IT1247034B - DIMETHYLAMINE-HYDROXY ACIDS DIPHOSPHONICS AND THEIR SALTS, THEIR PRODUCTION PROCESS AND PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEM - Google Patents
DIMETHYLAMINE-HYDROXY ACIDS DIPHOSPHONICS AND THEIR SALTS, THEIR PRODUCTION PROCESS AND PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEMInfo
- Publication number
- IT1247034B IT1247034B ITFI910160A ITFI910160A IT1247034B IT 1247034 B IT1247034 B IT 1247034B IT FI910160 A ITFI910160 A IT FI910160A IT FI910160 A ITFI910160 A IT FI910160A IT 1247034 B IT1247034 B IT 1247034B
- Authority
- IT
- Italy
- Prior art keywords
- production process
- diphosphonics
- dimethylamine
- salts
- pharmaceutical compositions
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids, i.e. RP(=X)(XH)2 (X = S, Se)
- C07F9/3804—Phosphonic acids RP(=O)(OH)2; Thiophosphonic acids, i.e. RP(=X)(XH)2 (X = S, Se) not used, see subgroups
- C07F9/3839—Polyphosphonic acids
- C07F9/3873—Polyphosphonic acids containing nitrogen substituent, e.g. N.....H or N-hydrocarbon group which can be substituted by halogen or nitro(so), N.....O, N.....S, N.....C(=X)- (X =O, S), N.....N, N...C(=X)...N (X =O, S)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
Acidi dimetilamino 1-idrossi-alcan-1,1-difosfonici di formula: (FORMULA) in cui n= 4, 5, e loro procedimento produttivo.Dimethylamino 1-hydroxy-alkan-1,1-diphosphonic acids of formula: (FORMULA) wherein n = 4, 5, and their production process.
Priority Applications (8)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ITFI910160A IT1247034B (en) | 1991-06-26 | 1991-06-26 | DIMETHYLAMINE-HYDROXY ACIDS DIPHOSPHONICS AND THEIR SALTS, THEIR PRODUCTION PROCESS AND PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEM |
AU21507/92A AU2150792A (en) | 1991-06-26 | 1992-05-27 | Dimethylamino-hydroxy-alkan diphosphonic acids and pharmaceutical compositions containing them |
EP92913148A EP0592488A1 (en) | 1991-06-26 | 1992-05-27 | Dimethylamino-hydroxy-alkan diphosphonic acids and pharmaceutical compositions containing them |
CA002112250A CA2112250A1 (en) | 1991-06-26 | 1992-05-27 | Dimethylamino-hydroxy-alkan diphosphonic acids and pharmaceutical compositions containing them |
JP5501416A JPH06508833A (en) | 1991-06-26 | 1992-05-27 | Dimethylamino-hydroxy-alkanediphosphonic acids and pharmaceutical compositions containing them |
PCT/IT1992/000058 WO1993000348A1 (en) | 1991-06-26 | 1992-05-27 | Dimethylamino-hydroxy-alkan diphosphonic acids and pharmaceutical compositions containing them |
MX9203205A MX9203205A (en) | 1991-06-26 | 1992-06-24 | NOVELTY DIMETILAMINO-HIDROXI-ALCAN-DIPHOSPHONIC ACIDS AND SALTS OF THE SAME, IN PRODUCTION PROCEDURE AND RELATED PHARMACEUTICAL COMPOSITIONS. |
PT100624A PT100624B (en) | 1991-06-26 | 1992-06-25 | NEW DIMETHYLAMINO-HYDROXY-ACANO-DIPHOSPHONIC ACIDS AND ITS SALTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ITFI910160A IT1247034B (en) | 1991-06-26 | 1991-06-26 | DIMETHYLAMINE-HYDROXY ACIDS DIPHOSPHONICS AND THEIR SALTS, THEIR PRODUCTION PROCESS AND PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEM |
