MX366118B - Combinacion sinergistica de paracetamol/celecoxib para el tratamiento de dolor inflamatorio. - Google Patents

Combinacion sinergistica de paracetamol/celecoxib para el tratamiento de dolor inflamatorio.

Info

Publication number
MX366118B
MX366118B MX2015013911A MX2015013911A MX366118B MX 366118 B MX366118 B MX 366118B MX 2015013911 A MX2015013911 A MX 2015013911A MX 2015013911 A MX2015013911 A MX 2015013911A MX 366118 B MX366118 B MX 366118B
Authority
MX
Mexico
Prior art keywords
paracetamol
celecoxib
treatment
inflammatory pain
synergistic combination
Prior art date
Application number
MX2015013911A
Other languages
English (en)
Other versions
MX2015013911A (es
Inventor
Fernando Cantú Medellin Jorge
Original Assignee
More Pharma Corp S De R L De C V
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52279400&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX366118(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by More Pharma Corp S De R L De C V filed Critical More Pharma Corp S De R L De C V
Publication of MX2015013911A publication Critical patent/MX2015013911A/es
Publication of MX366118B publication Critical patent/MX366118B/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/63Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • A61K31/635Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Se describe y reclama una combinación de paracetamol y celecoxib que en cantidades específicas generan una potenciación analgésica contra el dolor de tipo inflamatorio. Específicamente, la invención se refiere una combinación sinergística de entre 375 a 500 mg de paracetamol y de entre 50 a 100 mg de celecoxib útil para el tratamiento de dolor inflamatorio en animales y seres humanos, así como el uso de dichos principios activos en las cantidades indicadas en la preparación de combinaciones farmacéuticas sinérgicas.
MX2015013911A 2013-07-11 2014-07-11 Combinacion sinergistica de paracetamol/celecoxib para el tratamiento de dolor inflamatorio. MX366118B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/IB2013/055710 WO2015004505A1 (es) 2013-07-11 2013-07-11 Combinación sinergística de paracetamol/celecoxib para el tratamiento de dolor inflamatorio
PCT/IB2014/063019 WO2015004634A2 (es) 2013-07-11 2014-07-11 Combinación sinergística de paracetamol/celecoxib para el tratamiento de dolor inflamatorio

Publications (2)

Publication Number Publication Date
MX2015013911A MX2015013911A (es) 2015-12-08
MX366118B true MX366118B (es) 2019-06-27

Family

ID=52279400

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2015013911A MX366118B (es) 2013-07-11 2014-07-11 Combinacion sinergistica de paracetamol/celecoxib para el tratamiento de dolor inflamatorio.

Country Status (8)

Country Link
CL (1) CL2015003211A1 (es)
CR (1) CR20160021A (es)
CU (1) CU24440B1 (es)
DO (1) DOP2016000008A (es)
EC (1) ECSP16005679A (es)
MX (1) MX366118B (es)
PE (2) PE20160239A1 (es)
WO (2) WO2015004505A1 (es)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4534077A1 (en) 2023-10-05 2025-04-09 Laboratorios Silanes, S.A. de C.V. Composition comprising cyanocobalamin, pyridoxine, thiamine, pregabalin and celecoxib
EP4534076A1 (en) 2023-10-05 2025-04-09 Laboratorios Silanes, S.A. de C.V. Celecoxib - acetaminophen combination of improved stability and procedure for the preparation thereof

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11147780B2 (en) * 2020-02-24 2021-10-19 Algia Pharma, Llc Multidrug pain management package

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL163637A0 (en) * 2002-02-19 2005-12-18 Adcock Ingram Ltd Pharmaceutical combinations of cox-2 inhibitors and opiates
GB0423103D0 (en) * 2004-10-19 2004-11-17 Boots Healthcare Int Ltd Therapeutic agents

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4534077A1 (en) 2023-10-05 2025-04-09 Laboratorios Silanes, S.A. de C.V. Composition comprising cyanocobalamin, pyridoxine, thiamine, pregabalin and celecoxib
EP4534076A1 (en) 2023-10-05 2025-04-09 Laboratorios Silanes, S.A. de C.V. Celecoxib - acetaminophen combination of improved stability and procedure for the preparation thereof

Also Published As

Publication number Publication date
CU24440B1 (es) 2019-09-04
CU20160002A7 (es) 2016-06-29
CR20160021A (es) 2016-04-08
DOP2016000008A (es) 2016-03-15
WO2015004505A1 (es) 2015-01-15
ECSP16005679A (es) 2017-08-31
WO2015004634A2 (es) 2015-01-15
PE20170305A1 (es) 2017-04-21
CL2015003211A1 (es) 2016-04-29
WO2015004634A3 (es) 2015-04-09
PE20160239A1 (es) 2016-05-13
MX2015013911A (es) 2015-12-08

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