MX9704667A - 6-[triazolil[3-trifluorometil)fenil]metil]-2-quinolinonas y quinolinotionas. - Google Patents
6-[triazolil[3-trifluorometil)fenil]metil]-2-quinolinonas y quinolinotionas.Info
- Publication number
- MX9704667A MX9704667A MX9704667A MX9704667A MX9704667A MX 9704667 A MX9704667 A MX 9704667A MX 9704667 A MX9704667 A MX 9704667A MX 9704667 A MX9704667 A MX 9704667A MX 9704667 A MX9704667 A MX 9704667A
- Authority
- MX
- Mexico
- Prior art keywords
- 4alkyl
- hydrogen
- quinolinethiones
- quinolinones
- triazolyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/12—Keratolytics, e.g. wart or anti-corn preparations
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Esta invencion se refiere a compuestos de formula (I), las sales ácidas de adicion farmacéuticamente aceptables y las formas estereoquímicamente isoméricas de los mismos, en donde R1 es hidrogeno, amino o alquilo C1-4; R2 es hidrogeno, halogeno o alquilo C1-4; R3 es hidrogeno, halogeno o alquilo C1-4; Y es O o S y -X1=X2- es un radical bivalente que tiene la formula: -N=CH- (a-1) o -CH=N- (a-2); composiciones que contienen los mismos y procedimientos para preparar estos compuestos; se refiere además a su uso como medicina, en particular su uso como medicina para tratar desordenes de queratinizacion.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP94203773 | 1994-12-28 | ||
EP94203773.0 | 1994-12-28 | ||
PCT/EP1995/005173 WO1996020200A1 (en) | 1994-12-28 | 1995-12-21 | 6-[triazolyl[3-(trifluoromethyl)phenyl]methyl]-2-quinolinones and -quinolinethiones |
Publications (2)
Publication Number | Publication Date |
---|---|
MX9704667A true MX9704667A (es) | 1997-09-30 |
MXPA97004667A MXPA97004667A (es) | 1998-07-03 |
Family
ID=
Also Published As
Publication number | Publication date |
---|---|
ATE207924T1 (de) | 2001-11-15 |
US5922734A (en) | 1999-07-13 |
AU698199B2 (en) | 1998-10-29 |
NZ298789A (en) | 1999-07-29 |
WO1996020200A1 (en) | 1996-07-04 |
CA2207268A1 (en) | 1996-07-04 |
DE69523629T2 (de) | 2002-07-18 |
IL116577A (en) | 2000-02-29 |
EP0800524B1 (en) | 2001-10-31 |
PL182956B1 (pl) | 2002-05-31 |
CN1171789A (zh) | 1998-01-28 |
AU4436296A (en) | 1996-07-19 |
DE69523629D1 (de) | 2001-12-06 |
ZA9510989B (en) | 1997-06-27 |
JPH10511654A (ja) | 1998-11-10 |
PL321041A1 (en) | 1997-11-24 |
TR199501688A2 (tr) | 1996-07-21 |
FI972794A0 (fi) | 1997-06-27 |
TW316902B (es) | 1997-10-01 |
MY131690A (en) | 2007-08-30 |
PT800524E (pt) | 2002-04-29 |
CN1085668C (zh) | 2002-05-29 |
HRP950616A2 (en) | 1997-10-31 |
EP0800524A1 (en) | 1997-10-15 |
IL116577A0 (en) | 1996-03-31 |
NO311220B1 (no) | 2001-10-29 |
RU2165419C2 (ru) | 2001-04-20 |
FI972794A (fi) | 1997-06-27 |
AR002264A1 (es) | 1998-03-11 |
NO973029D0 (no) | 1997-06-27 |
BR9510504A (pt) | 1999-06-01 |
DK0800524T3 (da) | 2002-03-25 |
NO973029L (no) | 1997-06-27 |
ES2166838T3 (es) | 2002-05-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Grant or registration | ||
MM | Annulment or lapse due to non-payment of fees |