MX9304931A - Anticonceptivos que contienen antiprogestogenos. - Google Patents

Anticonceptivos que contienen antiprogestogenos.

Info

Publication number
MX9304931A
MX9304931A MX9304931A MX9304931A MX9304931A MX 9304931 A MX9304931 A MX 9304931A MX 9304931 A MX9304931 A MX 9304931A MX 9304931 A MX9304931 A MX 9304931A MX 9304931 A MX9304931 A MX 9304931A
Authority
MX
Mexico
Prior art keywords
phase
regimen
sequential
daily
contraceptive
Prior art date
Application number
MX9304931A
Other languages
English (en)
Inventor
Engelbert Willem Bergink
Original Assignee
Akzo Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nv filed Critical Akzo Nv
Publication of MX9304931A publication Critical patent/MX9304931A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se describen regímenes de anticonceptivos orales efectivos que contienen una fase antiprogestógenos combinada con una fase de progestógenos. Un régimen de anticonceptivos que tiene: una primera fase de 5-20, en especial 14, unidades de dosis secuenciales diarias que contienen un antiprogestógeno a una dosis diaria suficiente para inhibir la ovulación en la mujer, y una segunda fase de 10 a 25, especialmente 14, unidades de dosis diarias secuenciales que contienen un progestógenos a una dosis equivalente a 40-120 µg de desogestrel administrado oralmente. A la primera fase preferencialmente se añade un estrógeno como el 17ß-estradio (de 0.50 a 2.5mg diariamente) para permitir la posibilidad de hacer régimen secuencial. La presente invención también incluye un producto anticonceptivo (es decir, el paquete que contiene el régimen de dosis unitaria), y un proceso para fabricar este producto.
MX9304931A 1992-08-14 1993-08-13 Anticonceptivos que contienen antiprogestogenos. MX9304931A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP92202504 1992-08-14

Publications (1)

Publication Number Publication Date
MX9304931A true MX9304931A (es) 1994-08-31

Family

ID=8210854

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9304931A MX9304931A (es) 1992-08-14 1993-08-13 Anticonceptivos que contienen antiprogestogenos.

Country Status (4)

Country Link
AU (1) AU4708993A (es)
MX (1) MX9304931A (es)
WO (1) WO1994004156A1 (es)
ZA (1) ZA935617B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1993021926A1 (en) * 1992-05-06 1993-11-11 Medical College Of Hampton Roads Minimizing progestin associated breakthrough bleeding
US5521166A (en) * 1994-12-19 1996-05-28 Ortho Pharmaceitical Corporation Antiprogestin cyclophasic hormonal regimen
US6506390B2 (en) 1996-06-25 2003-01-14 Akzo Nobel Progestogen-anti-progestogen regimens
WO1997049407A1 (en) * 1996-06-25 1997-12-31 Akzo Nobel N.V. Progestogen-anti-progestogen regimens
KR20010032056A (ko) * 1997-11-14 2001-04-16 에프.지.엠. 헤르만스 ; 이.에이치. 리링크 황체 호르몬-항 황체 호르몬 투약법
DE69934113T2 (de) * 1998-05-22 2007-06-06 Abbott Laboratories, Abbott Park Antiangiogene substanz zur behandlung von krebs, arthritis und netzhauterkrankungen
US6632961B1 (en) 1998-05-22 2003-10-14 Abbott Laboratories Antiangiogenic drug to treat cancer, arthritis and retinopathy
DE60014358D1 (de) * 1999-04-29 2004-11-04 Akzo Nobel Nv Verwendung von org 33245 in der kombinierten intermittierenden hormontherapie und empfängnisverhütung

Also Published As

Publication number Publication date
ZA935617B (en) 1994-03-07
AU4708993A (en) 1994-03-15
WO1994004156A1 (en) 1994-03-03

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