NO146095C - Analogifremgangsmaate ved fremstilling av terapeutisk aktive kinazolin-derivater - Google Patents

Analogifremgangsmaate ved fremstilling av terapeutisk aktive kinazolin-derivater

Info

Publication number
NO146095C
NO146095C NO764135A NO764135A NO146095C NO 146095 C NO146095 C NO 146095C NO 764135 A NO764135 A NO 764135A NO 764135 A NO764135 A NO 764135A NO 146095 C NO146095 C NO 146095C
Authority
NO
Norway
Prior art keywords
preparation
therapeutically active
analogy procedure
chinazoline derivatives
chinazoline
Prior art date
Application number
NO764135A
Other languages
English (en)
Norwegian (no)
Other versions
NO146095B (no
NO764135L (xx
Inventor
Gianfedrico Doria
Ciriaco Romeo
Piernicola Giraldi
Francesco Lauria
Maria Luisa Corno
Piero Sberze
Marcello Tibolla
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of NO764135L publication Critical patent/NO764135L/no
Publication of NO146095B publication Critical patent/NO146095B/no
Publication of NO146095C publication Critical patent/NO146095C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/91Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/90Oxygen atoms with acyclic radicals attached in position 2 or 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/93Sulfur atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pulmonology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO764135A 1975-12-05 1976-12-03 Analogifremgangsmaate ved fremstilling av terapeutisk aktive kinazolin-derivater NO146095C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT29998/75A IT1050750B (it) 1975-12-05 1975-12-05 Derivati della 3.4 di idro chinazolina

Publications (3)

Publication Number Publication Date
NO764135L NO764135L (xx) 1977-06-07
NO146095B NO146095B (no) 1982-04-19
NO146095C true NO146095C (no) 1982-08-11

Family

ID=11228830

Family Applications (1)

Application Number Title Priority Date Filing Date
NO764135A NO146095C (no) 1975-12-05 1976-12-03 Analogifremgangsmaate ved fremstilling av terapeutisk aktive kinazolin-derivater

Country Status (22)

Country Link
US (1) US4251531A (xx)
JP (1) JPS5271485A (xx)
AT (1) AT355029B (xx)
AU (1) AU505660B2 (xx)
BE (1) BE848696A (xx)
CA (1) CA1084051A (xx)
CH (2) CH626073A5 (xx)
CS (1) CS194786B2 (xx)
DE (1) DE2654215A1 (xx)
DK (1) DK147855C (xx)
FI (1) FI64359C (xx)
FR (1) FR2333511A1 (xx)
GB (1) GB1523081A (xx)
HU (1) HU177817B (xx)
IL (1) IL50849A (xx)
IT (1) IT1050750B (xx)
NL (1) NL7613450A (xx)
NO (1) NO146095C (xx)
NZ (1) NZ182778A (xx)
SE (1) SE7613588L (xx)
SU (1) SU786894A3 (xx)
ZA (1) ZA766745B (xx)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL69274A (en) * 1982-08-05 1986-08-31 Erba Farmitalia (substituted amino)derivatives of 3-benzylidene-pyrrolo(2,1-b)quinazolin-9-ones and 6-benzylidene-pyrido(2,1-b)quinazolin-11-ones,their preparation and pharmaceutical compositions containing them
JPS5925224U (ja) * 1982-08-10 1984-02-16 株式会社根来 かばん
US4666913A (en) * 1985-11-22 1987-05-19 William H. Rorer, Inc. Hydroxy and aminothiazolyl-benzodiazinone compounds, cardiotonic compositions including the same, and their uses
GB8827988D0 (en) * 1988-11-30 1989-01-05 Smith Kline French Lab Chemical compounds
US5430148A (en) * 1992-03-31 1995-07-04 Agouron Pharmaceuticals, Inc. Antiproliferative quinazolines
WO1999061406A2 (en) * 1998-05-22 1999-12-02 Abbott Laboratories Antiangiogenic drug to treat cancer, arthritis and retinopathy
US6632961B1 (en) 1998-05-22 2003-10-14 Abbott Laboratories Antiangiogenic drug to treat cancer, arthritis and retinopathy
CO5170498A1 (es) * 1999-05-28 2002-06-27 Abbott Lab Biaril sulfonamidas son utiles como inhibidores de proliferacion celular
AU2002257195A1 (en) * 2001-04-23 2002-11-05 University Of Virginia Patent Foundation Synthesis and evaluation of novel phthalimide mimics as anti-angiogenic agents
CN100518740C (zh) * 2003-06-06 2009-07-29 阿里克斯股份公司 杂环化合物作为scce抑制剂的制药用途
KR101099409B1 (ko) * 2003-06-06 2011-12-27 아렉시스 악티에볼라그 피부 상태 또는 암 치료를 위한 scce 저해제로서의융합된 헤테로사이클 화합물의 용도
CA2659967C (en) * 2006-08-08 2014-05-13 Aska Pharmaceutical Co., Ltd. Quinazoline derivatives
PL2118074T3 (pl) 2007-02-01 2014-06-30 Resverlogix Corp Związki chemiczne do celów profilaktyki i leczenia chorób układu sercowo-naczyniowego
EP2408454A2 (en) 2009-03-18 2012-01-25 Resverlogix Corp. Novel anti-inflammatory agents
JP5813626B2 (ja) 2009-04-22 2015-11-17 レスバーロジックス コーポレイション 新規抗炎症剤
JO3789B1 (ar) 2015-03-13 2021-01-31 Resverlogix Corp التراكيب والوسائل العلاجية المعتمدة لمعالجة الامراض المتعلقة بالمتممة
GB201510254D0 (en) * 2015-06-12 2015-07-29 Syngenta Participations Ag Improvements in or relating to organic compounds
CA3105174A1 (en) * 2018-06-27 2020-01-02 Reborna Biosciences, Inc. Prophylactic or therapeutic agent for spinal muscular atrophy

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3696102A (en) * 1970-03-09 1972-10-03 Pfizer & Co C Process for the synthesis of substituted quinazolin-4-ones

Also Published As

Publication number Publication date
NL7613450A (nl) 1977-06-07
DK147855B (da) 1984-12-24
NZ182778A (en) 1978-07-28
DK147855C (da) 1985-06-10
FR2333511B1 (xx) 1979-03-02
IL50849A (en) 1980-11-30
ATA894376A (de) 1979-07-15
SE7613588L (sv) 1977-06-06
ZA766745B (en) 1977-10-26
GB1523081A (en) 1978-08-31
AU1947276A (en) 1978-05-18
SU786894A3 (ru) 1980-12-07
NO146095B (no) 1982-04-19
US4251531A (en) 1981-02-17
NO764135L (xx) 1977-06-07
AU505660B2 (en) 1979-11-29
CS194786B2 (en) 1979-12-31
FI64359C (fi) 1983-11-10
CA1084051A (en) 1980-08-19
AT355029B (de) 1980-02-11
FI763391A (xx) 1977-06-06
DE2654215A1 (de) 1977-06-16
CH626073A5 (xx) 1981-10-30
DK546776A (da) 1977-06-06
FI64359B (fi) 1983-07-29
HU177817B (en) 1981-12-28
IL50849A0 (en) 1977-01-31
CH626075A5 (xx) 1981-10-30
JPS5271485A (en) 1977-06-14
JPS5543464B2 (xx) 1980-11-06
IT1050750B (it) 1981-03-20
BE848696A (fr) 1977-03-16
FR2333511A1 (fr) 1977-07-01

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