
IE44794L (en) 1977-09-25
ES469287A1 (en) 1979-09-16
PT66346B (en) 1978-08-16
HK46882A (en) 1982-11-19
HU172720B (en) 1978-11-28
DD129792A5 (en) 1978-02-08
NO771023L (en) 1977-09-27
GR61146B (en) 1978-09-27
NO158505B (en) 1988-06-13

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