NO157738C - ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE BENZOCSAZINONES AND BENZOCSAZOLINONES. - Google Patents

ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE BENZOCSAZINONES AND BENZOCSAZOLINONES.

Info

Publication number
NO157738C
NO157738C NO822932A NO822932A NO157738C NO 157738 C NO157738 C NO 157738C NO 822932 A NO822932 A NO 822932A NO 822932 A NO822932 A NO 822932A NO 157738 C NO157738 C NO 157738C
Authority
NO
Norway
Prior art keywords
benzocsazolinones
benzocsazinones
preparation
therapeutically active
analogue procedure
Prior art date
Application number
NO822932A
Other languages
Norwegian (no)
Other versions
NO157738B (en
NO822932L (en
Inventor
Kurt Schromm
Anton Mentrup
Ernst-Otto Renth
Armin Fugner
Original Assignee
Boehringer Ingelheim Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg
Publication of NO822932L publication Critical patent/NO822932L/en
Publication of NO157738B publication Critical patent/NO157738B/en
Publication of NO157738C publication Critical patent/NO157738C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/341,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/361,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
NO822932A 1981-09-01 1982-08-31 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE BENZOCSAZINONES AND BENZOCSAZOLINONES. NO157738C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19813134590 DE3134590A1 (en) 1981-09-01 1981-09-01 NEW BENZO HETEROCYCLES

Publications (3)

Publication Number Publication Date
NO822932L NO822932L (en) 1983-03-02
NO157738B NO157738B (en) 1988-02-01
NO157738C true NO157738C (en) 1988-05-11

Family

ID=6140603

Family Applications (1)

Application Number Title Priority Date Filing Date
NO822932A NO157738C (en) 1981-09-01 1982-08-31 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE BENZOCSAZINONES AND BENZOCSAZOLINONES.

Country Status (25)

Country Link
EP (1) EP0073505B1 (en)
JP (1) JPS5852278A (en)
KR (1) KR890000380B1 (en)
AR (2) AR231976A1 (en)
AT (1) ATE16703T1 (en)
AU (1) AU553589B2 (en)
CA (1) CA1180012A (en)
CS (1) CS236679B2 (en)
DD (1) DD204477A5 (en)
DE (2) DE3134590A1 (en)
DK (1) DK158664C (en)
ES (3) ES8308318A1 (en)
FI (1) FI78475C (en)
GB (1) GB2106105B (en)
GR (1) GR77275B (en)
HU (1) HU186112B (en)
IE (1) IE53615B1 (en)
IL (1) IL66683A0 (en)
NO (1) NO157738C (en)
NZ (1) NZ201777A (en)
PL (1) PL139375B1 (en)
PT (1) PT75478A (en)
SU (1) SU1149876A3 (en)
YU (1) YU42794B (en)
ZA (1) ZA826349B (en)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4554284A (en) * 1984-09-12 1985-11-19 Smithkline Beckman Corporation 7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones
DE3743265A1 (en) * 1987-12-19 1989-06-29 Boehringer Ingelheim Kg NEW AMMONIUM COMPOUNDS, THEIR MANUFACTURE AND USE
TW372967B (en) * 1994-12-27 1999-11-01 Kanebo Ltd 1,4 benzoxazine derivative, pharmaceutical composition containing the same and use thereof
DE10253282A1 (en) * 2002-11-15 2004-05-27 Boehringer Ingelheim Pharma Gmbh & Co. Kg Treatment of chronic obstructive pulmonary disease, using new or known N-substituted 2-amino-1-(benz-(1,4)-oxazin-3-on-8-yl)-ethanol derivative beta-mimetic agents, suitable for once-daily administration
US7056916B2 (en) 2002-11-15 2006-06-06 Boehringer Ingelheim Pharma Gmbh & Co. Kg Medicaments for the treatment of chronic obstructive pulmonary disease
PE20040950A1 (en) 2003-02-14 2005-01-01 Theravance Inc BIPHENYL DERIVATIVES AS AGONISTS OF ß2-ADRENERGIC RECEPTORS AND AS ANTAGONISTS OF MUSCARINAL RECEPTORS
GB0307856D0 (en) * 2003-04-04 2003-05-14 Novartis Ag Organic compounds
EP1613315B1 (en) * 2003-04-04 2009-01-21 Novartis AG Quinoline-2-one-derivatives for the treatment of airways diseases
EP1789394A1 (en) * 2004-05-13 2007-05-30 Boehringer Ingelheim International Gmbh Hydroxy-substituted benzo-condensed heterocycles for use as beta agonists in the treatment of respiratory diseases
US7307076B2 (en) 2004-05-13 2007-12-11 Boehringer Ingelheim International Gmbh Beta agonists for the treatment of respiratory diseases
DE102004024451A1 (en) 2004-05-14 2005-12-22 Boehringer Ingelheim Pharma Gmbh & Co. Kg Powder formulations for inhalation containing enantiomerically pure beta agonists
DE102004024454A1 (en) * 2004-05-14 2005-12-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Novel enantiomerically pure beta agonists, process for their preparation and their use as pharmaceuticals
US7220742B2 (en) 2004-05-14 2007-05-22 Boehringer Ingelheim International Gmbh Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments
DE102004024453A1 (en) * 2004-05-14 2006-01-05 Boehringer Ingelheim Pharma Gmbh & Co. Kg New long-acting bronchodilators for the treatment of respiratory diseases
US7745621B2 (en) 2004-05-14 2010-06-29 Boehringer Ingelheim International Gmbh Long acting bronchodilators for the treatment of respiratory diseases
DE102004024452A1 (en) * 2004-05-14 2005-12-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Aerosol formulation for the inhalation of beta agonists
PL1917253T3 (en) * 2005-08-15 2015-06-30 Boehringer Ingelheim Int Method for producing betamimetics
US20070088030A1 (en) 2005-10-10 2007-04-19 Barbara Niklaus-Humke Aerosol formulations for the inhalation of beta-agonists
GB0602778D0 (en) 2006-02-10 2006-03-22 Glaxo Group Ltd Novel compound
WO2008017638A1 (en) * 2006-08-07 2008-02-14 Boehringer Ingelheim International Gmbh Single enantiomer beta-agonists, methods for the production thereof and the use thereof as medication
UY30543A1 (en) * 2006-08-18 2008-03-31 Boehringer Ingelheim Int AEROSOL FORMULATION FOR INHALATION OF BETA- AGONISTS
US20100022770A1 (en) * 2007-01-25 2010-01-28 Boehringer Ingelheim International Gmbh Process for the manufacturing of beta mimetics

