AR231977A1 - PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 8- (1-HYDROXI-2-AMINO-ETIL) -2H-1,4-BENZOXAZIN-3- (44) -ONE AND OF 7- (1-HYDROXI-2-AMINO-ETIL ) -2-BENZOXAZOLINONE - Google Patents

PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 8- (1-HYDROXI-2-AMINO-ETIL) -2H-1,4-BENZOXAZIN-3- (44) -ONE AND OF 7- (1-HYDROXI-2-AMINO-ETIL ) -2-BENZOXAZOLINONE

Info

Publication number
AR231977A1
AR231977A1 AR294856A AR29485683A AR231977A1 AR 231977 A1 AR231977 A1 AR 231977A1 AR 294856 A AR294856 A AR 294856A AR 29485683 A AR29485683 A AR 29485683A AR 231977 A1 AR231977 A1 AR 231977A1
Authority
AR
Argentina
Prior art keywords
etil
hydroxi
amino
benzoxazolinone
benzoxazin
Prior art date
Application number
AR294856A
Other languages
Spanish (es)
Original Assignee
Boehringer Ingelheim Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg
Application granted granted Critical
Publication of AR231977A1 publication Critical patent/AR231977A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Feed For Specific Animals (AREA)
  • Fodder In General (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AR294856A 1981-09-01 1983-11-17 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 8- (1-HYDROXI-2-AMINO-ETIL) -2H-1,4-BENZOXAZIN-3- (44) -ONE AND OF 7- (1-HYDROXI-2-AMINO-ETIL ) -2-BENZOXAZOLINONE AR231977A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19813134590 DE3134590A1 (en) 1981-09-01 1981-09-01 NEW BENZO HETEROCYCLES

Publications (1)

Publication Number Publication Date
AR231977A1 true AR231977A1 (en) 1985-04-30

Family

ID=6140603

Family Applications (2)

Application Number Title Priority Date Filing Date
AR290473A AR231976A1 (en) 1981-09-01 1982-08-30 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 8- (1-HYDROXI-2-AMINO-ETIL) -2H-1,4-BENZOXAZIN-3- (4H) -ONE AND OF (7-1-HYDROXI-2-AMINO-ETIL ) -2-BENZOLINONE, AND NEW INTERMEDIATE COMPOUNDS FOR EXCLUSIVE USE IN SUCH PROCEDURE
AR294856A AR231977A1 (en) 1981-09-01 1983-11-17 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 8- (1-HYDROXI-2-AMINO-ETIL) -2H-1,4-BENZOXAZIN-3- (44) -ONE AND OF 7- (1-HYDROXI-2-AMINO-ETIL ) -2-BENZOXAZOLINONE

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AR290473A AR231976A1 (en) 1981-09-01 1982-08-30 PROCEDURE FOR THE PREPARATION OF DERIVATIVES OF 8- (1-HYDROXI-2-AMINO-ETIL) -2H-1,4-BENZOXAZIN-3- (4H) -ONE AND OF (7-1-HYDROXI-2-AMINO-ETIL ) -2-BENZOLINONE, AND NEW INTERMEDIATE COMPOUNDS FOR EXCLUSIVE USE IN SUCH PROCEDURE

Country Status (25)

