MXPA06000988A - Derivados de nicotinamida utiles como inhibidores de pde4. - Google Patents
Derivados de nicotinamida utiles como inhibidores de pde4.Info
- Publication number
- MXPA06000988A MXPA06000988A MXPA06000988A MXPA06000988A MXPA06000988A MX PA06000988 A MXPA06000988 A MX PA06000988A MX PA06000988 A MXPA06000988 A MX PA06000988A MX PA06000988 A MXPA06000988 A MX PA06000988A MX PA06000988 A MXPA06000988 A MX PA06000988A
- Authority
- MX
- Mexico
- Prior art keywords
- inhibitors
- pdea4
- derivatives useful
- nicotinamide derivatives
- nicotinamide
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Immunology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Esta invencion se refiere a derivados de nicotinamida de formula general (I): (ver formula (I) en la que R1, R2 y R3 tienen los significados definidos en la presente memoria, y a procesos para la preparacion de intermedios utilizados en la preparacion de composiciones que los contienen, y a los usos de estos derivados.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0317509.8A GB0317509D0 (en) | 2003-07-25 | 2003-07-25 | Nicotinamide derivatives useful as PDE4 inhibitors |
PCT/IB2004/002365 WO2005010001A1 (en) | 2003-07-25 | 2004-07-13 | Nicotinamide derivatives useful as pdea4 inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
MXPA06000988A true MXPA06000988A (es) | 2006-04-11 |
Family
ID=27772736
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MXPA06000988A MXPA06000988A (es) | 2003-07-25 | 2004-07-13 | Derivados de nicotinamida utiles como inhibidores de pde4. |
Country Status (7)
Country | Link |
---|---|
EP (1) | EP1651647A1 (es) |
JP (1) | JP2006528623A (es) |
BR (1) | BRPI0412933A (es) |
CA (1) | CA2533681A1 (es) |
GB (1) | GB0317509D0 (es) |
MX (1) | MXPA06000988A (es) |
WO (1) | WO2005010001A1 (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR049384A1 (es) | 2004-05-24 | 2006-07-26 | Glaxo Group Ltd | Derivados de purina |
JP5846711B2 (ja) * | 2005-06-09 | 2016-01-20 | メダ アーベー | 炎症性疾患の治療のための方法及び組成物 |
GB0514809D0 (en) | 2005-07-19 | 2005-08-24 | Glaxo Group Ltd | Compounds |
WO2007019232A2 (en) * | 2005-08-03 | 2007-02-15 | Immunogen, Inc. | Immunoconjugate formulations |
CN102105448B (zh) * | 2008-05-27 | 2013-11-13 | 阿斯利康(瑞典)有限公司 | 苯氧基吡啶基酰胺衍生物和它们在治疗由pde4介导的病症中的用途 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR9810733A (pt) * | 1997-04-04 | 2000-09-12 | Pfizer Prod Inc | Derivados de nicotinamida |
GEP20074055B (en) * | 2002-02-11 | 2007-03-12 | Pfizer | Nicotinamide derivatives useful as pde4 inhibitors |
GB0203193D0 (en) * | 2002-02-11 | 2002-03-27 | Pfizer Ltd | Nicotinamide derivatives useful as pde4 inhibitors |
-
2003
- 2003-07-25 GB GBGB0317509.8A patent/GB0317509D0/en not_active Ceased
-
2004
- 2004-07-13 MX MXPA06000988A patent/MXPA06000988A/es not_active Application Discontinuation
- 2004-07-13 BR BRPI0412933-4A patent/BRPI0412933A/pt not_active Application Discontinuation
- 2004-07-13 WO PCT/IB2004/002365 patent/WO2005010001A1/en not_active Application Discontinuation
- 2004-07-13 JP JP2006520932A patent/JP2006528623A/ja active Pending
- 2004-07-13 EP EP04744024A patent/EP1651647A1/en not_active Withdrawn
- 2004-07-13 CA CA002533681A patent/CA2533681A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CA2533681A1 (en) | 2005-02-03 |
JP2006528623A (ja) | 2006-12-21 |
WO2005010001A1 (en) | 2005-02-03 |
GB0317509D0 (en) | 2003-08-27 |
BRPI0412933A (pt) | 2006-09-26 |
EP1651647A1 (en) | 2006-05-03 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal |