NO146571C - ANALOGY PROCEDURE FOR THE PREPARATION OF ANTI-INFLAMMATORALLY ACTIVE IMIDAZOLS - Google Patents

ANALOGY PROCEDURE FOR THE PREPARATION OF ANTI-INFLAMMATORALLY ACTIVE IMIDAZOLS

Info

Publication number
NO146571C
NO146571C NO762754A NO762754A NO146571C NO 146571 C NO146571 C NO 146571C NO 762754 A NO762754 A NO 762754A NO 762754 A NO762754 A NO 762754A NO 146571 C NO146571 C NO 146571C
Authority
NO
Norway
Prior art keywords
inflammatorally
imidazols
active
preparation
analogy procedure
Prior art date
Application number
NO762754A
Other languages
Norwegian (no)
Other versions
NO146571B (en
NO762754L (en
Inventor
Saul Carl Cherkofsky
Thomas Ray Sharpe
Original Assignee
Du Pont
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont filed Critical Du Pont
Publication of NO762754L publication Critical patent/NO762754L/no
Publication of NO146571B publication Critical patent/NO146571B/en
Publication of NO146571C publication Critical patent/NO146571C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/84Sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
NO762754A 1975-08-11 1976-08-09 ANALOGY PROCEDURE FOR THE PREPARATION OF ANTI-INFLAMMATORALLY ACTIVE IMIDAZOLS NO146571C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US60365075A 1975-08-11 1975-08-11
US69128276A 1976-06-09 1976-06-09

Publications (3)

Publication Number Publication Date
NO762754L NO762754L (en) 1977-02-14
NO146571B NO146571B (en) 1982-07-19
NO146571C true NO146571C (en) 1982-10-27

Family

ID=27084480

Family Applications (1)

Application Number Title Priority Date Filing Date
NO762754A NO146571C (en) 1975-08-11 1976-08-09 ANALOGY PROCEDURE FOR THE PREPARATION OF ANTI-INFLAMMATORALLY ACTIVE IMIDAZOLS

Country Status (26)

Country Link
JP (1) JPS6011702B2 (en)
AR (2) AR215591A1 (en)
AU (1) AU508605B2 (en)
CA (1) CA1074327A (en)
CH (1) CH638791A5 (en)
DD (1) DD126244A5 (en)
DE (1) DE2635876A1 (en)
DK (1) DK361376A (en)
ES (2) ES450601A1 (en)
FI (1) FI66177C (en)
FR (1) FR2320745A1 (en)
GB (1) GB1516908A (en)
GR (1) GR61145B (en)
HU (1) HU174707B (en)
IE (1) IE44019B1 (en)
IL (1) IL50230A (en)
LU (1) LU75578A1 (en)
MX (1) MX3932E (en)
NL (1) NL7608915A (en)
NO (1) NO146571C (en)
NZ (1) NZ181731A (en)
PH (1) PH11857A (en)
PT (1) PT65464B (en)
SE (1) SE428686B (en)
SU (1) SU640662A3 (en)
YU (1) YU198176A (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK16778A (en) * 1977-02-09 1978-08-10 Du Pont IMIDAZOLE DERIVATIVES THEIR USES AND MANUFACTURE
LU77703A1 (en) * 1977-07-07 1979-03-26 Ciba Geigy Ag METHOD FOR PRODUCING BICYCLIC THIA-DIAZA COMPOUNDS
EP0004648B1 (en) * 1978-04-11 1982-08-25 Ciba-Geigy Ag Mercapto-imidazole derivatives, their preparation, mercapto-imidazole derivatives for the treatment of inflammatory diseases and their pharmaceutical compositions
DE2823197A1 (en) 1978-05-24 1979-11-29 Schering Ag NEW IMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM
US4308277A (en) * 1978-08-10 1981-12-29 Ciba-Geigy Corporation 2,4,5-Trisubstituted imidazolines and pharmaceutical compositions containing same
US4188397A (en) * 1978-09-22 1980-02-12 Smithkline Corporation 2,2-Alkyldiylbis(thio)bis(imidazoles)
US4215135A (en) * 1979-06-08 1980-07-29 E. I. Du Pont De Nemours And Company Antiinflammatory 2-substituted-1H-phenanthro[9,10-d]imidazoles
DE2856909A1 (en) * 1978-12-28 1980-07-17 Schering Ag NEW IMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM
GB8907656D0 (en) * 1989-04-05 1989-05-17 May & Baker Ltd New compositions of matter
KR20010014288A (en) * 1997-06-30 2001-02-26 오르토-맥네일 파마슈티칼, 인코퍼레이티드 2-Substituted imidazoles useful in the treatment of inflammatory diseases
DE10222103A1 (en) * 2002-05-17 2003-11-27 Merckle Gmbh Chem Pharm Fabrik New 2-(substituted thio)-imidazole derivatives are immunomodulators and cytokine release inhibitors, useful for treating diseases associated with immune system disorders, e.g. cancer or rheumatoid arthritis

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL6614808A (en) * 1965-10-21 1967-04-24
US3651080A (en) * 1969-11-07 1972-03-21 Ciba Geigy Corp Certain substituted 2-alkylmercaptoimidazole derivatives
US3636003A (en) * 1969-11-17 1972-01-18 Geigy Chem Corp Substituted 2-mercaptoimidazole derivatives
US3714179A (en) * 1970-09-08 1973-01-30 Searle & Co 1-alkyl-2-furfurylthioimidazoles and congeners
US3707475A (en) * 1970-11-16 1972-12-26 Pfizer Antiinflammatory imidazoles

Also Published As

Publication number Publication date
NL7608915A (en) 1977-02-15
GB1516908A (en) 1978-07-05
DD126244A5 (en) 1977-07-06
FI762290A (en) 1977-02-12
PH11857A (en) 1978-08-03
DK361376A (en) 1977-02-12
ES461193A1 (en) 1978-12-01
IL50230A (en) 1979-07-25
FR2320745A1 (en) 1977-03-11
PT65464B (en) 1978-08-02
LU75578A1 (en) 1978-04-13
ES450601A1 (en) 1978-01-16
NO146571B (en) 1982-07-19
AU508605B2 (en) 1980-03-27
DE2635876A1 (en) 1977-03-03
CA1074327A (en) 1980-03-25
AR218054A1 (en) 1980-05-15
FI66177B (en) 1984-05-31
HU174707B (en) 1980-03-28
FI66177C (en) 1984-09-10
NO762754L (en) 1977-02-14
JPS5223076A (en) 1977-02-21
FR2320745B1 (en) 1978-12-22
SE7607615L (en) 1977-02-12
IL50230A0 (en) 1976-10-31
MX3932E (en) 1981-10-02
IE44019B1 (en) 1981-07-29
AR215591A1 (en) 1979-10-31
NZ181731A (en) 1978-11-13
AU1671176A (en) 1978-02-16
SE428686B (en) 1983-07-18
SU640662A3 (en) 1978-12-30
PT65464A (en) 1976-09-01
JPS6011702B2 (en) 1985-03-27
GR61145B (en) 1978-09-27
IE44019L (en) 1977-02-11
YU198176A (en) 1982-10-31
CH638791A5 (en) 1983-10-14

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