MXPA05011775A - Sulfonamidas y pirazolamidas como moduladores de canal de sodio. - Google Patents
Sulfonamidas y pirazolamidas como moduladores de canal de sodio.Info
- Publication number
- MXPA05011775A MXPA05011775A MXPA05011775A MXPA05011775A MXPA05011775A MX PA05011775 A MXPA05011775 A MX PA05011775A MX PA05011775 A MXPA05011775 A MX PA05011775A MX PA05011775 A MXPA05011775 A MX PA05011775A MX PA05011775 A MXPA05011775 A MX PA05011775A
- Authority
- MX
- Mexico
- Prior art keywords
- formula
- sulfonamides
- pyrazole
- amides
- sodium channel
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US10/427,847 US20040220170A1 (en) | 2003-05-01 | 2003-05-01 | Pyrazole-amides and sulfonamides as sodium channel modulators |
PCT/US2004/013530 WO2004099154A2 (fr) | 2003-05-01 | 2004-04-29 | Pyrazole-amides et sulfonamides modulateurs des canaux sodiques |
Publications (1)
Publication Number | Publication Date |
---|---|
MXPA05011775A true MXPA05011775A (es) | 2006-02-17 |
Family
ID=35529848
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MXPA05011775A MXPA05011775A (es) | 2003-05-01 | 2004-04-29 | Sulfonamidas y pirazolamidas como moduladores de canal de sodio. |
Country Status (4)
Country | Link |
---|---|
EP (1) | EP1620405A2 (fr) |
JP (1) | JP2006525355A (fr) |
CA (1) | CA2525325A1 (fr) |
MX (1) | MXPA05011775A (fr) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7638541B2 (en) | 2006-12-28 | 2009-12-29 | Metabolex Inc. | 5-ethyl-2-{4-[4-(4-tetrazol-1-yl-phenoxymethyl)-thiazol-2-yl]-piperidin-1-yl}-pyrimidine |
US8183381B2 (en) * | 2007-07-19 | 2012-05-22 | Metabolex Inc. | N-linked heterocyclic receptor agonists for the treatment of diabetes and metabolic disorders |
US8410127B2 (en) | 2009-10-01 | 2013-04-02 | Metabolex, Inc. | Substituted tetrazol-1-yl-phenoxymethyl-thiazol-2-yl-piperidinyl-pyrimidine salts |
WO2012177263A1 (fr) * | 2011-06-24 | 2012-12-27 | Intra-Cellular Therapies, Inc. | Composés et procédés de prophylaxie et de traitement concernant des antagonistes de récepteur nicotinique |
HUE040489T2 (hu) * | 2014-06-03 | 2019-03-28 | Idorsia Pharmaceuticals Ltd | Pirazolvegyületek és alkalmazásuk t-típusú kalciumcsatorna-blokkolókként |
JP2019504840A (ja) * | 2016-01-28 | 2019-02-21 | ソルヴェイ(ソシエテ アノニム) | ハロゲン置換ジケトン、ピラゾール化合物およびピラゾール化合物の製造方法 |
US10292983B2 (en) | 2016-08-03 | 2019-05-21 | Cymabay Therapeutics, Inc. | Oxymethylene aryl compounds for treating inflammatory gastrointestinal diseases or gastrointestinal conditions |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE443698T1 (de) * | 1996-12-23 | 2009-10-15 | Bristol Myers Squibb Pharma Co | Stickstoffhaltige heterocyclen als faktor xa- hemmer |
BR9810151A (pt) * | 1997-06-19 | 2000-08-08 | Du Pont Pharm Co | Composto, composição farmacêutica e método para tratamento ou prevenção de uma desordem tromoboembólica |
IL136637A0 (en) * | 1997-12-22 | 2001-06-14 | Du Pont Pharm Co | Nitrogen containing heteroaromatics with ortho-substituted pi's as factor xa inhibitors |
CA2373510A1 (fr) * | 1999-05-12 | 2000-11-23 | Ortho-Mcneil Pharmaceutical, Inc. | Carboxamides de pyrazole utiles pour le traitement de l'obesite et d'autres troubles |
IL148698A0 (en) * | 1999-09-17 | 2002-09-12 | Cor Therapeutics Inc | INHIBITORS OF FACTOR Xa |
CA2409827C (fr) * | 2000-05-22 | 2010-06-01 | Aventis Pharmaceuticals Products Inc. | Derives d'arylmethylamine utilises comme inhibiteurs de la tryptase |
US6604974B2 (en) * | 2000-12-22 | 2003-08-12 | Thomson Licensing S.A. | Method and apparatus for applying crosswires to a tension focus mask |
MXPA04012959A (es) * | 2002-06-29 | 2005-05-16 | Zentaris Gmbh | Arilcarbonilpiperacinas y heteroarilcarbonilpiperacinas y su uso para tratamiento de enfermedades de tumor benigno y maligno. |
GB0226178D0 (en) * | 2002-11-11 | 2002-12-18 | Johnson Matthey Plc | Desulphurisation |
AU2004218260A1 (en) * | 2003-01-28 | 2004-09-16 | Aventis Pharma S.A. | N-aryl heteroaromatic products, compositions containing same and use thereof |
-
2004
- 2004-04-29 MX MXPA05011775A patent/MXPA05011775A/es not_active Application Discontinuation
- 2004-04-29 CA CA002525325A patent/CA2525325A1/fr not_active Abandoned
- 2004-04-29 EP EP04751090A patent/EP1620405A2/fr not_active Withdrawn
- 2004-04-29 JP JP2006514200A patent/JP2006525355A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
EP1620405A2 (fr) | 2006-02-01 |
JP2006525355A (ja) | 2006-11-09 |
CA2525325A1 (fr) | 2004-11-18 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal |