MX368424B - Enaminocetonas que contienen cf3o y su uso para la preparacion de pirazoles que contienen cf3o. - Google Patents
Enaminocetonas que contienen cf3o y su uso para la preparacion de pirazoles que contienen cf3o.Info
- Publication number
- MX368424B MX368424B MX2014009442A MX2014009442A MX368424B MX 368424 B MX368424 B MX 368424B MX 2014009442 A MX2014009442 A MX 2014009442A MX 2014009442 A MX2014009442 A MX 2014009442A MX 368424 B MX368424 B MX 368424B
- Authority
- MX
- Mexico
- Prior art keywords
- cf3o
- enaminoketones
- preparation
- pyrazoles
- utilization
- Prior art date
Links
- 125000000876 trifluoromethoxy group Chemical group FC(F)(F)O* 0.000 title abstract 3
- 150000003217 pyrazoles Chemical class 0.000 title 1
- VEXXKRRZTWOPFP-UHFFFAOYSA-N 5-(trifluoromethoxy)-1h-pyrazole Chemical class FC(F)(F)OC1=CC=NN1 VEXXKRRZTWOPFP-UHFFFAOYSA-N 0.000 abstract 1
- 150000002429 hydrazines Chemical class 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 238000007363 ring formation reaction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C221/00—Preparation of compounds containing amino groups and doubly-bound oxygen atoms bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C225/00—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones
- C07C225/02—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton
- C07C225/14—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated
- C07C225/16—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Furan Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
La presente invención se refiere a nuevas enaminocetonas que contienen un grupo CF3O, a nuevos derivados de pirazol que contienen un grupo CF3O, así como a un nuevo procedimiento para su preparación que comprende aminoformilacion de CF3O-cetonas y ciclación de las CF3O-enaminocetonas obtenidas con hidrazinas para dar trifluorometoxi pirazoles.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP12356003.9A EP2628722A1 (en) | 2012-02-16 | 2012-02-16 | CF3O-containing enaminoketones and their utilization for the preparation of CF3O-containing pyrazoles |
| PCT/EP2013/052829 WO2013120876A1 (en) | 2012-02-16 | 2013-02-13 | CF3O-containing enaminoketones and their utilization for the preparation of CF3O-containing pyrazoles |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MX2014009442A MX2014009442A (es) | 2014-11-12 |
| MX368424B true MX368424B (es) | 2019-10-02 |
Family
ID=47716032
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2014009442A MX368424B (es) | 2012-02-16 | 2013-02-13 | Enaminocetonas que contienen cf3o y su uso para la preparacion de pirazoles que contienen cf3o. |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US9096535B2 (es) |
| EP (2) | EP2628722A1 (es) |
| JP (2) | JP6212056B2 (es) |
| KR (1) | KR102085012B1 (es) |
| CN (1) | CN104220419B (es) |
| BR (1) | BR112014019346B1 (es) |
| DK (1) | DK2822925T3 (es) |
| ES (1) | ES2701082T3 (es) |
| IL (1) | IL233625A (es) |
| MX (1) | MX368424B (es) |
| TW (1) | TWI597261B (es) |
| WO (1) | WO2013120876A1 (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2663614T3 (es) | 2014-03-24 | 2018-04-16 | Bayer Cropscience Aktiengesellschaft | Procedimiento de preparación de derivados de 3,5-bis(haloalquil)pirazol a partir de alfa, alfa-dihaloaminas y cetiminas |
| EP3015458A1 (en) * | 2014-11-03 | 2016-05-04 | Bayer CropScience AG | Process for preparing 3,5-bis(haloalkyl)pyrazole derivatives from a,a-dihaloamines and ketimines |
| EP3313820A1 (en) * | 2015-06-26 | 2018-05-02 | Bayer CropScience Aktiengesellschaft | Process for preparing substituted pyrazoles containing haloalkoxy- and haloalkylthio groups from , -dihaloalkylamines and ketimines |
