NL7712570A - Piperidinederivaten, werkwijzen ter bereiding daarvan en farmaceutische mengsels die deze derivaten bevatten. - Google Patents

Piperidinederivaten, werkwijzen ter bereiding daarvan en farmaceutische mengsels die deze derivaten bevatten.

Info

Publication number
NL7712570A
NL7712570A NL7712570A NL7712570A NL7712570A NL 7712570 A NL7712570 A NL 7712570A NL 7712570 A NL7712570 A NL 7712570A NL 7712570 A NL7712570 A NL 7712570A NL 7712570 A NL7712570 A NL 7712570A
Authority
NL
Netherlands
Prior art keywords
derivatives
preparing
methods
mixtures containing
pharmaceutical mixtures
Prior art date
Application number
NL7712570A
Other languages
English (en)
Dutch (nl)
Original Assignee
Anphar Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anphar Sa filed Critical Anphar Sa
Publication of NL7712570A publication Critical patent/NL7712570A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • C07D211/58Nitrogen atoms attached in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
NL7712570A 1976-11-16 1977-11-15 Piperidinederivaten, werkwijzen ter bereiding daarvan en farmaceutische mengsels die deze derivaten bevatten. NL7712570A (nl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB47739/76A GB1574418A (en) 1976-11-16 1976-11-16 Piperidine derivatives

Publications (1)

Publication Number Publication Date
NL7712570A true NL7712570A (nl) 1978-05-18

Family

ID=10446086

Family Applications (2)

Application Number Title Priority Date Filing Date
NL7712559A NL7712559A (nl) 1976-11-16 1977-11-15 Piperidinederivaten, werkwijzen ter bereiding daarvan en farmaceutische preparaten die deze verbindingen bevatten.
NL7712570A NL7712570A (nl) 1976-11-16 1977-11-15 Piperidinederivaten, werkwijzen ter bereiding daarvan en farmaceutische mengsels die deze derivaten bevatten.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NL7712559A NL7712559A (nl) 1976-11-16 1977-11-15 Piperidinederivaten, werkwijzen ter bereiding daarvan en farmaceutische preparaten die deze verbindingen bevatten.

Country Status (13)

Country Link
US (1) US5026858A (xx)
JP (2) JPS5387365A (xx)
AT (2) AT360013B (xx)
AU (2) AU517004B2 (xx)
BE (2) BE860736A (xx)
CA (2) CA1094072A (xx)
DE (2) DE2751138A1 (xx)
ES (4) ES464145A1 (xx)
FR (2) FR2370733A1 (xx)
GB (1) GB1574418A (xx)
IE (2) IE46090B1 (xx)
NL (2) NL7712559A (xx)
ZA (2) ZA776587B (xx)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1574418A (en) * 1976-11-16 1980-09-03 Anphar Sa Piperidine derivatives
FR2546169B1 (fr) * 1983-05-20 1986-03-21 Delalande Sa N-oxydes de derives aminocycliques, leur procede de preparation et leur application en therapeutique
US4820715A (en) * 1984-06-28 1989-04-11 Bristol-Myers Company Anti-emetic quinuclidinyl benzamides
US4808624A (en) * 1984-06-28 1989-02-28 Bristol-Myers Company Pharmacologically active substituted benzamides
US5011992A (en) * 1984-06-28 1991-04-30 Bristol-Myers Squibb Company Pharmacologically active substituted benzamides
GB8519707D0 (en) * 1985-08-06 1985-09-11 Fordonal Sa Chemical compounds
US5721255A (en) * 1992-08-19 1998-02-24 Pfizer Inc. Substituted benzylamino nitrogen containing non-aromatic heterocycles
US5739135A (en) * 1993-09-03 1998-04-14 Bristol-Myers Squibb Company Inhibitors of microsomal triglyceride transfer protein and method
US5827875A (en) * 1996-05-10 1998-10-27 Bristol-Myers Squibb Company Inhibitors of microsomal triglyceride transfer protein and method
US5885983A (en) * 1996-05-10 1999-03-23 Bristol-Myers Squibb Company Inhibitors of microsomal triglyceride transfer protein and method
US5883109A (en) * 1996-07-24 1999-03-16 Bristol-Myers Squibb Company Method for lowering serum lipid levels employing an MTP inhibitor in combination with another cholesterol lowering drug
IL125658A0 (en) 1997-08-18 1999-04-11 Hoffmann La Roche Ccr-3 receptor antagonists
US6339087B1 (en) 1997-08-18 2002-01-15 Syntex (U.S.A.) Llc Cyclic amine derivatives-CCR-3 receptor antagonists
TR200101397T2 (tr) * 1998-11-20 2001-11-21 F.Hoffmann-La Roche Ag Piperidin CCR-3 reseptörü antagonistleri
FR2802206B1 (fr) * 1999-12-14 2005-04-22 Sod Conseils Rech Applic Derives de 4-aminopiperidine et leur utilisation en tant que medicament
TW200800953A (en) * 2002-10-30 2008-01-01 Theravance Inc Intermediates for preparing substituted 4-amino-1-(pyridylmethyl) piperidine
WO2005007645A1 (en) * 2003-07-11 2005-01-27 Theravance, Inc. Substituted 4-amino-1-benzylpiperidine compounds
WO2005053663A2 (en) * 2003-11-24 2005-06-16 Eli Lilly And Company Norepinephrine reuptake inhibitors useful for treatment of cognitive failure
DK1893603T3 (da) * 2005-06-02 2009-11-30 Hoffmann La Roche Piperidin-4-YL-amidderivater og anvendelsen deraf som SST-receptorundertype 5-antagonister
JP2009264436A (ja) 2008-04-23 2009-11-12 Funai Electric Co Ltd トルクリミッタ装置、トルクリミッタ装置を備えた表示画面旋回装置およびトルクリミッタ装置を含むテレビジョン装置

