NL171587B - METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION WITH ANACTIVITY AGAINST BACTERIA, AND METHOD FOR PREPARING AN SUITABLE ACTIVE COMPOUND. - Google Patents

METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION WITH ANACTIVITY AGAINST BACTERIA, AND METHOD FOR PREPARING AN SUITABLE ACTIVE COMPOUND.

Info

Publication number
NL171587B
NL171587B NLAANVRAGE7410363,A NL7410363A NL171587B NL 171587 B NL171587 B NL 171587B NL 7410363 A NL7410363 A NL 7410363A NL 171587 B NL171587 B NL 171587B
Authority
NL
Netherlands
Prior art keywords
preparing
anactivity
active compound
pharmaceutical preparation
suitable active
Prior art date
Application number
NLAANVRAGE7410363,A
Other languages
Dutch (nl)
Other versions
NL7410363A (en
NL171587C (en
Original Assignee
Scherico Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/452,586 external-priority patent/US4029882A/en
Application filed by Scherico Ltd filed Critical Scherico Ltd
Publication of NL7410363A publication Critical patent/NL7410363A/en
Publication of NL171587B publication Critical patent/NL171587B/en
Application granted granted Critical
Publication of NL171587C publication Critical patent/NL171587C/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • C07H15/236—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2 a saccharide radical being substituted by an alkylamino radical in position 3 and by two substituents different from hydrogen in position 4, e.g. gentamicin complex, sisomicin, verdamycin
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
NLAANVRAGE7410363,A 1973-08-06 1974-08-01 METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION WITH ANACTIVITY AGAINST BACTERIA, AND METHOD FOR PREPARING AN SUITABLE ACTIVE COMPOUND. NL171587C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US38575173A 1973-08-06 1973-08-06
US45260074A 1974-03-19 1974-03-19
US05/452,586 US4029882A (en) 1974-03-19 1974-03-19 Selective acylation of the C-1 amino group of aminoglycoside antibiotics

Publications (3)

Publication Number Publication Date
NL7410363A NL7410363A (en) 1975-02-10
NL171587B true NL171587B (en) 1982-11-16
NL171587C NL171587C (en) 1983-04-18

Family

ID=27409729

Family Applications (1)

Application Number Title Priority Date Filing Date
NLAANVRAGE7410363,A NL171587C (en) 1973-08-06 1974-08-01 METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION WITH ANACTIVITY AGAINST BACTERIA, AND METHOD FOR PREPARING AN SUITABLE ACTIVE COMPOUND.

Country Status (20)

Country Link
AR (1) AR215834A1 (en)
BE (1) BE818431A (en)
BG (1) BG25804A3 (en)
CH (1) CH606076A5 (en)
CY (1) CY1018A (en)
DD (1) DD119037A5 (en)
DE (2) DE2462485C2 (en)
DK (1) DK146298C (en)
FI (1) FI62100C (en)
FR (1) FR2240015B1 (en)
GB (1) GB1473733A (en)
HK (1) HK55179A (en)
IE (1) IE40437B1 (en)
IL (1) IL45385A (en)
KE (1) KE2981A (en)
LU (1) LU70661A1 (en)
MY (1) MY8000090A (en)
NL (1) NL171587C (en)
NO (1) NO139483C (en)
SE (1) SE424994B (en)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1464401A (en) * 1974-10-26 1977-02-16 Pfizer Ltd Aminoglycosides
US4217446A (en) 1974-10-26 1980-08-12 Pfizer Inc. ωAmino-2-hydroxyalkyl derivatives of aminoglycoside antibiotics
FR2405266A1 (en) * 1975-09-08 1979-05-04 Scherico Ltd Antibacterial desoxystreptamines - esp 5-epi-4,6-di-(aminoglycosyl)-2-desoxystreptamines and 5-epi-(amino or azido)-5-desoxy derivs
DE2861947D1 (en) * 1977-06-10 1982-09-02 Bayer Ag Selectively protected 4,6-di-o-(aminoglycosyl)-1,3-diamino-cyclitols
US4282350A (en) * 1977-08-05 1981-08-04 Schering Corporation Selective 3"-N-acylation of 1,3"-di-N-unprotected-poly-N-protected-4,6-di-O-(aminoglycosyl)-1,3-diaminocyclitols
JPS5492951A (en) * 1977-12-29 1979-07-23 Shionogi & Co Ltd Novel aminoglycoside derivative
JPS5538345A (en) * 1978-09-11 1980-03-17 Shionogi & Co Ltd Novel aminoglycoside derivative
DE2840907A1 (en) * 1978-09-20 1980-04-03 Bayer Ag SELECTIVELY PROTECTED 4,6-DI-O- (AMINOGLYKOSYL) -1,3-DIAMINOCYCLITOLE
DE2928183A1 (en) * 1979-07-12 1981-01-29 Bayer Ag 1-N-ALKYLSISOMICIN DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS MEDICINAL PRODUCTS
CN1040177C (en) * 1993-04-23 1998-10-14 江苏省微生物研究所 1-N-ethyl gentamicin derivative and its preparing method
AU2008326297B2 (en) 2007-11-21 2012-11-08 Cipla USA, Inc. Antibacterial aminoglycoside analogs
WO2010132765A2 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010132759A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of dibekacin
WO2010132768A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of sisomicin
WO2010132760A1 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial derivatives of tobramycin
WO2010132757A2 (en) 2009-05-15 2010-11-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
CN101575311B (en) * 2009-06-19 2011-05-04 无锡好芳德药业有限公司 Method for preparing epiphysin

