NL171585B - METHOD FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS WITH ACTION ON THE CENTRAL NERVOUS SYSTEM BASED ON 6-PHENYL-1-OXOIMIDAZO-Ÿ1,2-AŸBENZOŸPHŸ-1,4-DIAZEPINES AND METHOD FOR THE PREPARATION OF THESE COMPOUNDS. - Google Patents

METHOD FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS WITH ACTION ON THE CENTRAL NERVOUS SYSTEM BASED ON 6-PHENYL-1-OXOIMIDAZO-Ÿ1,2-AŸBENZOŸPHŸ-1,4-DIAZEPINES AND METHOD FOR THE PREPARATION OF THESE COMPOUNDS.

Info

Publication number
NL171585B
NL171585B NLAANVRAGE7601492,A NL7601492A NL171585B NL 171585 B NL171585 B NL 171585B NL 7601492 A NL7601492 A NL 7601492A NL 171585 B NL171585 B NL 171585B
Authority
NL
Netherlands
Prior art keywords
preparation
aÿbenzoÿphÿ
oxoimidazo
diazepines
phenyl
Prior art date
Application number
NLAANVRAGE7601492,A
Other languages
Dutch (nl)
Other versions
NL7601492A (en
NL171585C (en
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB6509/75A external-priority patent/GB1496426A/en
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of NL7601492A publication Critical patent/NL7601492A/en
Publication of NL171585B publication Critical patent/NL171585B/en
Application granted granted Critical
Publication of NL171585C publication Critical patent/NL171585C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65583Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NLAANVRAGE7601492,A 1975-02-15 1976-02-13 METHOD FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS WITH ACTION ON THE CENTRAL NERVOUS SYSTEM BASED ON 6-PHENYL-1-OXOIMIDAZO-Ÿ1,2-AŸBENZOŸPHŸ-1,4-DIAZEPINES AND METHOD FOR THE PREPARATION OF THESE COMPOUNDS. NL171585C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB6509/75A GB1496426A (en) 1975-02-15 1975-02-15 1,2-dihydro-4h-imidazo(1,2-alpha)(1,4)benzodiazepin-1-ones processes for their preparation and compositions incorporating them
GB4580075 1975-11-04

Publications (3)

Publication Number Publication Date
NL7601492A NL7601492A (en) 1976-08-17
NL171585B true NL171585B (en) 1982-11-16
NL171585C NL171585C (en) 1983-04-18

Family

ID=26240753

Family Applications (1)

Application Number Title Priority Date Filing Date
NLAANVRAGE7601492,A NL171585C (en) 1975-02-15 1976-02-13 METHOD FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS WITH ACTION ON THE CENTRAL NERVOUS SYSTEM BASED ON 6-PHENYL-1-OXOIMIDAZO-Ÿ1,2-AŸBENZOŸPHŸ-1,4-DIAZEPINES AND METHOD FOR THE PREPARATION OF THESE COMPOUNDS.

Country Status (26)

Country Link
JP (1) JPS5914034B2 (en)
AR (1) AR225721A1 (en)
AT (1) AT351030B (en)
CA (1) CA1073454A (en)
CH (2) CH613706A5 (en)
DE (1) DE2605652A1 (en)
DK (1) DK141250B (en)
EG (1) EG12462A (en)
ES (1) ES445188A1 (en)
FI (1) FI62090C (en)
FR (1) FR2300569A1 (en)
GR (1) GR60028B (en)
HK (1) HK47379A (en)
HU (1) HU173109B (en)
IE (1) IE43791B1 (en)
IL (1) IL48888A (en)
IT (1) IT8047823A0 (en)
LU (1) LU74341A1 (en)
MX (1) MX3327E (en)
NL (1) NL171585C (en)
NO (1) NO146201C (en)
NZ (1) NZ179990A (en)
PH (3) PH14669A (en)
PT (1) PT64796B (en)
SE (1) SE422686B (en)
YU (1) YU42471B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2479818A1 (en) * 1980-04-03 1981-10-09 Roussel Uclaf 2-Substd. phenyl 7-nitro 3H 1,4-benzodiazepinyl aminoacid derivs. - are anxiolytics, tranquillisers, sedatives and anticonvulsants, prepd. by reacting aminoacid or peptide with benzodiazepin-2-thione
FR2502621B1 (en) * 1981-03-27 1983-10-28 Roussel Uclaf

