MX9203205A - NOVELTY DIMETILAMINO-HIDROXI-ALCAN-DIPHOSPHONIC ACIDS AND SALTS OF THE SAME, IN PRODUCTION PROCEDURE AND RELATED PHARMACEUTICAL COMPOSITIONS. - Google Patents

NOVELTY DIMETILAMINO-HIDROXI-ALCAN-DIPHOSPHONIC ACIDS AND SALTS OF THE SAME, IN PRODUCTION PROCEDURE AND RELATED PHARMACEUTICAL COMPOSITIONS.

Info

Publication number
MX9203205A
MX9203205A MX9203205A MX9203205A MX9203205A MX 9203205 A MX9203205 A MX 9203205A MX 9203205 A MX9203205 A MX 9203205A MX 9203205 A MX9203205 A MX 9203205A MX 9203205 A MX9203205 A MX 9203205A
Authority
MX
Mexico
Prior art keywords
dimetilamino
hidroxi
alcan
novelty
salts
Prior art date
Application number
MX9203205A
Other languages
Spanish (es)
Inventor
Guainai Ricci Giuseppe
Rosini Sergio
Mian Maurizio
Original Assignee
Gentili Ist Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gentili Ist Spa filed Critical Gentili Ist Spa
Publication of MX9203205A publication Critical patent/MX9203205A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic System
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids, i.e. RP(=X)(XH)2 (X = S, Se)
    • C07F9/3804Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids, i.e. RP(=X)(XH)2 (X = S, Se) not used, see subgroups
    • C07F9/3839Polyphosphonic acids
    • C07F9/3873Polyphosphonic acids containing nitrogen substituent, e.g. N.....H or N-hydrocarbon group which can be substituted by halogen or nitro(so), N.....O, N.....S, N.....C(=X)- (X =O, S), N.....N, N...C(=X)...N (X =O, S)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

Acidos dimetilamino -1- hidroxi- alcan - 1,1, - difosfónicos de la fórmula (I), en donde n 4 ó 5 y un procedimiento para su producción, así como su uso para el tratamiento de enfermedades asociadas con trasntornos del metabolismo óseo.Dimethylamino -1-hydroxy-alkan-1,1,-diphosphonic acids of formula (I), where n 4 or 5 and a procedure for its production, as well as its use for the treatment of diseases associated with disorders of bone metabolism .

MX9203205A 1991-06-26 1992-06-24 NOVELTY DIMETILAMINO-HIDROXI-ALCAN-DIPHOSPHONIC ACIDS AND SALTS OF THE SAME, IN PRODUCTION PROCEDURE AND RELATED PHARMACEUTICAL COMPOSITIONS. MX9203205A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITFI910160A IT1247034B (en) 1991-06-26 1991-06-26 DIMETHYLAMINE-HYDROXY ACIDS DIPHOSPHONICS AND THEIR SALTS, THEIR PRODUCTION PROCESS AND PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEM

Publications (1)

Publication Number Publication Date
MX9203205A true MX9203205A (en) 1994-06-30

Family

ID=11349724

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9203205A MX9203205A (en) 1991-06-26 1992-06-24 NOVELTY DIMETILAMINO-HIDROXI-ALCAN-DIPHOSPHONIC ACIDS AND SALTS OF THE SAME, IN PRODUCTION PROCEDURE AND RELATED PHARMACEUTICAL COMPOSITIONS.

Country Status (8)

Country Link
EP (1) EP0592488A1 (en)
JP (1) JPH06508833A (en)
AU (1) AU2150792A (en)
CA (1) CA2112250A1 (en)
IT (1) IT1247034B (en)
MX (1) MX9203205A (en)
PT (1) PT100624B (en)
WO (1) WO1993000348A1 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1303672B1 (en) 1998-07-28 2001-02-23 Nicox Sa NITRATED SALTS OF DRUGS ACTIVE IN BONE DISORDERS
DE60235085D1 (en) * 2001-07-16 2010-03-04 Univ Paris Xiii PREPARATION OF DERIVATIVES OF BISPHOSPHONATES
DE102014115154A1 (en) * 2014-10-17 2016-04-21 SCV-SpezialChemikalien-Vertrieb GmbH Conjugated bisphosphonates for the diagnosis and treatment of bone diseases

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1194748B (en) * 1981-02-12 1988-09-28 Gentili Ist Spa PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF OSTEOPATHIES
IT1201087B (en) * 1982-04-15 1989-01-27 Gentili Ist Spa PHARMACOLOGICALLY ACTIVE BIPPHOSPHONES, PROCEDURE FOR THEIR PREPARATION AND RELATED PHARMACEUTICAL COMPOSITIONS
DE3434667A1 (en) * 1984-09-21 1986-04-03 Henkel KGaA, 4000 Düsseldorf 4-DIMETHYLAMINO-1-HYDROXYBUTANE-1,1-DIPHOSPHONIC ACID, THEIR WATER-SOLUBLE SALTS, PROCESS FOR THEIR PRODUCTION AND THEIR USE
DE3623397A1 (en) * 1986-07-11 1988-01-14 Boehringer Mannheim Gmbh NEW DIPHOSPHONIC ACID DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS

Also Published As

Publication number Publication date
PT100624B (en) 1999-07-30
IT1247034B (en) 1994-12-12
AU2150792A (en) 1993-01-25
ITFI910160A1 (en) 1992-12-26
CA2112250A1 (en) 1993-01-07
EP0592488A1 (en) 1994-04-20
ITFI910160A0 (en) 1991-06-26
JPH06508833A (en) 1994-10-06
PT100624A (en) 1993-10-29
WO1993000348A1 (en) 1993-01-07

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