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1019781A (xx) * 1963-03-05
FR1407055A (fr) * 1963-03-05 1965-07-30 Ile De France Nouveau procédé de préparation de benzamides substitués
US3342826A (en) * 1964-01-13 1967-09-19 Ile De France Heterocyclic aminoalkyl benzamides
FR5916M (xx) * 1966-01-21 1968-05-06
US3577440A (en) * 1968-12-23 1971-05-04 Robins Co Inc A H 1-substituted-3-amido-pyrrolidines
GB1345872A (en) * 1970-09-03 1974-02-06 Wyeth John & Brother Ltd Amino-and acylamino-pyridine and hydropyridine derivatives
US3963745A (en) * 1972-04-03 1976-06-15 A. H. Robins Company, Incorporated Method for controlling emesis with N-(1-substituted-3-pyrrolidinyl)benzamides and thiobenzamides
DE2513136C3 (de) * 1974-03-21 1981-04-30 Anphar S.A., Madrid N-(1-Benzylpiperid-4-yl)-benzamide, Verfahren zu ihrer Herstellung und sie enthaltende pharmazeutische Präparate
GB1513631A (en) * 1976-02-17 1978-06-07 Gallardo Antonio Sa Piperidine derivatives
US4163789A (en) * 1976-02-17 1979-08-07 Anphar, S.A. Anti-psychotic (cycloalkenylalkylpiperidino) benzamides
GB1574418A (en) * 1976-11-16 1980-09-03 Anphar Sa Piperidine derivatives

Also Published As

Publication number Publication date
IE45989B1 (en) 1983-01-26
AU517830B2 (en) 1981-08-27
ATA817177A (de) 1980-05-15
FR2370733A1 (fr) 1978-06-09
ZA776587B (en) 1978-09-27
US5026858A (en) 1991-06-25
DE2751139A1 (de) 1978-05-24
AU3067277A (en) 1979-05-24
CA1095046A (en) 1981-02-03
ATA817077A (de) 1980-05-15
ZA776588B (en) 1978-08-30
DE2751138A1 (de) 1978-05-24
BE860736A (fr) 1978-03-01
CA1094072A (en) 1981-01-20
ES464146A1 (es) 1978-09-01
AT360013B (de) 1980-12-10
IE46090L (en) 1978-05-16
FR2370733B1 (xx) 1980-07-04
NL7712559A (nl) 1978-05-18
FR2370732B1 (xx) 1980-07-04
JPS6127388B2 (xx) 1986-06-25
AT360014B (de) 1980-12-10
AU3067377A (en) 1979-05-24
JPS5390267A (en) 1978-08-08
FR2370732A1 (fr) 1978-06-09
IE45989L (en) 1978-05-16
IE46090B1 (en) 1983-02-23
JPS6126782B2 (xx) 1986-06-21
ES464147A1 (es) 1978-09-01
BE860737A (fr) 1978-03-01
ES464145A1 (es) 1978-09-01
GB1574418A (en) 1980-09-03
JPS5387365A (en) 1978-08-01
AU517004B2 (en) 1981-07-02
ES464144A1 (es) 1978-09-01

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BC A request for examination has been filed
DNT Communications of changes of names of applicants whose applications have been laid open to public inspection

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A85 Still pending on 85-01-01
BV The patent application has lapsed