Also Published As

Publication number Publication date
IL48888A0 (en) 1976-03-31
FR2300569B1 (en) 1979-09-21
CA1073454A (en) 1980-03-11
NO146201B (en) 1982-05-10
JPS5914034B2 (en) 1984-04-02
PH15282A (en) 1982-11-02
AR225721A1 (en) 1982-04-30
AT351030B (en) 1979-07-10
YU42471B (en) 1988-10-31
IT8047823A0 (en) 1980-02-06
SE7601592L (en) 1976-08-16
FI760347A (en) 1976-08-16
NL7601492A (en) 1976-08-17
PT64796B (en) 1978-02-06
SE422686B (en) 1982-03-22
LU74341A1 (en) 1976-12-31
ES445188A1 (en) 1977-09-16
NO760468L (en) 1976-08-17
FI62090B (en) 1982-07-30
DE2605652C2 (en) 1987-08-20
IE43791B1 (en) 1981-06-03
FI62090C (en) 1982-11-10
EG12462A (en) 1979-06-30
CH618171A5 (en) 1980-07-15
HU173109B (en) 1979-02-28
CH613706A5 (en) 1979-10-15
FR2300569A1 (en) 1976-09-10
PT64796A (en) 1976-03-01
IE43791L (en) 1976-08-15
JPS51105098A (en) 1976-09-17
DE2605652A1 (en) 1976-09-02
GR60028B (en) 1978-03-31
MX3327E (en) 1980-09-29
PH14669A (en) 1981-10-30
PH16286A (en) 1983-09-02
HK47379A (en) 1979-07-20
NZ179990A (en) 1978-06-02
IL48888A (en) 1979-03-12
DK141250C (en) 1980-08-04
NO146201C (en) 1982-08-18
AU1113776A (en) 1977-08-25
NL171585C (en) 1983-04-18
DK58776A (en) 1976-08-16
DK141250B (en) 1980-02-11
ATA107376A (en) 1978-12-15
YU34576A (en) 1984-12-31