Publications (3)
Publication Number | Publication Date |
---|---|
ITFI910160A0 ITFI910160A0 (en) | 1991-06-26 |
ITFI910160A1 ITFI910160A1 (en) | 1992-12-26 |
IT1247034B true IT1247034B (en) | 1994-12-12 |
Family
ID=11349724
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ITFI910160A IT1247034B (en) | 1991-06-26 | 1991-06-26 | DIMETHYLAMINE-HYDROXY ACIDS DIPHOSPHONICS AND THEIR SALTS, THEIR PRODUCTION PROCESS AND PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEM |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP0592488A1 (en) |
JP (1) | JPH06508833A (en) |
AU (1) | AU2150792A (en) |
CA (1) | CA2112250A1 (en) |
IT (1) | IT1247034B (en) |
MX (1) | MX9203205A (en) |
PT (1) | PT100624B (en) |
WO (1) | WO1993000348A1 (en) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1303672B1 (en) | 1998-07-28 | 2001-02-23 | Nicox Sa | NITRATED SALTS OF DRUGS ACTIVE IN BONE DISORDERS |
ES2336312T3 (en) * | 2001-07-16 | 2010-04-12 | Universite Paris 13 | PROCEDURE FOR PREPARATION OF BISPHOSPHONATE DERIVATIVES. |
DE102014115154A1 (en) * | 2014-10-17 | 2016-04-21 | SCV-SpezialChemikalien-Vertrieb GmbH | Conjugated bisphosphonates for the diagnosis and treatment of bone diseases |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1194748B (en) * | 1981-02-12 | 1988-09-28 | Gentili Ist Spa | PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF OSTEOPATHIES |
IT1201087B (en) * | 1982-04-15 | 1989-01-27 | Gentili Ist Spa | PHARMACOLOGICALLY ACTIVE BIPPHOSPHONES, PROCEDURE FOR THEIR PREPARATION AND RELATED PHARMACEUTICAL COMPOSITIONS |
DE3434667A1 (en) * | 1984-09-21 | 1986-04-03 | Henkel KGaA, 4000 Düsseldorf | 4-DIMETHYLAMINO-1-HYDROXYBUTANE-1,1-DIPHOSPHONIC ACID, THEIR WATER-SOLUBLE SALTS, PROCESS FOR THEIR PRODUCTION AND THEIR USE |
DE3623397A1 (en) * | 1986-07-11 | 1988-01-14 | Boehringer Mannheim Gmbh | NEW DIPHOSPHONIC ACID DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS |
-
1991
- 1991-06-26 IT ITFI910160A patent/IT1247034B/en active IP Right Grant
-
1992
- 1992-05-27 AU AU21507/92A patent/AU2150792A/en not_active Abandoned
- 1992-05-27 CA CA002112250A patent/CA2112250A1/en not_active Abandoned
- 1992-05-27 EP EP92913148A patent/EP0592488A1/en not_active Withdrawn
- 1992-05-27 WO PCT/IT1992/000058 patent/WO1993000348A1/en not_active Application Discontinuation
- 1992-05-27 JP JP5501416A patent/JPH06508833A/en active Pending
- 1992-06-24 MX MX9203205A patent/MX9203205A/en unknown
- 1992-06-25 PT PT100624A patent/PT100624B/en not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
CA2112250A1 (en) | 1993-01-07 |
MX9203205A (en) | 1994-06-30 |
PT100624B (en) | 1999-07-30 |
AU2150792A (en) | 1993-01-25 |
WO1993000348A1 (en) | 1993-01-07 |
ITFI910160A1 (en) | 1992-12-26 |
EP0592488A1 (en) | 1994-04-20 |
ITFI910160A0 (en) | 1991-06-26 |
JPH06508833A (en) | 1994-10-06 |
PT100624A (en) | 1993-10-29 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
0001 | Granted | ||
TA | Fee payment date (situation as of event date), data collected since 19931001 |
Effective date: 19950622 |