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1235311B (en) 1963-03-25 1967-03-02 Roussel Uclaf Process for the production of N-monophenylaethylneomycin B or its therapeutically acceptable salts

Also Published As

Publication number Publication date
IL45385A (en) 1978-10-31
IE40437B1 (en) 1979-06-06
FI62100B (en) 1982-07-30
NO139483C (en) 1979-03-21
NO139483B (en) 1978-12-11
BE818431A (en) 1975-02-03
DK146298C (en) 1984-02-06
NL7410363A (en) 1975-02-10
DE2437160A1 (en) 1975-02-20
LU70661A1 (en) 1975-05-21
BG25804A3 (en) 1978-12-12
DE2462485A1 (en) 1977-04-21
CY1018A (en) 1979-11-23
DE2437160B2 (en) 1979-01-04
FR2240015B1 (en) 1978-08-18
GB1473733A (en) 1977-05-18
DD119037A5 (en) 1976-04-05
CH606076A5 (en) 1978-10-13
AR215834A1 (en) 1979-11-15
DE2462485C2 (en) 1987-04-09
IL45385A0 (en) 1974-11-29
AU7194274A (en) 1976-02-05
DK146298B (en) 1983-08-29
NL171587C (en) 1983-04-18
SE7409946L (en) 1975-02-07
KE2981A (en) 1979-07-20
HK55179A (en) 1979-08-17
MY8000090A (en) 1980-12-31
SE424994B (en) 1982-08-23
IE40437L (en) 1975-02-06
DE2437160C3 (en) 1979-08-30
FI62100C (en) 1982-11-10
FI230474A (en) 1975-02-07
FR2240015A1 (en) 1975-03-07
NO742787L (en) 1975-03-03
DK412474A (en) 1975-04-01

