MXPA04002445A - Analogos de wortmanina y metodos para utilizar los mismos. - Google Patents
Analogos de wortmanina y metodos para utilizar los mismos.Info
- Publication number
- MXPA04002445A MXPA04002445A MXPA04002445A MXPA04002445A MXPA04002445A MX PA04002445 A MXPA04002445 A MX PA04002445A MX PA04002445 A MXPA04002445 A MX PA04002445A MX PA04002445 A MXPA04002445 A MX PA04002445A MX PA04002445 A MXPA04002445 A MX PA04002445A
- Authority
- MX
- Mexico
- Prior art keywords
- compound
- effective amount
- wortmanin
- administering
- chemical formula
- Prior art date
Links
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/94—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Distillation Of Fermentation Liquor, Processing Of Alcohols, Vinegar And Beer (AREA)
- Compounds Of Unknown Constitution (AREA)
- Pyrane Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US32214301P | 2001-09-14 | 2001-09-14 | |
| US32213901P | 2001-09-14 | 2001-09-14 | |
| PCT/US2002/029365 WO2003024183A2 (en) | 2001-09-14 | 2002-09-16 | Wortmannin analogs and methods of using same |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA04002445A true MXPA04002445A (es) | 2005-07-25 |
Family
ID=26983283
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA04002445A MXPA04002445A (es) | 2001-09-14 | 2002-09-16 | Analogos de wortmanina y metodos para utilizar los mismos. |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP1435941B8 (https=) |
| JP (1) | JP4540986B2 (https=) |
| AT (1) | ATE334671T1 (https=) |
| AU (1) | AU2002330029B2 (https=) |
| CA (1) | CA2458318C (https=) |
| DE (1) | DE60213633T2 (https=) |
| MX (1) | MXPA04002445A (https=) |
| WO (1) | WO2003024183A2 (https=) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7081475B2 (en) * | 2001-09-14 | 2006-07-25 | Prolx Pharmaceuticals Corp. | Wortmannin analogs and methods of using same |
| DE10219545A1 (de) * | 2002-04-26 | 2003-11-06 | Lang Florian | Regulation der Apoptose |
| US7230139B2 (en) | 2002-12-05 | 2007-06-12 | Gemin X Biotechnologies | Diterpenoid compounds, compositions thereof and their use as anti-cancer or anti-fungal agents |
| MXPA05011248A (es) * | 2003-04-23 | 2005-12-14 | Wyeth Corp | Derivados de wortmanina solubles en agua. |
| DE102004043463A1 (de) * | 2004-06-09 | 2006-02-09 | Heinz Voigt | Mittel zur Krebsbekämpfung unter Verwendung von Schimmelpilzextrakten |
| JP5371426B2 (ja) * | 2004-07-09 | 2013-12-18 | プロルックス ファーマシューティカルズ コープ． | ワートマニン類似体及び化学療法薬と組み合わせた同一物を使用する方法 |
| EP1799699A1 (en) | 2004-10-13 | 2007-06-27 | Wyeth | Analogs of 17-hydroxywortmannin as pi3k inhibitors |
| WO2006132675A2 (en) * | 2004-12-20 | 2006-12-14 | University Of South Florida | Xiap-targeted prostate cancer therapy |
| EP1940386A4 (en) * | 2005-09-01 | 2010-06-23 | Beth Israel Hospital | WORDMAN'S CONJUGATES AND USES THEREOF |
| US20070116736A1 (en) * | 2005-11-23 | 2007-05-24 | Argentieri Dennis C | Local vascular delivery of PI3 kinase inhibitors alone or in combination with sirolimus to prevent restinosis following vascular injury |
| EP1965790B1 (en) * | 2005-12-30 | 2011-12-07 | Arizona Board of Regents, Acting on Behalf of The University of Arizona | Metabolites of wortmannin analogs and methods of using the same |
| EP2012794B1 (en) * | 2006-04-13 | 2014-09-17 | The Trustees of Columbia University in the City of New York | Compositions and intraluminal devices for inhibiting vascular stenosis |
| EP2576535A4 (en) * | 2010-06-04 | 2014-03-12 | Oncothyreon Inc | COMBINED CANCER THERAPIES WITH WORDMAN ANALOG |
| CA2801448A1 (en) * | 2010-06-04 | 2011-12-08 | Oncothyreon Inc. | Cancer treatment with wortmannin analogs |
| US11197854B1 (en) | 2018-11-14 | 2021-12-14 | National Technology & Engineering Solutions Of Sandia, Llc | Inhibitors for targeting flaviviruses |
| US20220040324A1 (en) | 2018-12-21 | 2022-02-10 | Daiichi Sankyo Company, Limited | Combination of antibody-drug conjugate and kinase inhibitor |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2302021A (en) * | 1996-10-16 | 1997-01-08 | Lilly Co Eli | Inhibiting bone loss or resorption |
-
2002
- 2002-09-16 MX MXPA04002445A patent/MXPA04002445A/es active IP Right Grant
- 2002-09-16 EP EP02766286A patent/EP1435941B8/en not_active Expired - Lifetime
- 2002-09-16 DE DE60213633T patent/DE60213633T2/de not_active Expired - Lifetime
- 2002-09-16 AU AU2002330029A patent/AU2002330029B2/en not_active Ceased
- 2002-09-16 CA CA2458318A patent/CA2458318C/en not_active Expired - Fee Related
- 2002-09-16 WO PCT/US2002/029365 patent/WO2003024183A2/en not_active Ceased
- 2002-09-16 JP JP2003528088A patent/JP4540986B2/ja not_active Expired - Fee Related
- 2002-09-16 AT AT02766286T patent/ATE334671T1/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| AU2002330029B2 (en) | 2006-07-06 |
| EP1435941A4 (en) | 2004-12-08 |
| DE60213633T2 (de) | 2007-11-08 |
| WO2003024183A2 (en) | 2003-03-27 |
| CA2458318A1 (en) | 2003-03-27 |
| EP1435941B8 (en) | 2006-10-25 |
| WO2003024183A3 (en) | 2003-06-12 |
| CA2458318C (en) | 2011-03-15 |
| JP2005507880A (ja) | 2005-03-24 |
| EP1435941A2 (en) | 2004-07-14 |
| EP1435941B1 (en) | 2006-08-02 |
| DE60213633D1 (de) | 2006-09-14 |
| ATE334671T1 (de) | 2006-08-15 |
| JP4540986B2 (ja) | 2010-09-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant or registration |