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2035749A1 (en) * 1969-02-06 1970-12-24 Bellon Labor Sa Roger
CA1041523A (en) * 1974-06-19 1978-10-31 Queen's University Preparation of 1-oxapenicillins and novel intermediates therefor

Also Published As

Publication number Publication date
GB2106105B (en) 1985-07-10
CS236679B2 (en) 1985-05-15
ES515380A0 (en) 1983-08-16
DE3134590A1 (en) 1983-03-10
PT75478A (en) 1982-09-01
DK158664B (en) 1990-07-02
CA1180012A (en) 1984-12-27
YU194982A (en) 1984-12-31
KR840001560A (en) 1984-05-07
PL238077A1 (en) 1984-04-09
GB2106105A (en) 1983-04-07
SU1149876A3 (en) 1985-04-07
AU553589B2 (en) 1986-07-24
IE822105L (en) 1983-03-01
EP0073505A1 (en) 1983-03-09
KR890000380B1 (en) 1989-03-15
FI822985L (en) 1983-03-02
AR231977A1 (en) 1985-04-30
ES521871A0 (en) 1984-06-16
JPS5852278A (en) 1983-03-28
DK389082A (en) 1983-03-02
AU8787482A (en) 1983-03-10
HU186112B (en) 1985-06-28
GR77275B (en) 1984-09-11
ES8308318A1 (en) 1983-08-16
FI78475B (en) 1989-04-28
IL66683A0 (en) 1982-12-31
ES8405778A1 (en) 1984-06-16
IE53615B1 (en) 1988-12-21
ATE16703T1 (en) 1985-12-15
AR231976A1 (en) 1985-04-30
JPH035392B2 (en) 1991-01-25
ES521870A0 (en) 1984-01-16
NZ201777A (en) 1985-08-30
FI822985A0 (en) 1982-08-30
ES8402279A1 (en) 1984-01-16
DD204477A5 (en) 1983-11-30
ZA826349B (en) 1984-04-25
DE3267702D1 (en) 1986-01-09
DK158664C (en) 1991-01-14
NO157738B (en) 1988-02-01
FI78475C (en) 1989-08-10
YU42794B (en) 1988-12-31
EP0073505B1 (en) 1985-11-27
NO822932L (en) 1983-03-02
PL139375B1 (en) 1987-01-31

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