MX9707073A - Preparaciones de aerosol de prilocaina e hidrofluorocarbono. - Google Patents

Preparaciones de aerosol de prilocaina e hidrofluorocarbono.

Info

Publication number
MX9707073A
MX9707073A MX9707073A MX9707073A MX9707073A MX 9707073 A MX9707073 A MX 9707073A MX 9707073 A MX9707073 A MX 9707073A MX 9707073 A MX9707073 A MX 9707073A MX 9707073 A MX9707073 A MX 9707073A
Authority
MX
Mexico
Prior art keywords
hydrofluorocarbon
prilocaine
aerosol preparations
prilocaine base
liquid
Prior art date
Application number
MX9707073A
Other languages
English (en)
Other versions
MXPA97007073A (es
Inventor
Richard A Henry
Original Assignee
Richard A Henry
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27410659&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX9707073(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US08/405,930 external-priority patent/US5593661A/en
Priority claimed from US08/408,877 external-priority patent/US5534242A/en
Application filed by Richard A Henry filed Critical Richard A Henry
Publication of MX9707073A publication Critical patent/MX9707073A/es
Publication of MXPA97007073A publication Critical patent/MXPA97007073A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/235Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
    • A61K31/24Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group having an amino or nitro group
    • A61K31/245Amino benzoic acid types, e.g. procaine, novocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/008Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy comprising drug dissolved or suspended in liquid propellant for inhalation via a pressurized metered dose inhaler [MDI]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/12Aerosols; Foams
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/12Aerosols; Foams
    • A61K9/124Aerosols; Foams characterised by the propellant
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics
    • A61P23/02Local anaesthetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

Una base de prilocaína, en forma líquida y de cristal de microbarras, se puede solubilizar dentro de propulsores de hidrofluorocarbono para producir un líquido oleoso estable; la base de prilocaína se puede usar para solubilizar medicamentos adicionales dentro de propulsores de hidrofluorocarbono que no son ordinariamente solubles; la combinacion de base de prilocaína y propulsor de hidrofluorocarbono se puede usar como una aspersion aerosolizada para proveer anestesia topica.
MXPA/A/1997/007073A 1995-03-17 1997-09-17 Preparaciones de aerosol de prilocaina e hidrofluorocarbono MXPA97007073A (es)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US08405930 1995-03-17
US08/405,930 US5593661A (en) 1993-03-29 1995-03-17 Lidocaine aerosol anaesthetic
US08/408,877 US5534242A (en) 1994-05-02 1995-03-24 Lidocaine-vasoconstrictor aerosol preparation
US08408877 1995-03-24
US08/435,812 US5589156A (en) 1994-05-02 1995-05-05 Prilocaine and hydrofluourocarbon aerosol preparations
US08435812 1995-05-05

Publications (2)

Publication Number Publication Date
MX9707073A true MX9707073A (es) 1998-08-30
MXPA97007073A MXPA97007073A (es) 1998-11-12

Family

ID=

Also Published As

Publication number Publication date
ES2203676T3 (es) 2004-04-16
PT814793E (pt) 2003-12-31
US5589156A (en) 1996-12-31
AU710600B2 (en) 1999-09-23
DE69629109D1 (de) 2003-08-21
WO1996029066A1 (en) 1996-09-26
LU92402I2 (fr) 2014-05-19
CN1149080C (zh) 2004-05-12
CN1179103A (zh) 1998-04-15
JP4117707B2 (ja) 2008-07-16
BR9607988A (pt) 1999-11-30
EP0814793A1 (en) 1998-01-07
EP0814793B1 (en) 2003-07-16
DK0814793T3 (da) 2003-12-01
ATE245025T1 (de) 2003-08-15
AU4711396A (en) 1996-10-08
JPH11502202A (ja) 1999-02-23
DE69629109T2 (de) 2004-04-15

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