| US20200039920A1 (en) * | 2016-10-19 | 2020-02-06 | AGC Inc. | Method for producing nitrogen-containing compound |
| IL277978B2 (en) | 2018-04-25 | 2024-07-01 | Bayer Ag | Novel heteroaryl-triazole and heteroaryl-tetrazole compounds as pesticides |
| EP4495125A1 (en) * | 2023-07-19 | 2025-01-22 | Freie Universität Berlin | A catalyst free synthesis method for introducing a trifluoromethoxy moiety into at least one organic compound |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2743473B2 (ja) * | 1988-07-04 | 1998-04-22 | 日産化学工業株式会社 | ピラゾールカルボン酸類の製造方法 |
| FR2682379B1 (fr) * | 1991-10-09 | 1994-02-11 | Rhone Poulenc Agrochimie | Nouveaux phenylpyrazoles fongicides. |
| FR2707295A1 (fr) * | 1993-06-07 | 1995-01-13 | Rhone Poulenc Agrochimie | Fongicides pyrazoles substitués en position 3 par un hétérocycle. |
| JPH09169736A (ja) * | 1995-12-21 | 1997-06-30 | Nissan Chem Ind Ltd | ピラゾール誘導体及び有害生物防除剤 |
| JP2008513426A (ja) * | 2004-09-20 | 2008-05-01 | バイオリポックス エービー | 炎症の治療に有用なピラゾール化合物 |
| DE102006050516A1 (de) * | 2006-10-26 | 2008-04-30 | Bayer Healthcare Ag | Substituierte Dihydropyrazolone und ihre Verwendung |
| WO2009001126A1 (en) | 2007-06-27 | 2008-12-31 | Astrazeneca Ab | Substituted piperidine derivatives and their use as antibaterial agents |
| DE102007036702A1 (de) * | 2007-08-03 | 2009-02-05 | Bayer Cropscience Ag | Synergistische kulturpflanzenverträgliche herbizide Kombinationen enthaltend Herbizide aus der Gruppe der Pyrazolyloxyphenyl-Derivate |
| JP2011520897A (ja) * | 2008-05-16 | 2011-07-21 | シェーリング コーポレイション | グルカゴン受容体アンタゴニスト、組成物およびそれらの使用方法 |
| DE102008024221A1 (de) | 2008-05-19 | 2009-11-26 | Merck Patent Gmbh | Herstellung von CF3O-Gruppen enthaltenden Verbindungen |
-
2012
- 2012-02-16 EP EP12356003.9A patent/EP2628722A1/en not_active Withdrawn
-
2013
- 2013-02-07 TW TW102104714A patent/TWI597261B/zh not_active IP Right Cessation
- 2013-02-13 JP JP2014557016A patent/JP6212056B2/ja not_active Expired - Fee Related
- 2013-02-13 WO PCT/EP2013/052829 patent/WO2013120876A1/en not_active Ceased
- 2013-02-13 MX MX2014009442A patent/MX368424B/es active IP Right Grant
- 2013-02-13 EP EP13704421.0A patent/EP2822925B1/en not_active Not-in-force
- 2013-02-13 DK DK13704421.0T patent/DK2822925T3/en active
- 2013-02-13 ES ES13704421T patent/ES2701082T3/es active Active
- 2013-02-13 BR BR112014019346-0A patent/BR112014019346B1/pt not_active IP Right Cessation
- 2013-02-13 CN CN201380009409.3A patent/CN104220419B/zh not_active Expired - Fee Related
- 2013-02-13 KR KR1020147024063A patent/KR102085012B1/ko not_active Expired - Fee Related
- 2013-02-13 US US14/378,372 patent/US9096535B2/en not_active Expired - Fee Related
-
2014
- 2014-07-13 IL IL233625A patent/IL233625A/en active IP Right Grant
-
2017
- 2017-05-30 JP JP2017106304A patent/JP2018008928A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| US20150018561A1 (en) | 2015-01-15 |
| MX2014009442A (es) | 2014-11-12 |
| EP2628722A1 (en) | 2013-08-21 |
| CN104220419B (zh) | 2017-03-29 |
| EP2822925B1 (en) | 2018-09-05 |
| US9096535B2 (en) | 2015-08-04 |
| JP2015511944A (ja) | 2015-04-23 |
| ES2701082T3 (es) | 2019-02-20 |
| IL233625A (en) | 2017-10-31 |
| JP6212056B2 (ja) | 2017-10-11 |
| BR112014019346A2 (es) | 2017-06-20 |
| KR102085012B1 (ko) | 2020-03-05 |
| CN104220419A (zh) | 2014-12-17 |
| TW201336810A (zh) | 2013-09-16 |
| BR112014019346A8 (pt) | 2017-07-11 |
| EP2822925A1 (en) | 2015-01-14 |
| WO2013120876A1 (en) | 2013-08-22 |
| TWI597261B (zh) | 2017-09-01 |
| JP2018008928A (ja) | 2018-01-18 |
| KR20150002596A (ko) | 2015-01-07 |
| BR112014019346B1 (pt) | 2020-09-15 |
| IL233625A0 (en) | 2014-08-31 |
| DK2822925T3 (en) | 2019-01-07 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant or registration |