MX340272B - Composicion sinergica de nitazoxanida y mebendazol, procesos para prepararla y el uso de dicha composicion para el tratamiento de la parasitosis humana. - Google Patents
Composicion sinergica de nitazoxanida y mebendazol, procesos para prepararla y el uso de dicha composicion para el tratamiento de la parasitosis humana.Info
- Publication number
- MX340272B MX340272B MX2015003941A MX2015003941A MX340272B MX 340272 B MX340272 B MX 340272B MX 2015003941 A MX2015003941 A MX 2015003941A MX 2015003941 A MX2015003941 A MX 2015003941A MX 340272 B MX340272 B MX 340272B
- Authority
- MX
- Mexico
- Prior art keywords
- ntzx
- mbdz
- synergic
- composition
- treatment
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/04—Amoebicides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
La presente invención se refiere a una composición farmacéutica sinérgica para el tratamiento de parasitosis humana de Mebendazol (MBDZ) con Nitazoxanida (NTZX), que amplía significativamente el espectro del MBDZ contra protozoos y refuerza la acción antihelmíntica de la NTZX. Además, al usar dicha combinación farmacéutica de MBDZ y NTZX, la acción sistémica del metabolito activo de la NTZX, la Tizoxanida, y el tratamiento de algunas formas sistémicas de parasitosis, mantienen los mismos efectos de los principios activos individuales. También, la combinación farmacéutica sinérgica de MBDZ con NTZX logra un mayor espectro antiparasitario, mientras mantienen la eficacia y los perfiles de seguridad de ambos principios activos por separado. Todos estos efectos permiten que la combinación farmacéutica de la presente invención se diferencie del resto de los tratamientos antiparasitarios clásicos que tienen espectros más acotados. Los efectos sinérgicos de la combinación farmacéutica MBDZ y NTZX son, por consiguiente, el objeto principal de la presente invención.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/IB2012/055166 WO2014049397A1 (es) | 2012-09-27 | 2012-09-27 | Composición sinérgica de nitazoxanida y mebendazol, procesos para prepararla y el uso de dicha composición para el tratamiento de la parasitosis humana |
Publications (2)
Publication Number | Publication Date |
---|---|
MX2015003941A MX2015003941A (es) | 2015-07-21 |
MX340272B true MX340272B (es) | 2016-06-30 |
Family
ID=50387067
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2015003941A MX340272B (es) | 2012-09-27 | 2012-09-27 | Composicion sinergica de nitazoxanida y mebendazol, procesos para prepararla y el uso de dicha composicion para el tratamiento de la parasitosis humana. |
Country Status (10)
Country | Link |
---|---|
US (1) | US20150250765A1 (es) |
EP (1) | EP2902024B1 (es) |
AR (1) | AR092169A1 (es) |
BR (1) | BR112015006861B1 (es) |
CL (1) | CL2015000778A1 (es) |
CR (1) | CR20150190A (es) |
MX (1) | MX340272B (es) |
NI (1) | NI201500045A (es) |
UY (1) | UY34967A (es) |
WO (1) | WO2014049397A1 (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2610791B1 (es) * | 2016-12-22 | 2018-02-07 | Elena TEIJEIRA PRIETO | Uso del mebendazol para la eliminación de los gusanos de fuego en acuarios de arrecife |
CN111494327B (zh) * | 2020-06-23 | 2023-09-05 | 瑞阳制药股份有限公司 | 甲苯咪唑咀嚼片的制备方法 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3657267A (en) | 1969-06-20 | 1972-04-18 | Janssen Pharmaceutica Nv | Benzimidazole carbamates |
GB1437800A (en) | 1973-08-08 | 1976-06-03 | Phavic Sprl | Derivatives of 2-benzamido-5-nitro-thiazoles |
US5387598A (en) | 1994-04-13 | 1995-02-07 | Rossignol; Jean-Francois | Composition and galenic formulation suitable for combatting affections of the lower abdomen |
US20050171169A1 (en) * | 2004-02-02 | 2005-08-04 | Rossignol Jean F. | Combination chemotherapy for helminth infections |
US8158152B2 (en) * | 2005-11-18 | 2012-04-17 | Scidose Llc | Lyophilization process and products obtained thereby |
-
2012
- 2012-09-27 EP EP12885371.0A patent/EP2902024B1/en active Active
- 2012-09-27 MX MX2015003941A patent/MX340272B/es active IP Right Grant
- 2012-09-27 BR BR112015006861-8A patent/BR112015006861B1/pt active IP Right Grant
- 2012-09-27 WO PCT/IB2012/055166 patent/WO2014049397A1/es active Application Filing
- 2012-09-27 US US14/431,623 patent/US20150250765A1/en not_active Abandoned
-
2013
- 2013-08-06 UY UY0001034967A patent/UY34967A/es unknown
- 2013-08-16 AR ARP130102935A patent/AR092169A1/es unknown
-
2015
- 2015-03-26 NI NI201500045A patent/NI201500045A/es unknown
- 2015-03-27 CL CL2015000778A patent/CL2015000778A1/es unknown
- 2015-04-13 CR CR20150190A patent/CR20150190A/es unknown
Also Published As
Publication number | Publication date |
---|---|
EP2902024A1 (en) | 2015-08-05 |
BR112015006861B1 (pt) | 2021-10-13 |
MX2015003941A (es) | 2015-07-21 |
CL2015000778A1 (es) | 2015-08-21 |
BR112015006861A2 (pt) | 2017-07-04 |
EP2902024A4 (en) | 2016-06-22 |
CR20150190A (es) | 2015-07-09 |
EP2902024B1 (en) | 2017-11-29 |
WO2014049397A1 (es) | 2014-04-03 |
UY34967A (es) | 2014-04-30 |
AR092169A1 (es) | 2015-03-25 |
US20150250765A1 (en) | 2015-09-10 |
NI201500045A (es) | 2016-02-16 |
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Legal Events
Date | Code | Title | Description |
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FG | Grant or registration |