Similar Documents

Publication Publication Date Title
NL164561C (en) METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION, AND METHOD FOR PREPARING AN AGAINST BACTERIA ACTIVE 7- (THIAZOLYLACETYLAMINO) CEPHOSPORIC ACID DERIVATIVE.
NL182369B (en) METHOD FOR PREPARING AN ORAL EXTENDED MEDICINE PREPARATION
NL179924C (en) METHOD FOR PREPARING AN ANTIBIOTIC AND METHOD FOR PREPARING C.Q. MANUFACTURE OF A PHARMACEUTICAL PREPARATION WITH AN EFFICIENCY AGAINST MICRO-ORGANISMS.
NL152864B (en) PROCEDURE FOR PREPARING A PHARMACEUTICAL PREPARATION WITH TRANSMETHYLING ACTIVITY, PREPARATIONS FORMED THEREFORE OBTAINED AND PROCEDURE FOR PREPARING THE ACTIVE SUBSTANCES THEREFORE.
NL170144C (en) METHOD FOR PREPARING AN ANTHELMINTIC PREPARATION AND AN ACTIVE SUBSTANCE SUITABLE THEREFOR.
NL179202C (en) PROCESS FOR PREPARING ALKYNYL CYCLOPROPANIC CARBOXYLATES, AND AT LEAST CONTAINING SUCH COMPOUND INSECTICIDE PREPARATIONS.
NL171587C (en) METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION WITH ANACTIVITY AGAINST BACTERIA, AND METHOD FOR PREPARING AN SUITABLE ACTIVE COMPOUND.
NL164273C (en) PROCESS FOR PREPARING A PHARMACEUTICAL PREPARATION BASED ON A PROSTAGLANDINE DERIVATIVE, THE PREPARED PHARMACEUTICAL PREPARATION, AND A METHOD FOR PREPARING A PROSTAGLANDINE DERIVATIVE SUITABLE FOR SUCH APPLICATION.
NL164184C (en) METHOD FOR PREPARING AN INSECTICIDE PREPARATION.
NL177688C (en) METHOD FOR PREPARING MEDICINAL PRODUCTS WITH ANALGETIC ACTIVITY, SO CONTAINED MEDICINAL PRODUCTS OBTAINED, AND METHOD FOR PREPARING A SUITABLE SALT.
NL181483C (en) METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION WITH ANTIBACTERIAL ACTIVITY; METHOD FOR PREPARING AN ANTIBACTERIAL ACTIVE COMPOUND
NL180422C (en) METHOD FOR PREPARING MEDICINES WITH AN ANTIMICROBE ACTIVITY, AND METHOD FOR PREPARING A CEPHALOSPORINE COMPOUND WITH A THIADIAZOLYLTHIOMETHYL OR TETRAZOLYLTHIOMETHYL-SUBOMETHYL-3-SUBTHOMETHYL
NL172057C (en) METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION AND AN ACTIVE INGREDIENT THEREFOR
NL165462C (en) METHOD FOR PREPARING A MEDICINAL PRODUCT, AND METHOD FOR PREPARING A COMPOUND SUITABLE FOR USE IN THE FOREGOING PROCESS
NL152246B (en) PROCEDURE FOR PREPARING A PREPARATION WITH ANTI-ARHYTHMIC ACTIVITY, PREPARATION FORMED, AND PROCEDURE FOR PREPARING A SUITABLE COMPOUND.
NL170283C (en) METHOD FOR PREPARING COMPOUNDS WITH ANALGETIC AND ANTI-INFLAMMATIVE ACTIVITY, AND PREPARED MEDICINES PRODUCED THEREFOR
NL181009C (en) PROCESS FOR PREPARING A PHARMACEUTICAL PREPARATION WITH ANTIBACTERIAL ACTION, AND METHOD FOR PREPARING A 7-BETA-ACYLAMINO-7-ALFA-METHOXY-3- (1-ALKYL-1H-TETRAZOL-5-YYL-THYL-THYL) CARBONIC ACID DERIVATIVE.
NL163707C (en) METHOD FOR PREPARING AN INSECTICIDE AND ACARICIDE PREPARATION
NL157655B (en) METHOD FOR PREPARING AN ANTIBIOTIC AND ANTIBIOTIC PREPARATIONS, AND FORMED MEDICINAL OR DISINFECTANT.
NL161154C (en) METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION CONTAINING A 4-OXAZOLINE-2-ON DERIVATIVE, FORMED PREPARATION AND METHOD FOR PREPARING A COMPOUND SUITABLE FOR USE IN THE FOREGOING PROCESS
NL7412254A (en) METHOD FOR PREPARING AN ORAL PREPARATION AGAINST DIABETES.
NL174945C (en) METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION WITH NEUROMUSCULAR BLOCKING ACTION, FORMED PHARMACEUTICAL PREPARATION AND METHOD FOR PREPARING A COMPOUND SUITABLE FOR THIS USE
NL159378B (en) PROCESS FOR PREPARING 2-AMINOALKYL-6-METHYL-7-NITRO-1,2,3,4-TETRAHYDROCHINOLINS, METHOD FOR PREPARING A PHARMACEUTICAL PREPARATION AND FORMED PHARMACEUTICAL PREPARATION.
NL7409947A (en) METHOD FOR PREPARING A MICROBIOLOGICAL RANDOM.
NL169872C (en) METHOD FOR PREPARING A MICROBICIDE PREPARATION AND METHOD FOR PREPARING SUITABLE COMPOUNDS

Legal Events

Date Code Title Description
V4 Discontinued because of reaching the maximum lifetime of a patent