Similar Documents

Publication Publication Date Title
NL7701584A (en) PROCEDURE FOR PREPARING MEDICINAL PRODUCTS WITH ANTIHYPERTENSIVE ACTION.
NL181628C (en) PROCESS FOR PREPARING PHARMACEUTICAL PREPARATIONS WITH PROSTAGLANDINE-LIKE ACTION, AND METHOD FOR PREPARING 9-ALFA, 11-ALFA, 15-ALFA-TRIHYDROXY-PROSTA-4,5,13-TRI-ACID DERIVATIVES, PREVIOUSLY USED
NL7706532A (en) PROCESS FOR PREPARING ESTERS WITH ANTI-BACTERIAL ACTION, AND PHARMACEUTICAL PREPARATIONS CONTAINING ESTERS.
NL7905375A (en) PROSTANOIDS, METHOD FOR PREPARING THE SAME AND PHARMACEUTICAL PREPARATIONS BASED ON THAT
NL7409344A (en) PROCEDURE FOR PREPARING ALKOXYALKYL 1,4-DIHYDROPYRIDINS AND THEIR USE AS PHARMACEUTICAL PREPARATIONS.
NL7705881A (en) PYRIDINE COMPOUNDS, METHOD FOR PREPARING SUCH PYRIDINE COMPOUNDS, PROCESS FOR PREPARING PHARMACEUTICAL PREPARATIONS WITH SUCH PYRIDINE COMPOUNDS AND THE PREPARATIONS FORMED.
NL7601085A (en) PROCEDURE FOR PREPARING OXADIAZOLINONE COMPOUNDS, PROCEDURE FOR PREPARING PREPARATIONS WITH AN INSECTICIDE, ACARICIDE AND NEMATOCIDE ACTION, AND THE PREPARATIONS FORMED.
NL192206B (en) Process for the preparation of a 13β-alkyl-17O-ethynyl-17β-alkanoyloxy-gon-4-en-3-on-oxime compound, process for the preparation of pharmaceutical preparations with such a compound and the pharmaceutical preparations formed.
NL173523B (en) PROCESS FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS WITH ACTION ON THE CENTRAL NERVOUS SYSTEM BASED ON TRIAZOLOŸ4.3-AŸŸ1.4ZBENZODIAZEPINE DERIVATIVES, AND METHOD FOR THE PREPARATION OF TRIAZOLO.34Z-AEDIAZEDZAPZZAPZ.4Z-AZIAZZ.4.4
NL183718C (en) METHOD FOR PREPARING PHARMACEUTICAL PREPARATIONS WITH ACTIVITY ON THE ENZYME SYSTEM OF THE LIVER, METHOD FOR PREPARING COMPOUNDS SUITABLE FOR USE, AND PHARMACEUTICAL ARTICLES
NL7612937A (en) THIENAMYCINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS AND THE PROCESS FOR PREPARING THEM.
NL7415815A (en) PROCEDURE FOR PREPARING PYRIMIDINE-THIONOTHIOLPHOSPHORIC ESTERS, AND THEIR USE AS INSECTICIDES AND ACARICIDES.
NL7705883A (en) PYRIDINE COMPOUNDS, METHOD FOR PREPARING SUCH PYRIDINE COMPOUNDS, PROCESS FOR PREPARING PHARMACEUTICAL PREPARATIONS WITH SUCH PYRIDINE COMPOUNDS, AND THE PREPARATION THEREFORE OBTAINED.
NL167697C (en) PROCESS FOR THE PREPARATION OF A PHARMACEUTICAL PREPARATION ACTING ON THE CENTRAL NERVOUS SYSTEM BASED ON 5-PHENYLBENZODIAZEPINE DERIVATIVES, AND METHOD FOR PREPARING 5-PHENYLBODODIA ZEPARIC THESE BEFORE USE THEREFORE
NL7501914A (en) PROCESS FOR THE PREPARATION OF CEPHALOSSPORINS AND THEIR USE AS PHARMACEUTICAL PREPARATIONS.
NL174045B (en) PROCEDURE FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS WITH ACTION ON THE CENTRAL NERVOUS SYSTEM BASED ON 6H-THIENO-3,2-F-S-TRIAZOLO4,3-A 1,4DIAZEPINE DERIVATIVES, AND METHOD FOR PREPARING THESE DERIVATIVES.
NL177828C (en) METHODS FOR PREPARING MEDICINES WITH ANTI-INFLAMMATORY AND ANALGETIC EFFECTS AND N-PHENYL-PYROLIC COMPOUNDS SUITABLE FOR THAT.
NL7612941A (en) THIENAMYCINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS AND THE PROCESS FOR PREPARING THEM.
NL7602391A (en) METHODS FOR PREPARING AND USING L-3- (3,4-DIHYDROXY-PHENYL) -2-METHYL-ALANINE -PEPTIDES.
NL7612894A (en) PROCEDURE FOR THE PREPARATION OF HETEROCYCLIC COMPOUNDS ACTING ON THE CENTRAL NERVOUS SYSTEM, PROCESS FOR THE PREPARATION OF A MEDICINAL PRODUCT WITH SUCH ACTION AND MEDICINAL PRODUCT.
NL7701833A (en) PROCEDURE FOR PREPARING PYRROLOBEN ZOXAZALKANES, PHARMACEUTICAL PREPARATIONS CONTAINING THESE COMPOUNDS, AND TREATMENT WITH THESE PHARMACEUTICAL PREPARATIONS.
NL7610058A (en) METHOD FOR THE PREPARATION OF ANIMAL FEED PREPARATIONS.
NL7604882A (en) PROCEDURE FOR THE PREPARATION OF BICYCLOOCTA DERIVATIVES ACTING ON THE CENTRAL NERVOUS SYSTEM, PROCESS FOR THE PREPARATION OF A MEDICINAL PRODUCT WITH SUCH ACTION AND OF ANY MEDICINAL PRODUCT.
NL7608164A (en) PROCESS FOR PREPARING CEFEM AND PENAM COMPOUNDS, AS WELL AS PROCEDURE FOR PREPARING PHARMACEUTICAL PREPARATIONS.
NL171585C (en) METHOD FOR THE PREPARATION OF PHARMACEUTICAL PREPARATIONS WITH ACTION ON THE CENTRAL NERVOUS SYSTEM BASED ON 6-PHENYL-1-OXOIMIDAZO-Ÿ1,2-AŸBENZOŸPHŸ-1,4-DIAZEPINES AND METHOD FOR THE PREPARATION OF THESE COMPOUNDS.

Legal Events

Date Code Title Description
V4 Discontinued because of reaching the maximum lifetime of a patent

Free format text: 960213