Country Link
EP (1) EP0073505B1 (en)
JP (1) JPS5852278A (en)
KR (1) KR890000380B1 (en)
AR (2) AR231976A1 (en)
AT (1) ATE16703T1 (en)
AU (1) AU553589B2 (en)
CA (1) CA1180012A (en)
CS (1) CS236679B2 (en)
DD (1) DD204477A5 (en)
DE (2) DE3134590A1 (en)
DK (1) DK158664C (en)
ES (3) ES515380A0 (en)
FI (1) FI78475C (en)
GB (1) GB2106105B (en)
GR (1) GR77275B (en)
HU (1) HU186112B (en)
IE (1) IE53615B1 (en)
IL (1) IL66683A0 (en)
NO (1) NO157738C (en)
NZ (1) NZ201777A (en)
PL (1) PL139375B1 (en)
PT (1) PT75478A (en)
SU (1) SU1149876A3 (en)
YU (1) YU42794B (en)
ZA (1) ZA826349B (en)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4554284A (en) * 1984-09-12 1985-11-19 Smithkline Beckman Corporation 7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones
DE3743265A1 (en) * 1987-12-19 1989-06-29 Boehringer Ingelheim Kg NEW AMMONIUM COMPOUNDS, THEIR MANUFACTURE AND USE
TW372967B (en) * 1994-12-27 1999-11-01 Kanebo Ltd 1,4 benzoxazine derivative, pharmaceutical composition containing the same and use thereof
DE10253282A1 (en) * 2002-11-15 2004-05-27 Boehringer Ingelheim Pharma Gmbh & Co. Kg Treatment of chronic obstructive pulmonary disease, using new or known N-substituted 2-amino-1-(benz-(1,4)-oxazin-3-on-8-yl)-ethanol derivative beta-mimetic agents, suitable for once-daily administration
US7056916B2 (en) 2002-11-15 2006-06-06 Boehringer Ingelheim Pharma Gmbh & Co. Kg Medicaments for the treatment of chronic obstructive pulmonary disease
PE20040950A1 (en) 2003-02-14 2005-01-01 Theravance Inc BIPHENYL DERIVATIVES AS AGONISTS OF ß2-ADRENERGIC RECEPTORS AND AS ANTAGONISTS OF MUSCARINAL RECEPTORS
GB0307856D0 (en) * 2003-04-04 2003-05-14 Novartis Ag Organic compounds
AU2004226824B2 (en) * 2003-04-04 2008-05-01 Novartis Ag Quinoline-2-one-derivatives for the treatment of airways diseases
US7307076B2 (en) 2004-05-13 2007-12-11 Boehringer Ingelheim International Gmbh Beta agonists for the treatment of respiratory diseases
JP2007537187A (en) * 2004-05-13 2007-12-20 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Hydroxy-substituted benzofused heterocyclic compounds for use as beta agonists in the treatment of respiratory diseases
US7745621B2 (en) 2004-05-14 2010-06-29 Boehringer Ingelheim International Gmbh Long acting bronchodilators for the treatment of respiratory diseases
DE102004024451A1 (en) * 2004-05-14 2005-12-22 Boehringer Ingelheim Pharma Gmbh & Co. Kg Powder formulations for inhalation containing enantiomerically pure beta agonists
DE102004024452A1 (en) * 2004-05-14 2005-12-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Aerosol formulation for the inhalation of beta agonists
DE102004024453A1 (en) * 2004-05-14 2006-01-05 Boehringer Ingelheim Pharma Gmbh & Co. Kg New long-acting bronchodilators for the treatment of respiratory diseases
DE102004024454A1 (en) * 2004-05-14 2005-12-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Novel enantiomerically pure beta agonists, process for their preparation and their use as pharmaceuticals
US7220742B2 (en) 2004-05-14 2007-05-22 Boehringer Ingelheim International Gmbh Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments
CA2619402C (en) 2005-08-15 2015-02-03 Boehringer Ingelheim International Gmbh Method for producing betamimetics
US20070088030A1 (en) 2005-10-10 2007-04-19 Barbara Niklaus-Humke Aerosol formulations for the inhalation of beta-agonists
GB0602778D0 (en) 2006-02-10 2006-03-22 Glaxo Group Ltd Novel compound
EP2057152A1 (en) * 2006-08-07 2009-05-13 Boehringer Ingelheim International GmbH Single enantiomer beta-agonists, methods for the production thereof and the use thereof as medication
UY30543A1 (en) * 2006-08-18 2008-03-31 Boehringer Ingelheim Int AEROSOL FORMULATION FOR INHALATION OF BETA- AGONISTS
ES2370952T3 (en) * 2007-01-25 2011-12-26 Boehringer Ingelheim International Gmbh PROCEDURE FOR THE PREPARATION OF BETAMIMETICS.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2035749A1 (en) * 1969-02-06 1970-12-24 Bellon Labor Sa Roger
CA1041523A (en) * 1974-06-19 1978-10-31 Queen's University Preparation of 1-oxapenicillins and novel intermediates therefor

Also Published As

Publication number Publication date
YU194982A (en) 1984-12-31
JPS5852278A (en) 1983-03-28
ZA826349B (en) 1984-04-25
EP0073505B1 (en) 1985-11-27
ES521870A0 (en) 1984-01-16
AU553589B2 (en) 1986-07-24
ATE16703T1 (en) 1985-12-15
DK158664C (en) 1991-01-14
PL139375B1 (en) 1987-01-31
IE53615B1 (en) 1988-12-21
PT75478A (en) 1982-09-01
FI822985L (en) 1983-03-02
IL66683A0 (en) 1982-12-31
CS236679B2 (en) 1985-05-15
PL238077A1 (en) 1984-04-09
HU186112B (en) 1985-06-28
CA1180012A (en) 1984-12-27
DD204477A5 (en) 1983-11-30
NZ201777A (en) 1985-08-30
NO822932L (en) 1983-03-02
KR840001560A (en) 1984-05-07
NO157738B (en) 1988-02-01
ES8308318A1 (en) 1983-08-16
DE3134590A1 (en) 1983-03-10
ES521871A0 (en) 1984-06-16
DK158664B (en) 1990-07-02
FI78475B (en) 1989-04-28
NO157738C (en) 1988-05-11
IE822105L (en) 1983-03-01
GB2106105B (en) 1985-07-10
JPH035392B2 (en) 1991-01-25
YU42794B (en) 1988-12-31
ES515380A0 (en) 1983-08-16
FI78475C (en) 1989-08-10
ES8405778A1 (en) 1984-06-16
ES8402279A1 (en) 1984-01-16
FI822985A0 (en) 1982-08-30
AU8787482A (en) 1983-03-10
GB2106105A (en) 1983-04-07
KR890000380B1 (en) 1989-03-15
DE3267702D1 (en) 1986-01-09
EP0073505A1 (en) 1983-03-09
DK389082A (en) 1983-03-02
AR231976A1 (en) 1985-04-30
GR77275B (en) 1984-09-11
SU1149876A3 (en) 1985-04-07

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